Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human)) | BDBM31096 (CHEMBL290084 | Staurosporine | cid_451705) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 0.280 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [T790M,L858R] (Homo sapiens (Human)) | BDBM195875 (US9670213, Compound 020 N-(3-(2-(4-(4-methyl-1-pip...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 0.820 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [T790M,L858R] (Homo sapiens (Human)) | BDBM50383274 (CHEMBL1229592 | US10167264, WZ4002 | US9670213, WZ...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | PDB US Patent | n/a | n/a | 1.02 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Epidermal growth factor receptor [T790M,L858R] (Homo sapiens (Human)) | BDBM195887 (US9670213, Compound 032 N-(3-(2-(2-methoxy-4-(4-me...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.17 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [L858R] (Homo sapiens (Human)) | BDBM195875 (US9670213, Compound 020 N-(3-(2-(4-(4-methyl-1-pip...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM195875 (US9670213, Compound 020 N-(3-(2-(4-(4-methyl-1-pip...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 1.47 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [L858R] (Homo sapiens (Human)) | BDBM195887 (US9670213, Compound 032 N-(3-(2-(2-methoxy-4-(4-me...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 2.36 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [L858R] (Homo sapiens (Human)) | BDBM50383274 (CHEMBL1229592 | US10167264, WZ4002 | US9670213, WZ...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | PDB US Patent | n/a | n/a | 2.60 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Epidermal growth factor receptor [T790M,L858R] (Homo sapiens (Human)) | BDBM195873 (US9670213, Compound 018 N-(3-(2-(4-morpholinopheny...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.02 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM195887 (US9670213, Compound 032 N-(3-(2-(2-methoxy-4-(4-me...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.67 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [T790M,L858R] (Homo sapiens (Human)) | BDBM195880 (US9670213, Compound 025 4-(8-(3-acrylamidephenyl)-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.39 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [T790M,L858R] (Homo sapiens (Human)) | BDBM195879 (US9670213, Compound 024 N-(3-(2-(4-(acetylamino)-p...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.12 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [T790M,L858R] (Homo sapiens (Human)) | BDBM195870 (US9670213, Compound 015 N-(3-(7-oxo-2-(phenylamino...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.28 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [T790M,L858R] (Homo sapiens (Human)) | BDBM195877 (US9670213, Compound 022 N-(3-(7-oxo-2-(4-(1-pyrrol...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.33 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [T790M,L858R] (Homo sapiens (Human)) | BDBM195876 (US9670213, Compound 021 N-(3-(7-oxo-2-(4-(1-piperi...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.49 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [T790M,L858R] (Homo sapiens (Human)) | BDBM195878 (US9670213, Compound 023 N-(3-(2-(4-(diethylamino)p...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.57 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase Blk (Homo sapiens (Human)) | BDBM31096 (CHEMBL290084 | Staurosporine | cid_451705) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | US Patent | n/a | n/a | 5.60 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [L858R] (Homo sapiens (Human)) | BDBM195873 (US9670213, Compound 018 N-(3-(2-(4-morpholinopheny...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5.83 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [L858R] (Homo sapiens (Human)) | BDBM195881 (US9670213, Compound 026 N-(3-(2-(4-methoxyphenylam...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | 5.93 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM195881 (US9670213, Compound 026 N-(3-(2-(4-methoxyphenylam...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | 7.24 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM195873 (US9670213, Compound 018 N-(3-(2-(4-morpholinopheny...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 7.94 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [T790M,L858R] (Homo sapiens (Human)) | BDBM195861 (US9670213, Compound 006 N-(3-(2-(4-methoxyphenylam...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 8.40 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50383274 (CHEMBL1229592 | US10167264, WZ4002 | US9670213, WZ...