Compile Data Set for Download or QSAR

Found 92 hits Enz. Inhib. hit(s) with all data for entry = 5921   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100728 (US8507676, 78) Show SMILES CC(N=O)c1ccc2nnc(Cc3c(F)cc4ncccc4c3F)n2n1 Show InChI InChI=1S/C17H12F2N6O/c1-9(24-26)13-4-5-15-21-22-16(25(15)23-13)7-11-12(18)8-14-10(17(11)19)3-2-6-20-14/h2-6,8-9H,7H2,1H3	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	0.400	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100726 (US8507676, 77-S) Show SMILES C[C@@H](c1nnc2ccc(nn12)C(C)=NOC(N)=O)c1c(F)cc2ncccc2c1F |r,w:13.15| Show InChI InChI=1S/C19H15F2N7O2/c1-9(16-12(20)8-14-11(17(16)21)4-3-7-23-14)18-25-24-15-6-5-13(26-28(15)18)10(2)27-30-19(22)29/h3-9H,1-2H3,(H2,22,29)/t9-/m1/s1	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	0.480	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100724 (US8507676, 75-S) Show SMILES CC(N=O)c1ccc2nnc([C@@H](C)c3c(F)cc4ncccc4c3F)n2n1 |r| Show InChI InChI=1S/C18H14F2N6O/c1-9(16-12(19)8-14-11(17(16)20)4-3-7-21-14)18-23-22-15-6-5-13(10(2)25-27)24-26(15)18/h3-10H,1-2H3/t9-,10?/m0/s1	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	1.20	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100659 (US8507676, 8) Show SMILES CO\N=C(/C)c1ccc2ncc(Cc3c(F)cc4ncccc4c3F)n2n1 Show InChI InChI=1S/C19H15F2N5O/c1-11(25-27-2)16-5-6-18-23-10-12(26(18)24-16)8-14-15(20)9-17-13(19(14)21)4-3-7-22-17/h3-7,9-10H,8H2,1-2H3/b25-11+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	1.80	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100674 (US8507676, 23) Show SMILES C\C(=N/OCCO)c1cnc2nnn(Cc3ccc4ncccc4c3)c2n1 Show InChI InChI=1S/C18H17N7O2/c1-12(23-27-8-7-26)16-10-20-17-18(21-16)25(24-22-17)11-13-4-5-15-14(9-13)3-2-6-19-15/h2-6,9-10,26H,7-8,11H2,1H3/b23-12+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	2.20	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100673 (US8507676, 22) Show SMILES CO\N=C(/C)c1cnc2nnn(Cc3ccc4ncccc4c3)c2n1 Show InChI InChI=1S/C17H15N7O/c1-11(22-25-2)15-9-19-16-17(20-15)24(23-21-16)10-12-5-6-14-13(8-12)4-3-7-18-14/h3-9H,10H2,1-2H3/b22-11+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	2.40	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100707 (US8507676, 56) Show SMILES C\C(=N/OCCCO)c1ccc2nnc(Cc3c(F)cc4ncccc4c3F)n2n1 Show InChI InChI=1S/C20H18F2N6O2/c1-12(27-30-9-3-8-29)16-5-6-18-24-25-19(28(18)26-16)10-14-15(21)11-17-13(20(14)22)4-2-7-23-17/h2,4-7,11,29H,3,8-10H2,1H3/b27-12+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	2.5	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100663 (US8507676, 12-S) Show SMILES C[C@H](c1cnc2ccc(nn12)C(\C)=N\OCCO)c1c(F)cc2ncccc2c1F |r| Show InChI InChI=1S/C21H19F2N5O2/c1-12(20-15(22)10-17-14(21(20)23)4-3-7-24-17)18-11-25-19-6-5-16(26-28(18)19)13(2)27-30-9-8-29/h3-7,10-12,29H,8-9H2,1-2H3/b27-13+/t12-/m1/s1	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	2.5	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100703 (US8507676, 51-R | US8507676, 51-S) Show SMILES