Affinity Data by Patent

Patent code US8927536

Found 14 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
11-beta-hydroxysteroid dehydrogenase 1 (Homo sapiens (Human))	BDBM142001 (US8927536, 26) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	0.300	n/a	n/a	n/a	n/a	7.4	25
Daiichi Sankyo Company, Limited US Patent					Assay Description A reaction was performed on a 384-well plate (Greiner Bio One) using a reaction volume of 24 �L, and all the samples were diluted with an assay buffe...				US Patent US8927536 (2015) BindingDB Entry DOI: 10.7270/Q2Q23XZP
Daiichi Sankyo Company, Limited US Patent					More data for this Ligand-Target Pair
11-beta-hydroxysteroid dehydrogenase 1 (Homo sapiens (Human))	BDBM142003 (US8927536, 34) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	1	n/a	n/a	n/a	n/a	7.4	25
Daiichi Sankyo Company, Limited US Patent					Assay Description A reaction was performed on a 384-well plate (Greiner Bio One) using a reaction volume of 24 �L, and all the samples were diluted with an assay buffe...				US Patent US8927536 (2015) BindingDB Entry DOI: 10.7270/Q2Q23XZP
Daiichi Sankyo Company, Limited US Patent					More data for this Ligand-Target Pair
11-beta-hydroxysteroid dehydrogenase 1 (Homo sapiens (Human))	BDBM142008 (US8927536, 89) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.30	n/a	n/a	n/a	n/a	7.4	25
Daiichi Sankyo Company, Limited US Patent					Assay Description A reaction was performed on a 384-well plate (Greiner Bio One) using a reaction volume of 24 �L, and all the samples were diluted with an assay buffe...				US Patent US8927536 (2015) BindingDB Entry DOI: 10.7270/Q2Q23XZP
Daiichi Sankyo Company, Limited US Patent					More data for this Ligand-Target Pair
11-beta-hydroxysteroid dehydrogenase 1 (Homo sapiens (Human))	BDBM141998 (US8927536, 4) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	1.30	n/a	n/a	n/a	n/a	7.4	25
Daiichi Sankyo Company, Limited US Patent					Assay Description A reaction was performed on a 384-well plate (Greiner Bio One) using a reaction volume of 24 �L, and all the samples were diluted with an assay buffe...				US Patent US8927536 (2015) BindingDB Entry DOI: 10.7270/Q2Q23XZP
Daiichi Sankyo Company, Limited US Patent					More data for this Ligand-Target Pair
11-beta-hydroxysteroid dehydrogenase 1 (Homo sapiens (Human))	BDBM142007 (US8927536, 88) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	1.70	n/a	n/a	n/a	n/a	7.4	25
Daiichi Sankyo Company, Limited US Patent					Assay Description A reaction was performed on a 384-well plate (Greiner Bio One) using a reaction volume of 24 �L, and all the samples were diluted with an assay buffe...				US Patent US8927536 (2015) BindingDB Entry DOI: 10.7270/Q2Q23XZP
Daiichi Sankyo Company, Limited US Patent					More data for this Ligand-Target Pair
11-beta-hydroxysteroid dehydrogenase 1 (Homo sapiens (Human))	BDBM142000 (US8927536, 9) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	1.80	n/a	n/a	n/a	n/a	7.4	25
Daiichi Sankyo Company, Limited US Patent					Assay Description A reaction was performed on a 384-well plate (Greiner Bio One) using a reaction volume of 24 �L, and all the samples were diluted with an assay buffe...				US Patent US8927536 (2015) BindingDB Entry DOI: 10.7270/Q2Q23XZP
Daiichi Sankyo Company, Limited US Patent					More data for this Ligand-Target Pair
11-beta-hydroxysteroid dehydrogenase 1 (Homo sapiens (Human))	BDBM142002 (US8927536, 32) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	2	n/a	n/a	n/a	n/a	7.4	25
Daiichi Sankyo Company, Limited US Patent					Assay Description A reaction was performed on a 384-well plate (Greiner Bio One) using a reaction volume of 24 �L, and all the samples were diluted with an assay buffe...				US Patent US8927536 (2015) BindingDB Entry DOI: 10.7270/Q2Q23XZP
Daiichi Sankyo Company, Limited US Patent					More data for this Ligand-Target Pair