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | PDB US Patent | n/a | n/a | 9.58 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Epidermal growth factor receptor [L858R] (Homo sapiens (Human)) | BDBM195880 (US9670213, Compound 025 4-(8-(3-acrylamidephenyl)-...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 9.64 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [L858R] (Homo sapiens (Human)) | BDBM195861 (US9670213, Compound 006 N-(3-(2-(4-methoxyphenylam...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM195861 (US9670213, Compound 006 N-(3-(2-(4-methoxyphenylam...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [T790M] (Homo sapiens (Human)) | BDBM195864 (US9670213, Compound 009 4-(dimethylamino)-N-(4-(2-...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [L858R] (Homo sapiens (Human)) | BDBM195870 (US9670213, Compound 015 N-(3-(7-oxo-2-(phenylamino...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [L858R] (Homo sapiens (Human)) | BDBM195876 (US9670213, Compound 021 N-(3-(7-oxo-2-(4-(1-piperi...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM195880 (US9670213, Compound 025 4-(8-(3-acrylamidephenyl)-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [L858R] (Homo sapiens (Human)) | BDBM195879 (US9670213, Compound 024 N-(3-(2-(4-(acetylamino)-p...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [L858R] (Homo sapiens (Human)) | BDBM195877 (US9670213, Compound 022 N-(3-(7-oxo-2-(4-(1-pyrrol...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase Blk (Homo sapiens (Human)) | BDBM195875 (US9670213, Compound 020 N-(3-(2-(4-(4-methyl-1-pip...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <14 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM195870 (US9670213, Compound 015 N-(3-(7-oxo-2-(phenylamino...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [T790M,L858R] (Homo sapiens (Human)) | BDBM195881 (US9670213, Compound 026 N-(3-(2-(4-methoxyphenylam...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | US Patent | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [L858R] (Homo sapiens (Human)) | BDBM195878 (US9670213, Compound 023 N-(3-(2-(4-(diethylamino)p...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM195879 (US9670213, Compound 024 N-(3-(2-(4-(acetylamino)-p...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM195869 (US9670213, Compound 014 N-(4-(7-oxo-2-(phenylamino...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [T790M] (Homo sapiens (Human)) | BDBM195861 (US9670213, Compound 006 N-(3-(2-(4-methoxyphenylam...) | PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM195876 (US9670213, Compound 021 N-(3-(7-oxo-2-(4-(1-piperi...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM195877 (US9670213, Compound 022 N-(3-(7-oxo-2-(4-(1-pyrrol...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM195878 (US9670213, Compound 023 N-(3-(2-(4-(diethylamino)p...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 23 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [L858R] (Homo sapiens (Human)) | BDBM195869 (US9670213, Compound 014 N-(4-(7-oxo-2-(phenylamino...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 26 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human)) | BDBM195081 (US9670213, Compound 001 8-(4-aminophenyl)-2-(4-met...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human)) | BDBM195860 (US9670213, Compound 005 8-(3-aminophenyl)-2-(4-met...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human)) | BDBM195883 (US9670213, Compound 028 2-(3-aminophenylamino)-8-(...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 34 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [T790M,L858R] (Homo sapiens (Human)) | BDBM195864 (US9670213, Compound 009 4-(dimethylamino)-N-(4-(2-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 39 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Epidermal growth factor receptor [T790M,L858R] (Homo sapiens (Human)) | BDBM195868 (US9670213, Compound 013 4-(dimethylamino)-N-(3-(7-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tyrosine-protein kinase Blk (Homo sapiens (Human)) | BDBM195873 (US9670213, Compound 018 N-(3-(2-(4-morpholinopheny...) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 41 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Receptor-type tyrosine-protein kinase FLT3 (Homo sapiens (Human)) | BDBM195885 (US9670213, Compound 030 2-(4-aminophenylamino)-8-(...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 43 | n/a | n/a | n/a | n/a | n/a | 25 |
East China University of Science and Technology US Patent | Assay Description In vitro enzyme activity assay: wild-type and various mutants (T790M, L858R, L861Q, L858 R/T790M) EGFR, Z′-Lyte Kinase Assay Kit were purchased... | US Patent US9670213 (2017) BindingDB Entry DOI: 10.7270/Q23R0R1P | |||||||||||
More data for this Ligand-Target Pair |
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