BindingDB PrimarySearch

Found 9 hits Enz. Inhib. hit(s) with all data for assayid = 1 entry = 5767
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Cathepsin B (Homo sapiens (Human))	BDBM93204 (Mercaptomethyl ketone Inhibitor, 53) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	2	n/a	n/a	n/a	n/a	n/a	n/a	5.5	n/a
University of California-Berkeley					Assay Description A fluorometric high-throughput assay for activity against cathepsin B was performed in 96-well microtiter plates. The assay were performed in Dynate...				J Comb Chem 5: 869-80 (2003) Article DOI: 10.1021/cc034008r BindingDB Entry DOI: 10.7270/Q28914GH
University of California-Berkeley					More data for this Ligand-Target Pair
Cathepsin B (Homo sapiens (Human))	BDBM93203 (Mercaptomethyl ketone Inhibitor, 52) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	4.70	n/a	n/a	n/a	n/a	n/a	n/a	5.5	n/a
University of California-Berkeley					Assay Description A fluorometric high-throughput assay for activity against cathepsin B was performed in 96-well microtiter plates. The assay were performed in Dynate...				J Comb Chem 5: 869-80 (2003) Article DOI: 10.1021/cc034008r BindingDB Entry DOI: 10.7270/Q28914GH
University of California-Berkeley					More data for this Ligand-Target Pair
Cathepsin B (Homo sapiens (Human))	BDBM93196 (Mercaptomethyl ketone Inhibitor, 45) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	13	n/a	n/a	n/a	n/a	n/a	n/a	5.5	n/a
University of California-Berkeley					Assay Description A fluorometric high-throughput assay for activity against cathepsin B was performed in 96-well microtiter plates. The assay were performed in Dynate...				J Comb Chem 5: 869-80 (2003) Article DOI: 10.1021/cc034008r BindingDB Entry DOI: 10.7270/Q28914GH
University of California-Berkeley					More data for this Ligand-Target Pair
Cathepsin B (Homo sapiens (Human))	BDBM93198 (Mercaptomethyl ketone Inhibitor, 47) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	50	n/a	n/a	n/a	n/a	n/a	n/a	5.5	n/a
University of California-Berkeley					Assay Description A fluorometric high-throughput assay for activity against cathepsin B was performed in 96-well microtiter plates. The assay were performed in Dynate...				J Comb Chem 5: 869-80 (2003) Article DOI: 10.1021/cc034008r BindingDB Entry DOI: 10.7270/Q28914GH
University of California-Berkeley					More data for this Ligand-Target Pair
Cathepsin B (Homo sapiens (Human))	BDBM93202 (Mercaptomethyl ketone Inhibitor, 51) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	50	n/a	n/a	n/a	n/a	n/a	n/a	5.5	n/a
University of California-Berkeley					Assay Description A fluorometric high-throughput assay for activity against cathepsin B was performed in 96-well microtiter plates. The assay were performed in Dynate...				J Comb Chem 5: 869-80 (2003) Article DOI: 10.1021/cc034008r BindingDB Entry DOI: 10.7270/Q28914GH
University of California-Berkeley					More data for this Ligand-Target Pair
Cathepsin B (Homo sapiens (Human))	BDBM93197 (Mercaptomethyl ketone Inhibitor, 46) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	110	n/a	n/a	n/a	n/a	n/a	n/a	5.5	n/a
University of California-Berkeley					Assay Description A fluorometric high-throughput assay for activity against cathepsin B was performed in 96-well microtiter plates. The assay were performed in Dynate...				J Comb Chem 5: 869-80 (2003) Article DOI: 10.1021/cc034008r BindingDB Entry DOI: 10.7270/Q28914GH
University of California-Berkeley					More data for this Ligand-Target Pair
Cathepsin B (Homo sapiens (Human))	BDBM93201 (Mercaptomethyl ketone Inhibitor, 50) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	111	n/a	n/a	n/a	n/a	n/a	n/a	5.5	n/a
University of California-Berkeley					Assay Description A fluorometric high-throughput assay for activity against cathepsin B was performed in 96-well microtiter plates. The assay were performed in Dynate...				J Comb Chem 5: 869-80 (2003) Article DOI: 10.1021/cc034008r BindingDB Entry DOI: 10.7270/Q28914GH
University of California-Berkeley					More data for this Ligand-Target Pair
Cathepsin B (Homo sapiens (Human))	BDBM93200 (Mercaptomethyl ketone Inhibitor, 49) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	130	n/a	n/a	n/a	n/a	n/a	n/a	5.5	n/a
University of California-Berkeley					Assay Description A fluorometric high-throughput assay for activity against cathepsin B was performed in 96-well microtiter plates. The assay were performed in Dynate...				J Comb Chem 5: 869-80 (2003) Article DOI: 10.1021/cc034008r BindingDB Entry DOI: 10.7270/Q28914GH
University of California-Berkeley					More data for this Ligand-Target Pair
Cathepsin B (Homo sapiens (Human))	BDBM93199 (Mercaptomethyl ketone Inhibitor, 48) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	Article PubMed	140	n/a	n/a	n/a	n/a	n/a	n/a	5.5	n/a
University of California-Berkeley					Assay Description A fluorometric high-throughput assay for activity against cathepsin B was performed in 96-well microtiter plates. The assay were performed in Dynate...				J Comb Chem 5: 869-80 (2003) Article DOI: 10.1021/cc034008r BindingDB Entry DOI: 10.7270/Q28914GH
University of California-Berkeley					More data for this Ligand-Target Pair