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Compile Data Set for Download or QSAR

Found 5 hits of kd for UniProtKB: P34947   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
G protein-coupled receptor kinase 5


(Homo sapiens (Human))
BDBM50554263
PNG
(CHEMBL4740635)
Show SMILES O=c1n(Cc2ccccc2)cnc2ccc(cc12)-c1cn[nH]c1
PDB

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PC cid
PC sid
PDB
UniChem
Article
PubMed
n/an/an/a 3.43E+4n/an/an/an/an/a


TBA

Assay Description
Binding affinity to GRK5 (unknown origin) by Thermofluor thermal shift assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2020.127602
BindingDB Entry DOI: 10.7270/Q2H135PS
More data for this
Ligand-Target Pair
G protein-coupled receptor kinase 5


(Homo sapiens (Human))
BDBM50554260
PNG
(CHEMBL4776422)
Show SMILES O=c1n(Cc2ccccc2)cnc2ccc(cc12)-c1cncnc1
PDB

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UniChem
Article
PubMed
n/an/an/a>8.33E+4n/an/an/an/an/a


TBA

Assay Description
Binding affinity to GRK5 (unknown origin) by Thermofluor thermal shift assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2020.127602
BindingDB Entry DOI: 10.7270/Q2H135PS
More data for this
Ligand-Target Pair
G protein-coupled receptor kinase 5


(Homo sapiens (Human))
BDBM50554262
PNG
(CHEMBL4791786)
Show SMILES O=c1n(Cc2ccccc2)cnc2ccc(cc12)-c1ccn[nH]1
PDB

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UniProtKB/SwissProt

antibodypedia
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PC cid
PC sid
UniChem
Article
PubMed
n/an/an/a>8.33E+4n/an/an/an/an/a


TBA

Assay Description
Binding affinity to GRK5 (unknown origin) by Thermofluor thermal shift assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2020.127602
BindingDB Entry DOI: 10.7270/Q2H135PS
More data for this
Ligand-Target Pair
G protein-coupled receptor kinase 5


(Homo sapiens (Human))
BDBM50554259
PNG
(CHEMBL4788026)
Show SMILES O=c1n(Cc2ccccc2)cnc2cc(ccc12)-c1cn[nH]c1
PDB

NCI pathway
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KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
PDB
UniChem
Article
PubMed
n/an/an/a>8.33E+4n/an/an/an/an/a


TBA

Assay Description
Binding affinity to GRK5 (unknown origin) by Thermofluor thermal shift assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2020.127602
BindingDB Entry DOI: 10.7270/Q2H135PS
More data for this
Ligand-Target Pair
G protein-coupled receptor kinase 5


(Homo sapiens (Human))
BDBM50554261
PNG
(CHEMBL4742242)
Show SMILES O=c1n(Cc2ccccc2)cnc2ccc(cc12)-c1ccncc1
PDB

NCI pathway
Reactome pathway
KEGG

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/a>8.33E+4n/an/an/an/an/a


TBA

Assay Description
Binding affinity to GRK5 (unknown origin) by Thermofluor thermal shift assay


Citation and Details

Article DOI: 10.1016/j.bmcl.2020.127602
BindingDB Entry DOI: 10.7270/Q2H135PS
More data for this
Ligand-Target Pair