11-beta-hydroxysteroid dehydrogenase 1 (Homo sapiens (Human))	BDBM142006 (US8927536, 81) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	2.20	n/a	n/a	n/a	n/a	7.4	25
Daiichi Sankyo Company, Limited US Patent					Assay Description A reaction was performed on a 384-well plate (Greiner Bio One) using a reaction volume of 24 �L, and all the samples were diluted with an assay buffe...				US Patent US8927536 (2015) BindingDB Entry DOI: 10.7270/Q2Q23XZP
Daiichi Sankyo Company, Limited US Patent					More data for this Ligand-Target Pair
11-beta-hydroxysteroid dehydrogenase 1 (Homo sapiens (Human))	BDBM141996 (US8927536, 2) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	2.60	n/a	n/a	n/a	n/a	7.4	25
Daiichi Sankyo Company, Limited US Patent					Assay Description A reaction was performed on a 384-well plate (Greiner Bio One) using a reaction volume of 24 �L, and all the samples were diluted with an assay buffe...				US Patent US8927536 (2015) BindingDB Entry DOI: 10.7270/Q2Q23XZP
Daiichi Sankyo Company, Limited US Patent					More data for this Ligand-Target Pair
11-beta-hydroxysteroid dehydrogenase 1 (Homo sapiens (Human))	BDBM141999 (US8927536, 6) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	2.60	n/a	n/a	n/a	n/a	7.4	25
Daiichi Sankyo Company, Limited US Patent					Assay Description A reaction was performed on a 384-well plate (Greiner Bio One) using a reaction volume of 24 �L, and all the samples were diluted with an assay buffe...				US Patent US8927536 (2015) BindingDB Entry DOI: 10.7270/Q2Q23XZP
Daiichi Sankyo Company, Limited US Patent					More data for this Ligand-Target Pair
11-beta-hydroxysteroid dehydrogenase 1 (Homo sapiens (Human))	BDBM141995 (US8927536, 1) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	3.30	n/a	n/a	n/a	n/a	7.4	25
Daiichi Sankyo Company, Limited US Patent					Assay Description A reaction was performed on a 384-well plate (Greiner Bio One) using a reaction volume of 24 �L, and all the samples were diluted with an assay buffe...				US Patent US8927536 (2015) BindingDB Entry DOI: 10.7270/Q2Q23XZP
Daiichi Sankyo Company, Limited US Patent					More data for this Ligand-Target Pair
11-beta-hydroxysteroid dehydrogenase 1 (Homo sapiens (Human))	BDBM142004 (US8927536, 67) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	5.40	n/a	n/a	n/a	n/a	7.4	25
Daiichi Sankyo Company, Limited US Patent					Assay Description A reaction was performed on a 384-well plate (Greiner Bio One) using a reaction volume of 24 �L, and all the samples were diluted with an assay buffe...				US Patent US8927536 (2015) BindingDB Entry DOI: 10.7270/Q2Q23XZP
Daiichi Sankyo Company, Limited US Patent					More data for this Ligand-Target Pair
11-beta-hydroxysteroid dehydrogenase 1 (Homo sapiens (Human))	BDBM141997 (US8927536, 3) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	6.30	n/a	n/a	n/a	n/a	7.4	25
Daiichi Sankyo Company, Limited US Patent					Assay Description A reaction was performed on a 384-well plate (Greiner Bio One) using a reaction volume of 24 �L, and all the samples were diluted with an assay buffe...				US Patent US8927536 (2015) BindingDB Entry DOI: 10.7270/Q2Q23XZP
Daiichi Sankyo Company, Limited US Patent					More data for this Ligand-Target Pair
11-beta-hydroxysteroid dehydrogenase 1 (Homo sapiens (Human))	BDBM142005 (US8927536, 68) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem Similars	US Patent	n/a	n/a	6.70	n/a	n/a	n/a	n/a	7.4	25
Daiichi Sankyo Company, Limited US Patent					Assay Description A reaction was performed on a 384-well plate (Greiner Bio One) using a reaction volume of 24 �L, and all the samples were diluted with an assay buffe...				US Patent US8927536 (2015) BindingDB Entry DOI: 10.7270/Q2Q23XZP
Daiichi Sankyo Company, Limited US Patent					More data for this Ligand-Target Pair

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* indicates data uncertainty>20%