Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Spike glycoprotein (SARS-CoV) | BDBM50559137 (CHEMBL4785828) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike protein in SARS-CoV infected in human HeLa cells haboring wild type ACE2 assessed as reduction in virus infectivity preincubated ... | Citation and Details Article DOI: 10.1016/j.bmc.2020.115745 BindingDB Entry DOI: 10.7270/Q25X2DM8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50233805 (CHEMBL4077922 | US11021454, Compound Salvianolic a...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.85E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50567444 (CHEMBL4873011) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.37E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50567440 (CHEMBL4847112) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.54E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50567449 (CHEMBL4874301) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.68E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50567447 (CHEMBL4852531) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 5.89E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50567443 (CHEMBL4852791) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.27E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50567450 (CHEMBL4859094) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6.32E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50567453 (CHEMBL4865746) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.37E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50567448 (CHEMBL4875210) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.76E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50567441 (CHEMBL4855702) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.33E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50567451 (CHEMBL4868650) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.57E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50567442 (CHEMBL4865677) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 9.97E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM78433 (2-[4-[3-[2-(trifluoromethyl)-10-phenothiazinyl]pro...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.18E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn | Assay Description This is a review article. | Med Res Rev (2020) Article DOI: 10.1002/med.21724 BindingDB Entry DOI: 10.7270/Q2JS9ST6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50001888 ((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn | Assay Description This is a review article. | Med Res Rev (2020) Article DOI: 10.1002/med.21724 BindingDB Entry DOI: 10.7270/Q2JS9ST6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50567454 (CHEMBL4857727) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.31E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50567455 (CHEMBL3902325) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.68E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50567452 (CHEMBL4852883) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.68E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50567439 (CHEMBL4849021) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.81E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50567446 (CHEMBL4869223) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50567445 (CHEMBL4876819) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ... | Citation and Details Article DOI: 10.1016/j.ejmech.2021.113242 BindingDB Entry DOI: 10.7270/Q27W6GZC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Spike glycoprotein (SARS-CoV) | BDBM50017696 ((2-dimethylamino-2-methyl)ethyl-N-dibenzoparathiaz...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 2.14E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Bonn | Assay Description This is a review article. | Med Res Rev (2020) Article DOI: 10.1002/med.21724 BindingDB Entry DOI: 10.7270/Q2JS9ST6 | |||||||||||
More data for this Ligand-Target Pair |