BindingDB logo
myBDB logout

Patent code US8492568

Compile Data Set for Download or QSAR
Found 1 hit of Enzyme Inhibition Constant Data   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Transient receptor potential cation channel subfamily V member 3


(Homo sapiens (Human))		BDBM98548
PNG
(US8492568, 2)
Show SMILES COc1cccc(CNC(=O)CC2CC3(CCC3)Oc3ccc(Cl)cc23)c1OC1CCCC1
Show InChI InChI=1S/C27H32ClNO4/c1-31-24-9-4-6-18(26(24)32-21-7-2-3-8-21)17-29-25(30)14-19-16-27(12-5-13-27)33-23-11-10-20(28)15-22(19)23/h4,6,9-11,15,19,21H,2-3,5,7-8,12-14,16-17H2,1H3,(H,29,30)
PDB

Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 725n/an/an/an/an/an/a



Glenmark Pharamceuticals S.A.

US Patent


Assay Description
Calcium uptake assay: The inhibition of TRPV3 receptor activation was followed as inhibition of 2-aminoethoxydiphenylborate (2-APB) induced cellular...

US Patent US8492568 (2013)


BindingDB Entry DOI: 10.7270/Q2J38R50
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%