Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50067880 (4-methoxy-7H-furo[3,2-g][1]benzopyran-7-one | 4-me...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | 1.77E+5 | n/a | n/a | n/a | n/a | n/a |
University of Kiel Curated by ChEMBL | Assay Description Blockade of peak K+ currents against Kv1.5 gene | J Med Chem 41: 4542-9 (1998) Article DOI: 10.1021/jm981032o BindingDB Entry DOI: 10.7270/Q2B56HWK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human)) | BDBM50067878 (9-Methoxy-furo[3',2':4,5]benzo[1,2-b][1,4]oxazin-3...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 2.70E+5 | n/a | n/a | n/a | n/a | n/a |
University of Kiel Curated by ChEMBL | Assay Description Blockade of peak K+ currents against Kv1.5 gene | J Med Chem 41: 4542-9 (1998) Article DOI: 10.1021/jm981032o BindingDB Entry DOI: 10.7270/Q2B56HWK | |||||||||||
More data for this Ligand-Target Pair |