Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Beta-galactoside alpha-2,6-sialyltransferase 1 (Homo sapiens (Human)) | BDBM50565994 (CHEMBL3596261) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human alpha-2,6-ST6GAL1 assessed as reduction in sialylated-product formation using Gal-beta1-4GlcNac and CMP-NeuSAc incubated for 15 m... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01477 BindingDB Entry DOI: 10.7270/Q2T43XVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-galactoside alpha-2,6-sialyltransferase 1 (Homo sapiens (Human)) | BDBM50565990 (CHEMBL4780118) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human alpha-2,6-ST6GAL1 assessed as reduction in sialylated-product formation using Gal-beta1-4GlcNac and CMP-NeuSAc incubated for 15 m... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01477 BindingDB Entry DOI: 10.7270/Q2T43XVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-galactoside alpha-2,6-sialyltransferase 1 (Homo sapiens (Human)) | BDBM50565988 (CHEMBL4785533) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human alpha-2,6-ST6GAL1 assessed as reduction in sialylated-product formation using Gal-beta1-4GlcNac and CMP-NeuSAc incubated for 15 m... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01477 BindingDB Entry DOI: 10.7270/Q2T43XVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-galactoside alpha-2,6-sialyltransferase 1 (Homo sapiens (Human)) | BDBM50565989 (CHEMBL4798770) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.33E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human alpha-2,6-ST6GAL1 assessed as reduction in sialylated-product formation using Gal-beta1-4GlcNac and CMP-NeuSAc incubated for 15 m... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01477 BindingDB Entry DOI: 10.7270/Q2T43XVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-galactoside alpha-2,6-sialyltransferase 1 (Homo sapiens (Human)) | BDBM50566002 (CHEMBL4776137) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human alpha-2,6-ST6GAL1 assessed as reduction in sialylated-product formation using Gal-beta1-4GlcNac and CMP-NeuSAc incubated for 15 m... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01477 BindingDB Entry DOI: 10.7270/Q2T43XVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-galactoside alpha-2,6-sialyltransferase 1 (Homo sapiens (Human)) | BDBM50565991 (CHEMBL4785375) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human alpha-2,6-ST6GAL1 assessed as reduction in sialylated-product formation using Gal-beta1-4GlcNac and CMP-NeuSAc incubated for 15 m... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01477 BindingDB Entry DOI: 10.7270/Q2T43XVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-galactoside alpha-2,6-sialyltransferase 1 (Homo sapiens (Human)) | BDBM50565992 (CHEMBL4795609) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human alpha-2,6-ST6GAL1 assessed as reduction in sialylated-product formation using Gal-beta1-4GlcNac and CMP-NeuSAc incubated for 15 m... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01477 BindingDB Entry DOI: 10.7270/Q2T43XVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-galactoside alpha-2,6-sialyltransferase 1 (Homo sapiens (Human)) | BDBM50566003 (CHEMBL4793980) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human alpha-2,6-ST6GAL1 assessed as reduction in sialylated-product formation using Gal-beta1-4GlcNac and CMP-NeuSAc incubated for 15 m... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01477 BindingDB Entry DOI: 10.7270/Q2T43XVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-galactoside alpha-2,6-sialyltransferase 1 (Homo sapiens (Human)) | BDBM50566001 (CHEMBL4797927) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human alpha-2,6-ST6GAL1 assessed as reduction in sialylated-product formation using Gal-beta1-4GlcNac and CMP-NeuSAc incubated for 15 m... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01477 BindingDB Entry DOI: 10.7270/Q2T43XVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-galactoside alpha-2,6-sialyltransferase 1 (Homo sapiens (Human)) | BDBM50565997 (CHEMBL4793269) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human alpha-2,6-ST6GAL1 assessed as reduction in sialylated-product formation using Gal-beta1-4GlcNac and CMP-NeuSAc incubated for 15 m... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01477 BindingDB Entry DOI: 10.7270/Q2T43XVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-galactoside alpha-2,6-sialyltransferase 1 (Homo sapiens (Human)) | BDBM50566000 (CHEMBL4800187) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human alpha-2,6-ST6GAL1 assessed as reduction in sialylated-product formation using Gal-beta1-4GlcNac and CMP-NeuSAc incubated for 15 m... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01477 BindingDB Entry DOI: 10.7270/Q2T43XVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-galactoside alpha-2,6-sialyltransferase 1 (Homo sapiens (Human)) | BDBM50565998 (CHEMBL4786588) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human alpha-2,6-ST6GAL1 assessed as reduction in sialylated-product formation using Gal-beta1-4GlcNac and CMP-NeuSAc incubated for 15 m... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01477 BindingDB Entry DOI: 10.7270/Q2T43XVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-galactoside alpha-2,6-sialyltransferase 1 (Homo sapiens (Human)) | BDBM50566004 (CHEMBL4777310) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human alpha-2,6-ST6GAL1 assessed as reduction in sialylated-product formation using Gal-beta1-4GlcNac and CMP-NeuSAc incubated for 15 m... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01477 BindingDB Entry DOI: 10.7270/Q2T43XVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-galactoside alpha-2,6-sialyltransferase 1 (Homo sapiens (Human)) | BDBM50565996 (CHEMBL4781666) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human alpha-2,6-ST6GAL1 assessed as reduction in sialylated-product formation using Gal-beta1-4GlcNac and CMP-NeuSAc incubated for 15 m... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01477 BindingDB Entry DOI: 10.7270/Q2T43XVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-galactoside alpha-2,6-sialyltransferase 1 (Homo sapiens (Human)) | BDBM50565995 (CHEMBL4790244) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human alpha-2,6-ST6GAL1 assessed as reduction in sialylated-product formation using Gal-beta1-4GlcNac and CMP-NeuSAc incubated for 15 m... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01477 BindingDB Entry DOI: 10.7270/Q2T43XVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-galactoside alpha-2,6-sialyltransferase 1 (Homo sapiens (Human)) | BDBM50565999 (CHEMBL4779174) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human alpha-2,6-ST6GAL1 assessed as reduction in sialylated-product formation using Gal-beta1-4GlcNac and CMP-NeuSAc incubated for 15 m... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01477 BindingDB Entry DOI: 10.7270/Q2T43XVZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-galactoside alpha-2,6-sialyltransferase 1 (Homo sapiens (Human)) | BDBM50565993 (CHEMBL4797481) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.58E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human alpha-2,6-ST6GAL1 assessed as reduction in sialylated-product formation using Gal-beta1-4GlcNac and CMP-NeuSAc incubated for 15 m... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01477 BindingDB Entry DOI: 10.7270/Q2T43XVZ | |||||||||||
More data for this Ligand-Target Pair |