Compile Data Set for Download or QSAR

Found 146 hits Enz. Inhib. hit(s) with all data for entry = 50020270   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211992 (CHEMBL236419 | N-(4-(chlorodifluoromethoxy)phenyl)...) Show SMILES FC(F)(Cl)Oc1cccc(NC(=O)c2ccnn2CCc2ccncc2)c1 Show InChI InChI=1S/C18H15ClF2N4O2/c19-18(20,21)27-15-3-1-2-14(12-15)24-17(26)16-6-10-23-25(16)11-7-13-4-8-22-9-5-13/h1-6,8-10,12H,7,11H2,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	70	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211983 (1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)p...) Show SMILES FC(F)(F)Oc1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C18H15F3N4O2/c19-18(20,21)27-15-3-1-14(2-4-15)24-17(26)16-7-11-23-25(16)12-8-13-5-9-22-10-6-13/h1-7,9-11H,8,12H2,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	80	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Displacement of [32P]ATP from human VEGFR2 after 45 mins				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211983 (1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)p...) Show SMILES FC(F)(F)Oc1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C18H15F3N4O2/c19-18(20,21)27-15-3-1-14(2-4-15)24-17(26)16-7-11-23-25(16)12-8-13-5-9-22-10-6-13/h1-7,9-11H,8,12H2,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	90	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211992 (CHEMBL236419 | N-(4-(chlorodifluoromethoxy)phenyl)...) Show SMILES FC(F)(Cl)Oc1cccc(NC(=O)c2ccnn2CCc2ccncc2)c1 Show InChI InChI=1S/C18H15ClF2N4O2/c19-18(20,21)27-15-3-1-2-14(12-15)24-17(26)16-6-10-23-25(16)11-7-13-4-8-22-9-5-13/h1-6,8-10,12H,7,11H2,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	90	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Displacement of [32P]ATP from human VEGFR2 after 45 mins				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211976 (CHEMBL397323 | N-(4-chlorophenyl)-1-(2-(pyridin-4-...) Show SMILES Clc1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C17H15ClN4O/c18-14-1-3-15(4-2-14)21-17(23)16-7-11-20-22(16)12-8-13-5-9-19-10-6-13/h1-7,9-11H,8,12H2,(H,21,23)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	90	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Displacement of [32P]ATP from human VEGFR2 after 45 mins				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211976 (CHEMBL397323 | N-(4-chlorophenyl)-1-(2-(pyridin-4-...) Show SMILES Clc1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C17H15ClN4O/c18-14-1-3-15(4-2-14)21-17(23)16-7-11-20-22(16)12-8-13-5-9-19-10-6-13/h1-7,9-11H,8,12H2,(H,21,23)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	110	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211979 (CHEMBL399605 | N-(4-tert-butylphenyl)-1-(2-(pyridi...) Show SMILES CC(C)(C)c1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C21H24N4O/c1-21(2,3)17-4-6-18(7-5-17)24-20(26)19-10-14-23-25(19)15-11-16-8-12-22-13-9-16/h4-10,12-14H,11,15H2,1-3H3,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	130	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211979 (CHEMBL399605 | N-(4-tert-butylphenyl)-1-(2-(pyridi...) Show SMILES CC(C)(C)c1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C21H24N4O/c1-21(2,3)17-4-6-18(7-5-17)24-20(26)19-10-14-23-25(19)15-11-16-8-12-22-13-9-16/h4-10,12-14H,11,15H2,1-3H3,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	140	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Displacement of [32P]ATP from human VEGFR2 after 45 mins				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211972 (CHEMBL233823 | N-(3-chloro-4-(trifluoromethyl)phen...) Show SMILES FC(F)(F)c1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1Cl Show InChI InChI=1S/C18H14ClF3N4O/c19-15-11-13(1-2-14(15)18(20,21)22)25-17(27)16-5-9-24-26(16)10-6-12-3-7-23-8-4-12/h1-5,7-9,11H,6,10H2,(H,25,27)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	160	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Displacement of [32P]ATP from human VEGFR2 after 45 mins				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211972 (CHEMBL233823 | N-(3-chloro-4-(trifluoromethyl)phen...) Show SMILES FC(F)(F)c1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1Cl Show InChI InChI=1S/C18H14ClF3N4O/c19-15-11-13(1-2-14(15)18(20,21)22)25-17(27)16-5-9-24-26(16)10-6-12-3-7-23-8-4-12/h1-5,7-9,11H,6,10H2,(H,25,27)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	