CC(c1cnc2ccc(nn12)C(\C)=N\OCCO)c1c(F)cc2n(C)ncc2c1F Show InChI InChI=1S/C20H20F2N6O2/c1-11(19-14(21)8-16-13(20(19)22)9-24-27(16)3)17-10-23-18-5-4-15(25-28(17)18)12(2)26-30-7-6-29/h4-5,8-11,29H,6-7H2,1-3H3/b26-12+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	2.80	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100666 (US8507676, 15) Show SMILES C\C(=N/OCCO)c1cnc2nnn(Cc3cc4cccnc4cc3F)c2n1 Show InChI InChI=1S/C18H16FN7O2/c1-11(24-28-6-5-27)16-9-21-17-18(22-16)26(25-23-17)10-13-7-12-3-2-4-20-15(12)8-14(13)19/h2-4,7-9,27H,5-6,10H2,1H3/b24-11+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	2.80	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100705 (US8507676, 54 | US8507676, 69) Show SMILES C\C(=N/OCCO)c1ccc2nnc(Cc3c(F)cc4ncccc4c3F)n2n1 Show InChI InChI=1S/C19H16F2N6O2/c1-11(26-29-8-7-28)15-4-5-17-23-24-18(27(17)25-15)9-13-14(20)10-16-12(19(13)21)3-2-6-22-16/h2-6,10,28H,7-9H2,1H3/b26-11+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	3	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100675 (US8507676, 24) Show SMILES CC(N=O)c1cnc2nnn(Cc3ccc4ncccc4c3)c2n1 Show InChI InChI=1S/C16H13N7O/c1-10(21-24)14-8-18-15-16(19-14)23(22-20-15)9-11-4-5-13-12(7-11)3-2-6-17-13/h2-8,10H,9H2,1H3	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	3	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM2214 (US8507676, 53-S) Show SMILES C[C@H](c1nnc2ccc(nn12)C(\C)=N\OCCO)c1c(F)cc2ncccc2c1F |r| Show InChI InChI=1S/C20H18F2N6O2/c1-11(18-14(21)10-16-13(19(18)22)4-3-7-23-16)20-25-24-17-6-5-15(26-28(17)20)12(2)27-30-9-8-29/h3-7,10-11,29H,8-9H2,1-2H3/b27-12+/t11-/m0/s1	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	3.5	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100691 (US8507676, 38) Show SMILES OCCO\N=C\c1cnc2nnn(Cc3ccc4ncccc4c3)c2n1 Show InChI InChI=1S/C17H15N7O2/c25-6-7-26-20-10-14-9-19-16-17(21-14)24(23-22-16)11-12-3-4-15-13(8-12)2-1-5-18-15/h1-5,8-10,25H,6-7,11H2/b20-10+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	3.60	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM2221 (US8507676, 80) Show SMILES C\C(=N/O)c1ccc2nnc(Cc3ccc4ncccc4c3)n2n1 Show InChI InChI=1S/C17H14N6O/c1-11(22-24)14-6-7-16-19-20-17(23(16)21-14)10-12-4-5-15-13(9-12)3-2-8-18-15/h2-9,24H,10H2,1H3/b22-11+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	3.80	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100706 (US8507676, 55) Show SMILES C\C(=N/OCCF)c1ccc2nnc(Cc3c(F)cc4ncccc4c3F)n2n1 Show InChI InChI=1S/C19H15F3N6O/c1-11(27-29-8-6-20)15-4-5-17-24-25-18(28(17)26-15)9-13-14(21)10-16-12(19(13)22)3-2-7-23-16/h2-5,7,10H,6,8-9H2,1H3/b27-11+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	3.80	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100690 (US8507676, 37B) Show SMILES C\C(=N/OCCNC(N)=O)c1cnc2nnn(Cc3ccc4ncccc4c3)c2n1 Show InChI InChI=1S/C19H19N9O2/c1-12(26-30-8-7-22-19(20)29)16-10-23-17-18(24-16)28(27-25-17)11-13-4-5-15-14(9-13)3-2-6-21-15/h2-6,9-10H,7-8,11H2,1H3,(H3,20,22,29)/b26-12+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	3.90	