Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527464 (CHEMBL4564389) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | n/a | n/a | 129 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527492 (CHEMBL4436229) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 145 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527468 (CHEMBL4530642) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 162 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527489 (CHEMBL4567723) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 191 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50611320 (CHEMBL5277000) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | UniChem | n/a | n/a | n/a | n/a | 220 | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50384616 (CHEMBL2036813) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | n/a | n/a | n/a | n/a | 220 | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50337031 (5-ethyl-2-mercapto-3H-pyrano[2,3-d]pyrimidine-4,7-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | n/a | n/a | n/a | n/a | 220 | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50611319 (CHEMBL5281556) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | UniChem | n/a | n/a | n/a | n/a | 220 | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50611318 (CHEMBL5284951) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | UniChem | n/a | n/a | n/a | n/a | 220 | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50611316 (CHEMBL5270112) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | UniChem | n/a | n/a | n/a | n/a | 220 | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50611317 (CHEMBL5275861) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | UniChem | n/a | n/a | n/a | n/a | 220 | n/a | n/a | n/a | n/a | |
TBA | Citation and Details | ||||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527499 (CHEMBL4547569) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 245 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527501 (CHEMBL4442868) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 251 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527488 (CHEMBL4581781) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 251 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527484 (CHEMBL4584743) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 263 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Positive allosteric modulation at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527505 (CHEMBL4513816) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 288 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527498 (CHEMBL4473184) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 355 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Positive allosteric modulation at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527474 (CHEMBL4567192) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 372 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527481 (CHEMBL4560915) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 380 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Positive allosteric modulation at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527465 (CHEMBL4516265) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 398 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Positive allosteric modulation at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Rattus norvegicus) | BDBM50527468 (CHEMBL4530642) | Reactome pathway UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 407 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at rat FFA3 receptor | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Rattus norvegicus) | BDBM50527464 (CHEMBL4564389) | Reactome pathway UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | n/a | 457 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at rat FFA3 receptor | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527510 (CHEMBL4447610) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 501 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Positive allosteric modulation at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527469 (CHEMBL4448591) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 525 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527475 (CHEMBL4470184) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 525 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Positive allosteric modulation at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527469 (CHEMBL4448591) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 537 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Positive allosteric modulation at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527478 (CHEMBL4569482) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 537 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527503 (CHEMBL4567938) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 589 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Positive allosteric modulation at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527483 (CHEMBL4547759) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 603 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527508 (CHEMBL4470725) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 617 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Positive allosteric modulation at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527491 (CHEMBL4440835) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 646 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527502 (CHEMBL4515057) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 692 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Positive allosteric modulation at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527493 (CHEMBL4457531) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 692 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Positive allosteric modulation at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527463 (CHEMBL4545039) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 692 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527462 (CHEMBL4452922) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 708 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527494 (CHEMBL4443269) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 724 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Positive allosteric modulation at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527511 (CHEMBL4592426) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 871 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527486 (CHEMBL4439667) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527490 (CHEMBL4450056) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.07E+3 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527485 (CHEMBL4449702) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Mus musculus) | BDBM50527468 (CHEMBL4530642) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at mouse FFA3 receptor | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527507 (CHEMBL4476587) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527466 (CHEMBL4570341) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Positive allosteric modulation at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527493 (CHEMBL4457531) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527470 (CHEMBL4578663) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.23E+3 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Mus musculus) | BDBM50527464 (CHEMBL4564389) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.32E+3 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at mouse FFA3 receptor | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527509 (CHEMBL4574477) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.35E+3 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Rattus norvegicus) | BDBM50527469 (CHEMBL4448591) | Reactome pathway UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.35E+3 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at rat FFA3 receptor | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527484 (CHEMBL4584743) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.38E+3 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Free fatty acid receptor 3 (Homo sapiens (Human)) | BDBM50527512 (CHEMBL4471380) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.38E+3 | n/a | n/a | n/a | n/a |
University of Copenhagen Curated by ChEMBL | Assay Description Agonist activity at human FFA3 receptor stably expressed in Flp-In T-Rex HEK293 cells cotransfected with eYFP assessed as inhibition of forskolin-ind... | J Med Chem 63: 3577-3595 (2020) Article DOI: 10.1021/acs.jmedchem.9b02036 BindingDB Entry DOI: 10.7270/Q27H1P0M | |||||||||||
More data for this Ligand-Target Pair |
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