Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252827 (CHEMBL493688 | N-Cyclohexylethyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 450 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252827 (CHEMBL493688 | N-Cyclohexylethyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 630 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339567 ((2S,5S,8S,11S)-11-(2-carboxyethyl)-14-cyclohexyl-8...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 630 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339545 ((4S,7S,10S,13S)-4-(2-carboxyethyl)-10-(carboxymeth...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 750 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252827 (CHEMBL493688 | N-Cyclohexylethyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 940 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252828 (CHEMBL493689 | N-(Naphthalene-2-yl)ethyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 950 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252754 (CHEMBL538410 | N-(3,4-Difluorophenyl)propyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 980 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252828 (CHEMBL493689 | N-(Naphthalene-2-yl)ethyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339569 ((2S,5S,8S,11S)-11-(2-carboxyethyl)-14-(3,4-dichlor...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252754 (CHEMBL538410 | N-(3,4-Difluorophenyl)propyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252826 (CHEMBL494486 | N-Cyclohexylmethyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339568 ((2S,5S,8S,11S)-11-(2-carboxyethyl)-8-((R)-1-hydrox...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252753 (CHEMBL495100 | N-(3,4-Dichlorophenyl)propyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339548 ((2S,5S,8S,11S)-11-(2-carboxyethyl)-5-(carboxymethy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339555 ((2S,5S,8S,11S)-11-(2-carboxyethyl)-14-cycloheptyl-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339552 ((3S,6S,9S,12S)-1-(bicyclo[2.2.1]heptan-2-yl)-3-(2-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252826 (CHEMBL494486 | N-Cyclohexylmethyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339554 ((3S,6S,9S,12S)-3-(2-carboxyethyl)-1-cycloheptyl-6-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339553 ((2S,5S,8S,11S)-14-(bicyclo[2.2.1]heptan-2-yl)-11-(...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252715 (CHEMBL494895 | N-Phenylethyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339556 ((2S,5S,8S,11S)-11-(2-carboxyethyl)-8-((R)-1-hydrox...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339547 ((2S,5S,8S,11S)-11-(2-carboxyethyl)-5-(carboxymethy...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50253144 (CHEMBL505051 | KSG-LDTKNYKQTSV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ3 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252752 (CHEMBL495099 | N-Phenylpropyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339551 ((S)-2-[(S)-2-((2S,3R)-2-{(S)-2-[(Adamantan-1-ylmet...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252713 (CHEMBL492642 | FETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252753 (CHEMBL495100 | N-(3,4-Dichlorophenyl)propyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252752 (CHEMBL495099 | N-Phenylpropyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339539 ((4S,7S,10S,13S)-10-(carboxymethyl)-1-cyclohexyl-7-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252825 (CHEMBL494485 | N-Butyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50253143 (CHEMBL445253 | KSG-YEKLSSIESDV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252824 (CHEMBL494287 | N-Propyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339557 ((2S,5S,8S,11S)-11-(2-carboxyethyl)-8-((R)-1-hydrox...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339546 ((4S,7S,10S,13S)-4-(3-amino-3-oxopropyl)-10-(carbox...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50253145 (CHEMBL502630 | YGRKKRRQRRR-KLSSIESDV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252715 (CHEMBL494895 | N-Phenylethyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50253145 (CHEMBL502630 | YGRKKRRQRRR-KLSSIESDV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339558 ((2S,5S,8S,11S)-11-(2-carboxyethyl)-8-((R)-1-hydrox...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252714 (CHEMBL492643 | N-Benzyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252713 (CHEMBL492642 | FETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252753 (CHEMBL495100 | N-(3,4-Dichlorophenyl)propyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ3 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339551 ((S)-2-[(S)-2-((2S,3R)-2-{(S)-2-[(Adamantan-1-ylmet...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ3 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50253143 (CHEMBL445253 | KSG-YEKLSSIESDV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ1-2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252824 (CHEMBL494287 | N-Propyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252714 (CHEMBL492643 | N-Benzyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252754 (CHEMBL538410 | N-(3,4-Difluorophenyl)propyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ3 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339538 ((4S,7S,10S,13S)-1-cyclohexyl-7-((R)-1-hydroxyethyl...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339569 ((2S,5S,8S,11S)-11-(2-carboxyethyl)-14-(3,4-dichlor...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ3 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50252825 (CHEMBL494485 | N-Butyl-ETAV) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assay | J Med Chem 51: 6450-9 (2008) Article DOI: 10.1021/jm800836w BindingDB Entry DOI: 10.7270/Q22807FQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Disks large homolog 4 (Homo sapiens (Human)) | BDBM50339556 ((2S,5S,8S,11S)-11-(2-carboxyethyl)-8-((R)-1-hydrox...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Inhibition of PSD-95 PDZ3 domain by competitive fluorescence polarization assay | J Med Chem 54: 1333-46 (2011) Article DOI: 10.1021/jm1013924 BindingDB Entry DOI: 10.7270/Q2H13300 | |||||||||||
More data for this Ligand-Target Pair |
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