170	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211983 (1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)p...) Show SMILES FC(F)(F)Oc1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C18H15F3N4O2/c19-18(20,21)27-15-3-1-14(2-4-15)24-17(26)16-7-11-23-25(16)12-8-13-5-9-22-10-6-13/h1-7,9-11H,8,12H2,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	18	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in human 293 cells by cell-based ELISA				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211992 (CHEMBL236419 | N-(4-(chlorodifluoromethoxy)phenyl)...) Show SMILES FC(F)(Cl)Oc1cccc(NC(=O)c2ccnn2CCc2ccncc2)c1 Show InChI InChI=1S/C18H15ClF2N4O2/c19-18(20,21)27-15-3-1-2-14(12-15)24-17(26)16-6-10-23-25(16)11-7-13-4-8-22-9-5-13/h1-6,8-10,12H,7,11H2,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	21	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in human 293 cells by cell-based ELISA				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211983 (1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)p...) Show SMILES FC(F)(F)Oc1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C18H15F3N4O2/c19-18(20,21)27-15-3-1-14(2-4-15)24-17(26)16-7-11-23-25(16)12-8-13-5-9-22-10-6-13/h1-7,9-11H,8,12H2,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	28	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211979 (CHEMBL399605 | N-(4-tert-butylphenyl)-1-(2-(pyridi...) Show SMILES CC(C)(C)c1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C21H24N4O/c1-21(2,3)17-4-6-18(7-5-17)24-20(26)19-10-14-23-25(19)15-11-16-8-12-22-13-9-16/h4-10,12-14H,11,15H2,1-3H3,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	33	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in human 293 cells by cell-based ELISA				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211979 (CHEMBL399605 | N-(4-tert-butylphenyl)-1-(2-(pyridi...) Show SMILES CC(C)(C)c1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C21H24N4O/c1-21(2,3)17-4-6-18(7-5-17)24-20(26)19-10-14-23-25(19)15-11-16-8-12-22-13-9-16/h4-10,12-14H,11,15H2,1-3H3,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	42	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50212000 (1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethyl)ph...) Show SMILES FC(F)(F)c1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C18H15F3N4O/c19-18(20,21)14-1-3-15(4-2-14)24-17(26)16-7-11-23-25(16)12-8-13-5-9-22-10-6-13/h1-7,9-11H,8,12H2,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	48	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in human 293 cells by cell-based ELISA				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211981 (CHEMBL236420 | N-(4-isopropylphenyl)-1-(2-(pyridin...) Show SMILES CC(C)c1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C20H22N4O/c1-15(2)17-3-5-18(6-4-17)23-20(25)19-9-13-22-24(19)14-10-16-7-11-21-12-8-16/h3-9,11-13,15H,10,14H2,1-2H3,(H,23,25)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	53	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in human 293 cells by cell-based ELISA				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50212000 (1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethyl)ph...) Show SMILES FC(F)(F)c1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C18H15F3N4O/c19-18(20,21)14-1-3-15(4-2-14)24-17(26)16-7-11-23-25(16)12-8-13-5-9-22-10-6-13/h1-7,9-11H,8,12H2,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	69	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211981 (CHEMBL236420 | N-(4-isopropylphenyl)-1-(2-(pyridin...) Show SMILES CC(C)c1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C20H22N4O/c1-15(2)17-3-5-18(6-4-17)23-20(25)19-9-13-22-24(19)14-10-16-7-11-21-12-8-16/h3-9,11-13,15H,10,14H2,1-2H3,(H,23,25)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	74	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211976 (CHEMBL397323 | N-(4-chlorophenyl)-1-(2-(pyridin-4-...) Show SMILES Clc1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C17H15ClN4O/c18-14-1-3-15(4-2-14)21-17(23)16-7-11-20-22(16)12-8-13-5-9-19-10-6-13/h1-7,9-11H,8,12H2,(H,21,23)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	77	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50212010 (CHEMBL392935 | N-(4-ethylphenyl)-1-(2-(pyridin-4-y...) Show SMILES CCc1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C19H20N4O/c1-2-15-3-5-17(6-4-15)22-19(24)18-9-13-21-23(18)14-10-16-7-11-20-12-8-16/h3-9,11-13H,2,10,14H2,1H3,(H,22,24)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	86	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in human 293 cells by cell-based ELISA				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211970 (CHEMBL234009 | N-(3,4-dimethoxyphenyl)-1-(2-(pyrid...) Show SMILES COc1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1OC Show InChI InChI=1S/C19H20N4O3/c1-25-17-4-3-15(13-18(17)26-2)22-19(24)16-7-11-21-23(16)12-8-14-5-9-20-10-6-14/h3-7,9-11,13H,8,12H2,1-2H3,(H,22,24)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	90	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in human 293 cells by cell-based ELISA				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211976 (CHEMBL397323 | N-(4-chlorophenyl)-1-(2-(pyridin-4-...) Show SMILES Clc1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C17H15ClN4O/c18-14-1-3-15(4-2-14)21-17(23)16-7-11-20-22(16)12-8-13-5-9-19-10-6-13/h1-7,9-11H,8,12H2,(H,21,23)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	90	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in human 293 cells by cell-based ELISA				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211972 (CHEMBL233823 | N-(3-chloro-4-(trifluoromethyl)phen...) Show SMILES FC(F)(F)c1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1Cl Show InChI InChI=1S/C18H14ClF3N4O/c19-15-11-13(1-2-14(15)18(20,21)22)25-17(27)16-5-9-24-26(16)10-6-12-3-7-23-8-4-12/h1-5,7-9,11H,6,10H2,(H,25,27)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	95	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in human 293 cells by cell-based ELISA				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 1 (Homo sapiens (Human))	BDBM50211976 (CHEMBL397323 | N-(4-chlorophenyl)-1-(2-(pyridin-4-...) Show SMILES Clc1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C17H15ClN4O/c18-14-1-3-15(4-2-14)21-17(23)16-7-11-20-22(16)12-8-13-5-9-19-10-6-13/h1-7,9-11H,8,12H2,(H,21,23)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	97	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR1 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211990 (CHEMBL392330 | N-(3,4-dichlorophenyl)-1-(2-(pyridi...) Show SMILES Clc1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1Cl Show InChI InChI=1S/C17H14Cl2N4O/c18-14-2-1-13(11-15(14)19)22-17(24)16-5-9-21-23(16)10-6-12-3-7-20-8-4-12/h1-5,7-9,11H,6,10H2,(H,22,24)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	120	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in human 293 cells by cell-based ELISA				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50212010 (CHEMBL392935 | N-(4-ethylphenyl)-1-(2-(pyridin-4-y...) Show SMILES CCc1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C19H20N4O/c1-2-15-3-5-17(6-4-15)22-19(24)18-9-13-21-23(18)14-10-16-7-11-20-12-8-16/h3-9,11-13H,2,10,14H2,1H3,(H,22,24)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	120	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211980 (1-(2-(pyridin-4-yl)ethyl)-N-(quinolin-3-yl)-1H-pyr...) Show SMILES O=C(Nc1cnc2ccccc2c1)c1ccnn1CCc1ccncc1 Show InChI InChI=1S/C20H17N5O/c26-20(24-17-13-16-3-1-2-4-18(16)22-14-17)19-7-11-23-25(19)12-8-15-5-9-21-10-6-15/h1-7,9-11,13-14H,8,12H2,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	180	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211972 (CHEMBL233823 | N-(3-chloro-4-(trifluoromethyl)phen...) Show SMILES FC(F)(F)c1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1Cl Show InChI InChI=1S/C18H14ClF3N4O/c19-15-11-13(1-2-14(15)18(20,21)22)25-17(27)16-5-9-24-26(16)10-6-12-3-7-23-8-4-12/h1-5,7-9,11H,6,10H2,(H,25,27)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	180	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 1 (Homo sapiens (Human))	BDBM50211983 (1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)p...) Show SMILES FC(F)(F)Oc1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C18H15F3N4O2/c19-18(20,21)27-15-3-1-14(2-4-15)24-17(26)16-7-11-23-25(16)12-8-13-5-9-22-10-6-13/h1-7,9-11H,8,12H2,(H,24,26)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	190	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR1 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 1 (Homo sapiens (Human))	BDBM50212010 (CHEMBL392935 | N-(4-ethylphenyl)-1-(2-(pyridin-4-y...) Show