Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50560840 (CHEMBL4753103) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 0.977 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01126 BindingDB Entry DOI: 10.7270/Q2KH0S11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50560840 (CHEMBL4753103) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01126 BindingDB Entry DOI: 10.7270/Q2KH0S11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096400 (CHEMBL3577182) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096400 (CHEMBL3577182) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096458 (CHEMBL3577179) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096458 (CHEMBL3577179) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096359 (CHEMBL3577171) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096359 (CHEMBL3577171) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096360 (CHEMBL3577174) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.60 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096360 (CHEMBL3577174) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.70 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096358 (CHEMBL3577170) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.20 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096358 (CHEMBL3577170) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.20 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096503 (CHEMBL3577262) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.30 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096503 (CHEMBL3577262) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.30 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096362 (CHEMBL3577178) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.70 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096362 (CHEMBL3577178) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.70 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50560837 (CHEMBL4745025) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 5.70 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01126 BindingDB Entry DOI: 10.7270/Q2KH0S11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50560837 (CHEMBL4745025) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 5.80 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01126 BindingDB Entry DOI: 10.7270/Q2KH0S11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50177139 (CHEMBL3814492) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.60 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assay | J Med Chem 59: 3750-76 (2016) Article DOI: 10.1021/acs.jmedchem.5b01925 BindingDB Entry DOI: 10.7270/Q2542QHQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50177139 (CHEMBL3814492) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.70 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assay | J Med Chem 59: 3750-76 (2016) Article DOI: 10.1021/acs.jmedchem.5b01925 BindingDB Entry DOI: 10.7270/Q2542QHQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096441 (CHEMBL3577172) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 12 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50560845 (CHEMBL4755564) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 12 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01126 BindingDB Entry DOI: 10.7270/Q2KH0S11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096441 (CHEMBL3577172) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 12 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50560845 (CHEMBL4755564) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 12 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01126 BindingDB Entry DOI: 10.7270/Q2KH0S11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096361 (CHEMBL3577175) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 13 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096361 (CHEMBL3577175) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 13 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50177150 (CHEMBL3813843) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 17 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assay | J Med Chem 59: 3750-76 (2016) Article DOI: 10.1021/acs.jmedchem.5b01925 BindingDB Entry DOI: 10.7270/Q2542QHQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50096422 (CHEMBL3577137) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 19 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01126 BindingDB Entry DOI: 10.7270/Q2KH0S11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50096349 (CHEBI:52649 | CHEMBL1742484) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 19 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01126 BindingDB Entry DOI: 10.7270/Q2KH0S11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50096349 (CHEBI:52649 | CHEMBL1742484) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 20 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01126 BindingDB Entry DOI: 10.7270/Q2KH0S11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50096422 (CHEMBL3577137) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 20 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01126 BindingDB Entry DOI: 10.7270/Q2KH0S11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096426 (CHEMBL3577150) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 21 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096426 (CHEMBL3577150) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 21 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50096349 (CHEBI:52649 | CHEMBL1742484) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 25 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assay | J Med Chem 59: 3750-76 (2016) Article DOI: 10.1021/acs.jmedchem.5b01925 BindingDB Entry DOI: 10.7270/Q2542QHQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50096349 (CHEBI:52649 | CHEMBL1742484) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 25 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assay | J Med Chem 59: 3750-76 (2016) Article DOI: 10.1021/acs.jmedchem.5b01925 BindingDB Entry DOI: 10.7270/Q2542QHQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096422 (CHEMBL3577137) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 25 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096422 (CHEMBL3577137) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 25 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50560843 (CHEMBL4759297) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 26 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01126 BindingDB Entry DOI: 10.7270/Q2KH0S11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096353 (CHEMBL3577145) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 26 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096353 (CHEMBL3577145) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 26 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50560843 (CHEMBL4759297) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 26 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01126 BindingDB Entry DOI: 10.7270/Q2KH0S11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096349 (CHEBI:52649 | CHEMBL1742484) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 28 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096349 (CHEBI:52649 | CHEMBL1742484) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 28 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096478 (CHEMBL3577180) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 32 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096478 (CHEMBL3577180) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 33 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50560822 (CHEMBL4764512) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 37 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01126 BindingDB Entry DOI: 10.7270/Q2KH0S11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50560822 (CHEMBL4764512) | UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 37 | n/a | n/a | n/a | n/a |
TBA | Assay Description Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ... | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c01126 BindingDB Entry DOI: 10.7270/Q2KH0S11 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096350 (CHEMBL3577138) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 39 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Homo sapiens (Human)) | BDBM50096350 (CHEMBL3577138) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 39 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assay | J Med Chem 58: 4204-19 (2015) Article DOI: 10.1021/jm5020082 BindingDB Entry DOI: 10.7270/Q2Q81FTD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Putative P2Y purinoceptor 10 (Mus musculus) | BDBM50177142 (CHEMBL3813751) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 42 | n/a | n/a | n/a | n/a |
The University of Tokyo Curated by ChEMBL | Assay Description Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assay | J Med Chem 59: 3750-76 (2016) Article DOI: 10.1021/acs.jmedchem.5b01925 BindingDB Entry DOI: 10.7270/Q2542QHQ | |||||||||||
More data for this Ligand-Target Pair |
Displayed 1 to 50 (of 202 total ) | Next | Last >> |