Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50170966 (10-hydroxy-3,4-dimethoxy-17-methyl-17-azatetracycl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 2.44 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H][DAMGO] from mu opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50026682 (10-hydroxy-3,4-dimethoxy-17-methyl-(10S)-17-azatet...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 3.88 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H][DAMGO] from mu opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50026687 (3-hydroxy-4,10-dimethoxy-17-methyl-(10S)-17-azatet...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 4.65 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H][DAMGO] from mu opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50170964 (3-hydroxy-4,10-dimethoxy-17-methyl-17-azatetracycl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 5.38 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H][DAMGO] from mu opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50000092 ((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | 6.55 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50170962 (3,10-dihydroxy-4-methoxy-17-methyl-17-azatetracycl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 31.7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H][DAMGO] from mu opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50170963 (3,10-dihydroxy-4-methoxy-17-methyl-17-azatetracycl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 32.6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H][DAMGO] from mu opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mu-type opioid receptor (Rattus norvegicus (rat)) | BDBM50370595 (OXYCODONE | Oxycontin | US1184575, oxycodone | US9...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase DrugBank KEGG PC cid PC sid PDB UniChem Similars | Article PubMed | 43.6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50026682 (10-hydroxy-3,4-dimethoxy-17-methyl-(10S)-17-azatet...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 91.6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H]Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50170966 (10-hydroxy-3,4-dimethoxy-17-methyl-17-azatetracycl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 107 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H]Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50000092 ((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 113 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H]U-69593 from kappa opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50026687 (3-hydroxy-4,10-dimethoxy-17-methyl-(10S)-17-azatet...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 180 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H]Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50170964 (3-hydroxy-4,10-dimethoxy-17-methyl-17-azatetracycl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 197 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H]Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50000092 ((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 217 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H[Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50170966 (10-hydroxy-3,4-dimethoxy-17-methyl-17-azatetracycl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 364 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of[3H]U69,593 from kappa opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50170964 (3-hydroxy-4,10-dimethoxy-17-methyl-17-azatetracycl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 378 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of[3H]U69,593 from kappa opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50170962 (3,10-dihydroxy-4-methoxy-17-methyl-17-azatetracycl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 498 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H]Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50026687 (3-hydroxy-4,10-dimethoxy-17-methyl-(10S)-17-azatet...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 592 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of[3H]U69,593 from kappa opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50026682 (10-hydroxy-3,4-dimethoxy-17-methyl-(10S)-17-azatet...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 693 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of[3H]U69,593 from kappa opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50170963 (3,10-dihydroxy-4-methoxy-17-methyl-17-azatetracycl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 763 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of[3H]U69,593 from kappa opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50170963 (3,10-dihydroxy-4-methoxy-17-methyl-17-azatetracycl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 881 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H]Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50370595 (OXYCODONE | Oxycontin | US1184575, oxycodone | US9...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase DrugBank KEGG PC cid PC sid PDB UniChem Similars | Article PubMed | 1.09E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H[Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50170962 (3,10-dihydroxy-4-methoxy-17-methyl-17-azatetracycl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.65E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of[3H]U69,593 from kappa opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kappa-type opioid receptor (Rattus norvegicus (rat)) | BDBM50370595 (OXYCODONE | Oxycontin | US1184575, oxycodone | US9...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase DrugBank KEGG PC cid PC sid PDB UniChem Similars | Article PubMed | 2.66E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Innsbruck Curated by ChEMBL | Assay Description Displacement of [3H]U-69593 from kappa opioid receptor of rat brain membranes | J Med Chem 48: 5052-5 (2005) Article DOI: 10.1021/jm0580205 BindingDB Entry DOI: 10.7270/Q2P26ZW1 | |||||||||||
More data for this Ligand-Target Pair |