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100705 (US8507676, 54 | US8507676, 69) Show SMILES C\C(=N/OCCO)c1ccc2nnc(Cc3c(F)cc4ncccc4c3F)n2n1 Show InChI InChI=1S/C19H16F2N6O2/c1-11(26-29-8-7-28)15-4-5-17-23-24-18(27(17)25-15)9-13-14(20)10-16-12(19(13)21)3-2-6-22-16/h2-6,10,28H,7-9H2,1H3/b26-11+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	4.70	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100672 (US8507676, 21) Show SMILES C\C(=N/O[C@H]1CCN(C1)C(N)=O)c1cnc2nnn(Cc3cc4cccnc4cc3F)c2n1 |r| Show InChI InChI=1S/C21H20FN9O2/c1-12(28-33-15-4-6-30(11-15)21(23)32)18-9-25-19-20(26-18)31(29-27-19)10-14-7-13-3-2-5-24-17(13)8-16(14)22/h2-3,5,7-9,15H,4,6,10-11H2,1H3,(H2,23,32)/b28-12+/t15-/m0/s1	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	5.10	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100670 (US8507676, 19) Show SMILES C\C(=N/O[C@H]1CCNC1)c1cnc2nnn(Cc3cc4cccnc4cc3F)c2n1 |r| Show InChI InChI=1S/C20H19FN8O/c1-12(27-30-15-4-6-22-9-15)18-10-24-19-20(25-18)29(28-26-19)11-14-7-13-3-2-5-23-17(13)8-16(14)21/h2-3,5,7-8,10,15,22H,4,6,9,11H2,1H3/b27-12+/t15-/m0/s1	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	5.40	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100657 (US8507676, 6) Show SMILES C\C(=N/OCCO)c1ccc2ncc(Cc3ccc4ncccc4c3)n2n1 Show InChI InChI=1S/C20H19N5O2/c1-14(24-27-10-9-26)18-6-7-20-22-13-17(25(20)23-18)12-15-4-5-19-16(11-15)3-2-8-21-19/h2-8,11,13,26H,9-10,12H2,1H3/b24-14+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	5.5	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100714 (US8507676, 63 | US9062045, Comparator No. 2) Show SMILES CN1CCN(CC1)c1cnc2ccc(Cc3nnc4ccc(nn34)C(\C)=N\OCCO)cc2c1 Show InChI InChI=1S/C24H28N8O2/c1-17(29-34-12-11-33)21-5-6-23-26-27-24(32(23)28-21)14-18-3-4-22-19(13-18)15-20(16-25-22)31-9-7-30(2)8-10-31/h3-6,13,15-16,33H,7-12,14H2,1-2H3/b29-17+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	6	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100662 (US8507676, 11-S) Show SMILES C[C@H](c1cnc2ccc(nn12)C(\C)=N\OCCO)c1cc2cccnc2cc1F |r| Show InChI InChI=1S/C21H20FN5O2/c1-13(16-10-15-4-3-7-23-19(15)11-17(16)22)20-12-24-21-6-5-18(25-27(20)21)14(2)26-29-9-8-28/h3-7,10-13,28H,8-9H2,1-2H3/b26-14+/t13-/m0/s1	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	6	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100660 (US8507676, 9) Show SMILES C\C(=N/OCCO)c1ccc2ncc(Cc3c(F)cc4ncccc4c3F)n2n1 Show InChI InChI=1S/C20H17F2N5O2/c1-12(26-29-8-7-28)17-4-5-19-24-11-13(27(19)25-17)9-15-16(21)10-18-14(20(15)22)3-2-6-23-18/h2-6,10-11,28H,7-9H2,1H3/b26-12+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	6.70	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100695 (US8507676, 42) Show SMILES CCO\N=C(/C)c1ccc2nnc(Cc3ccc4ncccc4c3)n2n1 Show InChI InChI=1S/C19H18N6O/c1-3-26-24-13(2)16-8-9-18-21-22-19(25(18)23-16)12-14-6-7-17-15(11-14)5-4-10-20-17/h4-11H,3,12H2,1-2H3/b24-13+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	7	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100721 (US8507676, 71) Show SMILES C\C(=N/OC1COC1)c1cnc2nnn(Cc3ccc4ncccc4c3)c2n1 Show InChI InChI=1S/C19H17N7O2/c1-12(24-28-15-10-27-11-15)17-8-21-18-19(22-17)26(25-23-18)9-13-4-5-16-14(7-13)3-2-6-20-16/h2-8,15H,9-11H2,1H3/b24-12+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	7	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100729 (US8507676, 79) Show SMILES C\C(=N/OCCO)c1cnc2ncc(Cc3ccc4ncccc4c3)n2n1 Show InChI InChI=1S/C19H18N6O2/c1-13(24-27-8-7-26)18-12-22-19-21-11-16(25(19)23-18)10-14-4-5-17-15(9-14)3-2-6-20-17/h2-6,9,11-12,26H,7-8,10H2,1H3/b24-13+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	7.10	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100667 (US8507676, 16) Show SMILES CO\N=C(/C)c1cnc2nnn(Cc3cc4cccnc4cc3F)c2n1 Show InChI InChI=1S/C17H14FN7O/c1-10(23-26-2)15-8-20-16-17(21-15)25(24-22-16)9-12-6-11-4-3-5-19-14(11)7-13(12)18/h3-8H,9H2,1-2H3/b23-10+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	7.30	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100654 (US8507676, 3) Show SMILES C\C(=N/OCCO)c1ccc2ncc(Cc3cc4cccnc4cc3F)n2n1 Show InChI InChI=1S/C20H18FN5O2/c1-13(25-28-8-7-27)18-4-5-20-23-12-16(26(20)24-18)10-15-9-14-3-2-6-22-19(14)11-17(15)21/h2-6,9,11-12,27H,7-8,10H2,1H3/b25-13+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	8	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100718 (US8507676, 67) Show SMILES C\C(=N/OCCO)c1cnc2ccc(Cn3nnc4ncc(nc34)C(\C)=N\OCCO)cc2c1 Show InChI InChI=1S/C22H24N8O4/c1-14(27-33-7-5-31)18-10-17-9-16(3-4-19(17)23-11-18)13-30-22-21(26-29-30)24-12-20(25-22)15(2)28-34-8-6-32/h3-4,9-12,31-32H,5-8,13H2,1-2H3/b27-14+,28-15+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	8	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100678 (US8507676, 26B) Show SMILES C\C(=N/OCC(O)CO)c1cnc2nnn(Cc3ccc4ncccc4c3)c2n1 Show InChI InChI=1S/C19H19N7O3/c1-12(24-29-11-15(28)10-27)17-8-21-18-19(22-17)26(25-23-18)9-13-4-5-16-14(7-13)3-2-6-20-16/h2-8,15,27-28H,9-11H2,1H3/b24-12+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	9	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100653 (US8507676, 2) Show SMILES CO\N=C(/C)c1ccc2ncc(Cc3cc4cccnc4cc3F)n2n1 Show InChI InChI=1S/C19H16FN5O/c1-12(24-26-2)17-5-6-19-22-11-15(25(19)23-17)9-14-8-13-4-3-7-21-18(13)10-16(14)20/h3-8,10-11H,9H2,1-2H3/b24-12+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	10	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100694 (US8507676, 41) Show SMILES CO\N=C(/C)c1ccc2nnc(Cc3ccc4ncccc4c3)n2n1 Show InChI InChI=1S/C18H16N6O/c1-12(23-25-2)15-7-8-17-20-21-18(24(17)22-15)11-13-5-6-16-14(10-13)4-3-9-19-16/h3-10H,11H2,1-2H3/b23-12+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	10	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100722 (US8507676, 72) Show SMILES CC(N=O)c1cnc2nnn(Cc3cc4cccnc4cc3F)c2n1 Show InChI InChI=1S/C16H12FN7O/c1-9(22-25)14-7-19-15-16(20-14)24(23-21-15)8-11-5-10-3-2-4-18-13(10)6-12(11)17/h2-7,9H,8H2,1H3	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	11	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100704 (US8507676, 52) Show SMILES C\C(=N/OCCO)c1ccc2ncc(Cc3c(F)cc4n(C)ncc4c3F)n2n1 Show InChI InChI=1S/C19H18F2N6O2/c1-11(25-29-6-5-28)16-3-4-18-22-9-12(27(18)24-16)7-13-15(20)8-17-14(19(13)21)10-23-26(17)2/h3-4,8-10,28H,5-7H2,1-2H3/b25-11+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	11	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100686 (US8507676, 34) Show SMILES C\C(=N/OCCN)c1cnc2nnn(Cc3ccc4ncccc4c3)c2n1 Show InChI InChI=1S/C18H18N8O/c1-12(24-27-8-6-19)16-10-21-17-18(22-16)26(25-23-17)11-13-4-5-15-14(9-13)3-2-7-20-15/h2-5,7,9-10H,6,8,11,19H2,1H3/b24-12+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	12	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100736 (US8507676, 73) Show SMILES CC(c1nnc2ncc(nn12)C(\C)=N\OCCO)c1c(F)cc2ncccc2c1F Show InChI InChI=1S/C19H17F2N7O2/c1-10(16-13(20)8-14-12(17(16)21)4-3-5-22-14)18-24-25-19-23-9-15(26-28(18)19)11(2)27-30-7-6-29/h3-5,8-10,29H,6-7H2,1-2H3/b27-11+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	12	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100719 (US8507676, 68-R | US8507676, 68-S) Show SMILES CC(c1nnc2ccc(nn12)C(\C)=N\OCC(O)=O)c1c(F)cc2ncccc2c1F Show InChI InChI=1S/C20H16F2N6O3/c1-10(18-13(21)8-15-12(19(18)22)4-3-7-23-15)20-25-24-16-6-5-14(26-28(16)20)11(2)27-31-9-17(29)30/h3-8,10H,9H2,1-2H3,(H,29,30)/b27-11+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	13	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100697 (US8507676, 44) Show SMILES C\C(=N/OCCO)c1ccc2nnc(Cc3ccc4ncccc4c3)n2n1 Show InChI InChI=1S/C19H18N6O2/c1-13(24-27-10-9-26)16-6-7-18-21-22-19(25(18)23-16)12-14-4-5-17-15(11-14)3-2-8-20-17/h2-8,11,26H,9-10,12H2,1H3/b24-13+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	13	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100709 (US8507676, 58) Show SMILES C\C(=N/OCCO)c1ccc2nnc(Cc3ccc4ncccc4c3F)n2n1 Show InChI InChI=1S/C19H17FN6O2/c1-12(25-28-10-9-27)15-6-7-17-22-23-18(26(17)24-15)11-13-4-5-16-14(19(13)20)3-2-8-21-16/h2-8,27H,9-11H2,1H3/b25-12+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	14	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100716 (US8507676, 65) Show SMILES C\C(=N/OCCCCO)c1ccc2nnc(Cc3c(F)cc4ncccc4c3F)n2n1 Show InChI InChI=1S/C21H20F2N6O2/c1-13(28-31-10-3-2-9-30)17-6-7-19-25-26-20(29(19)27-17)11-15-16(22)12-18-14(21(15)23)5-4-8-24-18/h4-8,12,30H,2-3,9-11H2,1H3/b28-13+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	15	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100689 (US8507676, 37A) Show SMILES COC(=O)NCCO\N=C(/C)c1cnc2nnn(Cc3ccc4ncccc4c3)c2n1 Show InChI InChI=1S/C20H20N8O3/c1-13(26-31-9-8-22-20(29)30-2)17-11-23-18-19(24-17)28(27-25-18)12-14-5-6-16-15(10-14)4-3-7-21-16/h3-7,10-11H,8-9,12H2,1-2H3,(H,22,29)/b26-13+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	16.5	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100723 (US8507676, 74) Show SMILES CC(N=O)c1cnc2nnn(C(C)c3c(F)cc4ncccc4c3F)c2n1 Show InChI InChI=1S/C17H13F2N7O/c1-8(24-27)13-7-21-16-17(22-13)26(25-23-16)9(2)14-11(18)6-12-10(15(14)19)4-3-5-20-12/h3-9H,1-2H3	