Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Protein mono-ADP-ribosyltransferase PARP3 [R100H] (355/355 = 100%)† (Homo sapiens (Human)) | BDBM50226518 (3-Aminobenzoesaeure | 3-aminobenzoic acid | CHEMBL...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | n/a | n/a | n/a | >2.00E+3 | n/a | n/a | n/a | n/a | n/a |
Institutet Curated by ChEMBL | Assay Description Binding affinity to human PARP3 PARP domain by isothermal titration colorimetry | J Med Chem 52: 3108-11 (2009) Article DOI: 10.1021/jm900052j BindingDB Entry DOI: 10.7270/Q2B56JNV | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |