Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM21281 ((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | 0.280 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Agonist activity at CB2 receptor (unknown origin) | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM21281 ((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Agonist activity at CB1 receptor (unknown origin) | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50160434 ((6-iodo-2-methyl-1-(2-morpholinoethyl)-1H-indol-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 31 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Inverse agonist activity at CB2 receptor (unknown origin) | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM60994 ((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL DrugBank KEGG PC cid PC sid PDB UniChem Similars | DrugBank Article PubMed | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Agonist activity at CB2 receptor (unknown origin) | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM60994 ((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL DrugBank KEGG PC cid PC sid PDB UniChem Similars | DrugBank Article PubMed | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Agonist activity at CB1 receptor (unknown origin) | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207242 (CHEMBL3901140) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207267 (CHEMBL3960083) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207271 (CHEMBL594935) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207259 (CHEMBL3892181) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207256 (CHEMBL3898407) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207269 (CHEMBL3907434) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207239 (CHEMBL3907898) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207261 (CHEMBL3891003) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207255 (CHEMBL3944807) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207247 (CHEMBL3920181) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207254 (CHEMBL3938131) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207257 (CHEMBL3950235) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207266 (CHEMBL3932295) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50207255 (CHEMBL3944807) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207244 (CHEMBL3916891) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50207258 (CHEMBL3889952) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207245 (CHEMBL3898882) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207250 (CHEMBL3915743) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207240 (CHEMBL3917967) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207263 (CHEMBL3922512) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50207271 (CHEMBL594935) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM106773 (2‐(4‐methoxyphenyl)‐1‐[(4&...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem Similars | Article PubMed | 700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50207244 (CHEMBL3916891) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207241 (CHEMBL3895577) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 800 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207262 (CHEMBL3898880) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 900 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207251 (CHEMBL3916164) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207258 (CHEMBL3889952) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207265 (CHEMBL3914550) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207270 (CHEMBL3926929) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207252 (CHEMBL3935866) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207248 (CHEMBL3904520) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207260 (CHEMBL3905573) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 2 (Homo sapiens (Human)) | BDBM50207246 (CHEMBL3984372) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50207251 (CHEMBL3916164) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50207254 (CHEMBL3938131) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50207267 (CHEMBL3960083) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50207246 (CHEMBL3984372) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50207240 (CHEMBL3917967) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50207269 (CHEMBL3907434) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 5.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50160434 ((6-iodo-2-methyl-1-(2-morpholinoethyl)-1H-indol-3-...) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 5.25E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Agonist activity at CB1 receptor (unknown origin) | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50207265 (CHEMBL3914550) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 5.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50207247 (CHEMBL3920181) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50207259 (CHEMBL3892181) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50207243 (CHEMBL3911245) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50207266 (CHEMBL3932295) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Pontificia Universidad Cat£lica de Chile Curated by ChEMBL | Assay Description Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cell membranes incubated for 1.5 hrs | Eur J Med Chem 124: 17-35 (2016) Article DOI: 10.1016/j.ejmech.2016.08.005 BindingDB Entry DOI: 10.7270/Q2Q2426V | |||||||||||
More data for this Ligand-Target Pair |
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