SMILES CCc1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C19H20N4O/c1-2-15-3-5-17(6-4-15)22-19(24)18-9-13-21-23(18)14-10-16-7-11-20-12-8-16/h3-9,11-13H,2,10,14H2,1H3,(H,22,24)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	220	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR1 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211990 (CHEMBL392330 | N-(3,4-dichlorophenyl)-1-(2-(pyridi...) Show SMILES Clc1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1Cl Show InChI InChI=1S/C17H14Cl2N4O/c18-14-2-1-13(11-15(14)19)22-17(24)16-5-9-21-23(16)10-6-12-3-7-20-8-4-12/h1-5,7-9,11H,6,10H2,(H,22,24)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	260	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211975 (1-(2-(pyridin-4-yl)ethyl)-N-(3-(trifluoromethoxy)p...) Show SMILES FC(F)(F)Oc1cccc(NC(=O)c2ccnn2CCc2ccncc2)c1 Show InChI InChI=1S/C18H15F3N4O2/c19-18(20,21)27-15-3-1-2-14(12-15)24-17(26)16-6-10-23-25(16)11-7-13-4-8-22-9-5-13/h1-6,8-10,12H,7,11H2,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	280	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in human 293 cells by cell-based ELISA				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 1 (Homo sapiens (Human))	BDBM50211992 (CHEMBL236419 | N-(4-(chlorodifluoromethoxy)phenyl)...) Show SMILES FC(F)(Cl)Oc1cccc(NC(=O)c2ccnn2CCc2ccncc2)c1 Show InChI InChI=1S/C18H15ClF2N4O2/c19-18(20,21)27-15-3-1-2-14(12-15)24-17(26)16-6-10-23-25(16)11-7-13-4-8-22-9-5-13/h1-6,8-10,12H,7,11H2,(H,24,26)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	320	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR1 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211975 (1-(2-(pyridin-4-yl)ethyl)-N-(3-(trifluoromethoxy)p...) Show SMILES FC(F)(F)Oc1cccc(NC(=O)c2ccnn2CCc2ccncc2)c1 Show InChI InChI=1S/C18H15F3N4O2/c19-18(20,21)27-15-3-1-2-14(12-15)24-17(26)16-6-10-23-25(16)11-7-13-4-8-22-9-5-13/h1-6,8-10,12H,7,11H2,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	370	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 1 (Homo sapiens (Human))	BDBM50212000 (1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethyl)ph...) Show SMILES FC(F)(F)c1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C18H15F3N4O/c19-18(20,21)14-1-3-15(4-2-14)24-17(26)16-7-11-23-25(16)12-8-13-5-9-22-10-6-13/h1-7,9-11H,8,12H2,(H,24,26)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	380	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR1 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50212004 (CHEMBL234202 | N-(4-chlorophenyl)-1-(2-(pyridin-4-...) Show SMILES Clc1ccc(NC(=O)c2nccn2CCc2ccncc2)cc1 Show InChI InChI=1S/C17H15ClN4O/c18-14-1-3-15(4-2-14)21-17(23)16-20-10-12-22(16)11-7-13-5-8-19-9-6-13/h1-6,8-10,12H,7,11H2,(H,21,23)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	380	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 1 (Homo sapiens (Human))	BDBM50211980 (1-(2-(pyridin-4-yl)ethyl)-N-(quinolin-3-yl)-1H-pyr...) Show SMILES O=C(Nc1cnc2ccccc2c1)c1ccnn1CCc1ccncc1 Show InChI InChI=1S/C20H17N5O/c26-20(24-17-13-16-3-1-2-4-18(16)22-14-17)19-7-11-23-25(19)12-8-15-5-9-21-10-6-15/h1-7,9-11,13-14H,8,12H2,(H,24,26)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	380	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR1 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211970 (CHEMBL234009 | N-(3,4-dimethoxyphenyl)-1-(2-(pyrid...) Show SMILES COc1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1OC Show InChI InChI=1S/C19H20N4O3/c1-25-17-4-3-15(13-18(17)26-2)22-19(24)16-7-11-21-23(16)12-8-14-5-9-20-10-6-14/h3-7,9-11,13H,8,12H2,1-2H3,(H,22,24)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	440	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 1 (Homo sapiens (Human))	BDBM50211981 (CHEMBL236420 | N-(4-isopropylphenyl)-1-(2-(pyridin...) Show SMILES CC(C)c1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C20H22N4O/c1-15(2)17-3-5-18(6-4-17)23-20(25)19-9-13-22-24(19)14-10-16-7-11-21-12-8-16/h3-9,11-13,15H,10,14H2,1-2H3,(H,23,25)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	440	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR1 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211991 (CHEMBL233822 | N-(4-chloro-3-(trifluoromethyl)phen...) Show SMILES FC(F)(F)c1cc(NC(=O)c2ccnn2CCc2ccncc2)ccc1Cl Show InChI