Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301193 (6-((5-ethyl-4-(fluoromethyl)thiazol-2-ylthio)methy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.130 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301204 (6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-meth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.160 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301192 (6-((4-(fluoromethyl)-5-methylthiazol-2-ylthio)meth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301203 (6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-fluo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.270 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301209 (6-((4,5-dimethylthiazol-2-ylthio)methyl)-N-((6-met...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.270 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301207 (6-((5-ethyl-4-methyloxazol-2-ylthio)methyl)-N-((6-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.390 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301208 (CHEMBL566040 | N-((6-methylpyridin-2-yl)methyl)-4-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.460 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301210 (6-((5-(fluoromethyl)-4-methylthiazol-2-ylthio)meth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.560 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301202 (6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-meth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.690 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301197 (6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-fluo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301206 (CHEMBL566889 | [6-(4,5-Dimethyl-oxazol-2-ylsulfany...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301200 (6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-(flu...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301198 (6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-(met...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301196 (6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((2-fluo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301195 (6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((2-fluo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301205 (CHEMBL566441 | [6-(4,5-Dimethyl-oxazol-2-ylsulfany...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301199 (6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-((2-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301201 (6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-(2-f...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50301194 (6-((4,5-dimethyloxazol-2-ylthio)methyl)-N-((6-fluo...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY1 receptor overexpressed in CHO cell membrane after 120 mins by scintillation counting | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 2 (Homo sapiens (Human)) | BDBM50301192 (6-((4-(fluoromethyl)-5-methylthiazol-2-ylthio)meth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY2 receptor | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 4 (Homo sapiens (Human)) | BDBM50301192 (6-((4-(fluoromethyl)-5-methylthiazol-2-ylthio)meth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY4 receptor | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50301192 (6-((4-(fluoromethyl)-5-methylthiazol-2-ylthio)meth...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY5 receptor | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 2 (Homo sapiens (Human)) | BDBM50301193 (6-((5-ethyl-4-(fluoromethyl)thiazol-2-ylthio)methy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY2 receptor | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 4 (Homo sapiens (Human)) | BDBM50301193 (6-((5-ethyl-4-(fluoromethyl)thiazol-2-ylthio)methy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY4 receptor | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 5 (Homo sapiens (Human)) | BDBM50301193 (6-((5-ethyl-4-(fluoromethyl)thiazol-2-ylthio)methy...) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Tsukuba Research Institute Curated by ChEMBL | Assay Description Displacement of [125I]-PYY from human NPYY5 receptor | Bioorg Med Chem Lett 19: 5124-7 (2009) Article DOI: 10.1016/j.bmcl.2009.07.030 BindingDB Entry DOI: 10.7270/Q26M36WZ | |||||||||||
More data for this Ligand-Target Pair |