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	17	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100715 (US8507676, 64) Show SMILES COCCO\N=C(/C)c1ccc2nnc(C(C)c3c(F)cc4ncccc4c3F)n2n1 Show InChI InChI=1S/C21H20F2N6O2/c1-12(19-15(22)11-17-14(20(19)23)5-4-8-24-17)21-26-25-18-7-6-16(27-29(18)21)13(2)28-31-10-9-30-3/h4-8,11-12H,9-10H2,1-3H3/b28-13+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	18	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100737 (US8507676, 75-R) Show SMILES CC(N=O)c1ccc2nnc([C@H](C)c3c(F)cc4ncccc4c3F)n2n1 |r| Show InChI InChI=1S/C18H14F2N6O/c1-9(16-12(19)8-14-11(17(16)20)4-3-7-21-14)18-23-22-15-6-5-13(10(2)25-27)24-26(15)18/h3-10H,1-2H3/t9-,10?/m1/s1	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	19	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM2212 (US8507676, 39-S) Show SMILES C[C@H](c1nnc2ccc(nn12)C(\C)=N\OCCO)c1cc2cnn(C)c2cc1C |r| Show InChI InChI=1S/C20H23N7O2/c1-12-9-18-15(11-21-26(18)4)10-16(12)13(2)20-23-22-19-6-5-17(24-27(19)20)14(3)25-29-8-7-28/h5-6,9-11,13,28H,7-8H2,1-4H3/b25-14+/t13-/m0/s1	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	19	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100727 (US8507676, 77-R) Show SMILES C[C@H](c1nnc2ccc(nn12)C(\C)=N\OC(N)=O)c1c(F)cc2ncccc2c1F |r| Show InChI InChI=1S/C19H15F2N7O2/c1-9(16-12(20)8-14-11(17(16)21)4-3-7-23-14)18-25-24-15-6-5-13(26-28(15)18)10(2)27-30-19(22)29/h3-9H,1-2H3,(H2,22,29)/b27-10+/t9-/m0/s1	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100677 (US8507676, 26A) Show SMILES C\C(=N/OC(CO)CO)c1cnc2nnn(Cc3ccc4ncccc4c3)c2n1 Show InChI InChI=1S/C19H19N7O3/c1-12(24-29-15(10-27)11-28)17-8-21-18-19(22-17)26(25-23-18)9-13-4-5-16-14(7-13)3-2-6-20-16/h2-8,15,27-28H,9-11H2,1H3/b24-12+	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100713 (US8507676, 62-S) Show SMILES C[C@H](c1nnc2ccc(nn12)C(\C)=N\OCCO)c1cc2cccnc2cc1F |r| Show InChI InChI=1S/C20H19FN6O2/c1-12(15-10-14-4-3-7-22-18(14)11-16(15)21)20-24-23-19-6-5-17(25-27(19)20)13(2)26-29-9-8-28/h3-7,10-12,28H,8-9H2,1-2H3/b26-13+/t12-/m0/s1	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	21	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair
Hepatocyte growth factor receptor (Homo sapiens (Human))	BDBM100725 (US8507676, 76-S) Show SMILES C[C@H](c1nnc2ccc(nn12)C(\C)=N\OCC1CC1)c1c(F)cc2ncccc2c1F |r| Show InChI InChI=1S/C22H20F2N6O/c1-12(20-16(23)10-18-15(21(20)24)4-3-9-25-18)22-27-26-19-8-7-17(28-30(19)22)13(2)29-31-11-14-5-6-14/h3-4,7-10,12,14H,5-6,11H2,1-2H3/b29-13+/t12-/m0/s1	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	24	n/a	n/a	n/a	n/a	n/a	n/a
Novartis AG US Patent					Assay Description The kinase assay is based on the LanthaScreen technology. LanthaScreen is the detection of Time-Resolved Fluorescence Resonance Energy Transfer (TR-...				US Patent US8507676 (2013) BindingDB Entry DOI: 10.7270/Q2MS3RC9
					More data for this Ligand-Target Pair

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