Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50118223 (AR-C67085 | Adenosine triphosphate derivative | CH...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 4.57 | n/a | n/a | n/a | n/a | n/a |
University of Bonn Curated by ChEMBL | Assay Description Binding affinity to P2Y12 receptor expressed in human platelets from 0.047 to 50 nM | Bioorg Med Chem Lett 15: 5450-2 (2005) Article DOI: 10.1016/j.bmcl.2005.08.104 BindingDB Entry DOI: 10.7270/Q2668CR0 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
P2Y purinoceptor 12 (Homo sapiens (Human)) | BDBM50589232 (CHEMBL5199350) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | 6.5 | n/a | n/a | n/a | n/a | n/a |
TBA | Citation and Details Article DOI: 10.1016/j.bmcl.2022.128837 BindingDB Entry DOI: 10.7270/Q2765K8C | ||||||||||||
More data for this Ligand-Target Pair |