InChI=1S/C18H14ClF3N4O/c19-15-2-1-13(11-14(15)18(20,21)22)25-17(27)16-5-9-24-26(16)10-6-12-3-7-23-8-4-12/h1-5,7-9,11H,6,10H2,(H,25,27)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	450	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in human 293 cells by cell-based ELISA				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 1 (Homo sapiens (Human))	BDBM50211975 (1-(2-(pyridin-4-yl)ethyl)-N-(3-(trifluoromethoxy)p...) Show SMILES FC(F)(F)Oc1cccc(NC(=O)c2ccnn2CCc2ccncc2)c1 Show InChI InChI=1S/C18H15F3N4O2/c19-18(20,21)27-15-3-1-2-14(12-15)24-17(26)16-6-10-23-25(16)11-7-13-4-8-22-9-5-13/h1-6,8-10,12H,7,11H2,(H,24,26)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	450	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR1 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211971 (1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethyl)ph...) Show SMILES FC(F)(F)c1ccc(NC(=O)c2nccn2CCc2ccncc2)cc1 Show InChI InChI=1S/C18H15F3N4O/c19-18(20,21)14-1-3-15(4-2-14)24-17(26)16-23-10-12-25(16)11-7-13-5-8-22-9-6-13/h1-6,8-10,12H,7,11H2,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	470	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 1 (Homo sapiens (Human))	BDBM50211979 (CHEMBL399605 | N-(4-tert-butylphenyl)-1-(2-(pyridi...) Show SMILES CC(C)(C)c1ccc(NC(=O)c2ccnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C21H24N4O/c1-21(2,3)17-4-6-18(7-5-17)24-20(26)19-10-14-23-25(19)15-11-16-8-12-22-13-9-16/h4-10,12-14H,11,15H2,1-3H3,(H,24,26)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	590	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR1 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211988 (CHEMBL393001 | N-(4-chlorophenyl)-1-(2-(pyridin-4-...) Show SMILES Clc1ccc(NC(=O)c2nnnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C15H13ClN6O/c16-12-1-3-13(4-2-12)18-15(23)14-19-20-21-22(14)10-7-11-5-8-17-9-6-11/h1-6,8-9H,7,10H2,(H,18,23)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	640	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211991 (CHEMBL233822 | N-(4-chloro-3-(trifluoromethyl)phen...) Show SMILES FC(F)(F)c1cc(NC(=O)c2ccnn2CCc2ccncc2)ccc1Cl Show InChI InChI=1S/C18H14ClF3N4O/c19-15-2-1-13(11-14(15)18(20,21)22)25-17(27)16-5-9-24-26(16)10-6-12-3-7-23-8-4-12/h1-5,7-9,11H,6,10H2,(H,25,27)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	750	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211982 (CHEMBL234010 | N-(4-chlorophenyl)-3-methyl-1-(2-(p...) Show SMILES Cc1cc(C(=O)Nc2ccc(Cl)cc2)n(CCc2ccncc2)n1 Show InChI InChI=1S/C18H17ClN4O/c1-13-12-17(18(24)21-16-4-2-15(19)3-5-16)23(22-13)11-8-14-6-9-20-10-7-14/h2-7,9-10,12H,8,11H2,1H3,(H,21,24)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	780	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 1 (Homo sapiens (Human))	BDBM50211971 (1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethyl)ph...) Show SMILES FC(F)(F)c1ccc(NC(=O)c2nccn2CCc2ccncc2)cc1 Show InChI InChI=1S/C18H15F3N4O/c19-18(20,21)14-1-3-15(4-2-14)24-17(26)16-23-10-12-25(16)11-7-13-5-8-22-9-6-13/h1-6,8-10,12H,7,11H2,(H,24,26)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	790	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR1 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50211967 (1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethoxy)p...) Show SMILES FC(F)(F)Oc1ccc(NC(=O)c2nccn2CCc2ccncc2)cc1 Show InChI InChI=1S/C18H15F3N4O2/c19-18(20,21)27-15-3-1-14(2-4-15)24-17(26)16-23-10-12-25(16)11-7-13-5-8-22-9-6-13/h1-6,8-10,12H,7,11H2,(H,24,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	790	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair
Vascular endothelial growth factor receptor 2 (Homo sapiens (Human))	BDBM50212007 (1-(2-(pyridin-4-yl)ethyl)-N-(4-(trifluoromethyl)ph...) Show SMILES FC(F)(F)c1ccc(NC(=O)c2nnnn2CCc2ccncc2)cc1 Show InChI InChI=1S/C16H13F3N6O/c17-16(18,19)12-1-3-13(4-2-12)21-15(26)14-22-23-24-25(14)10-7-11-5-8-20-9-6-11/h1-6,8-9H,7,10H2,(H,21,26)	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	850	n/a	n/a	n/a	n/a	n/a	n/a
Chemical Diversity, Inc. Curated by ChEMBL					Assay Description Inhibition of VEGFR2 assessed as inhibition of phosphorylation in presence of 2 uM ATP by HTRF assay				Bioorg Med Chem Lett 17: 3550-7 (2007) Article DOI: 10.1016/j.bmcl.2007.04.042 BindingDB Entry DOI: 10.7270/Q2MG7P6N
					More data for this Ligand-Target Pair

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