Affinity Data by Patent

Patent code US9242982

Found 7 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B (Homo sapiens (Human))	BDBM203459 (US9242982, 1k) Show SMILES Show InChI	PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	4.80	n/a	n/a	n/a	n/a	n/a	22
COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH US Patent					Assay Description PDE3 inhibition assay was performed a BIOMOL GREEN Quantizyme Assay System (catalogue No. BML-AK800-0001). The Platelets isolated from human blood ...				US Patent US9242982 (2016) BindingDB Entry DOI: 10.7270/Q2BV7FF6
COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH US Patent					More data for this Ligand-Target Pair
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B (Homo sapiens (Human))	BDBM203457 (US9242982, 1i) Show SMILES Show InChI	PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	6.60	n/a	n/a	n/a	n/a	n/a	22
COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH US Patent					Assay Description PDE3 inhibition assay was performed a BIOMOL GREEN Quantizyme Assay System (catalogue No. BML-AK800-0001). The Platelets isolated from human blood ...				US Patent US9242982 (2016) BindingDB Entry DOI: 10.7270/Q2BV7FF6
COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH US Patent					More data for this Ligand-Target Pair
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B (Homo sapiens (Human))	BDBM203455 (US9242982, 1g) Show SMILES Show InChI	PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	12.5	n/a	n/a	n/a	n/a	n/a	22
COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH US Patent					Assay Description PDE3 inhibition assay was performed a BIOMOL GREEN Quantizyme Assay System (catalogue No. BML-AK800-0001). The Platelets isolated from human blood ...				US Patent US9242982 (2016) BindingDB Entry DOI: 10.7270/Q2BV7FF6
COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH US Patent					More data for this Ligand-Target Pair
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B (Homo sapiens (Human))	BDBM203451 (US9242982, 1c) Show SMILES Show InChI	PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	32.3	n/a	n/a	n/a	n/a	n/a	22
COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH US Patent					Assay Description PDE3 inhibition assay was performed a BIOMOL GREEN Quantizyme Assay System (catalogue No. BML-AK800-0001). The Platelets isolated from human blood ...				US Patent US9242982 (2016) BindingDB Entry DOI: 10.7270/Q2BV7FF6
COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH US Patent					More data for this Ligand-Target Pair
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B (Homo sapiens (Human))	BDBM203450 (US9242982, 1b) Show SMILES Show InChI	PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	48.8	n/a	n/a	n/a	n/a	n/a	22
COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH US Patent					Assay Description PDE3 inhibition assay was performed a BIOMOL GREEN Quantizyme Assay System (catalogue No. BML-AK800-0001). The Platelets isolated from human blood ...				US Patent US9242982 (2016) BindingDB Entry DOI: 10.7270/Q2BV7FF6
COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH US Patent					More data for this Ligand-Target Pair
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B (Homo sapiens (Human))	BDBM15296 (6-methyl-2-oxo-5-(pyridin-4-yl)-1,2-dihydropyridin...) Show SMILES Cc1[nH]c(=O)c(cc1-c1ccncc1)C#N Show InChI	PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	US Patent	n/a	n/a	3.30E+3	n/a	n/a	n/a	n/a	n/a	22
COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH US Patent					Assay Description PDE3 inhibition assay was performed a BIOMOL GREEN Quantizyme Assay System (catalogue No. BML-AK800-0001). The Platelets isolated from human blood ...				US Patent US9242982 (2016) BindingDB Entry DOI: 10.7270/Q2BV7FF6
COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH US Patent					More data for this Ligand-Target Pair
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B (Homo sapiens (Human))	BDBM203449 (US9242982, 1a) Show SMILES Show InChI	PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.18E+4	n/a	n/a	n/a	n/a	n/a	22
COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH US Patent					Assay Description PDE3 inhibition assay was performed a BIOMOL GREEN Quantizyme Assay System (catalogue No. BML-AK800-0001). The Platelets isolated from human blood ...				US Patent US9242982 (2016) BindingDB Entry DOI: 10.7270/Q2BV7FF6
COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH US Patent					More data for this Ligand-Target Pair

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* indicates data uncertainty>20%