Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50039029 ((+)-4-((alpha R)-((2S,5R)-4-allyl-2,5-dimethylpipe...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | 1.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Inhibitory activity against Opioid receptor delta 1 in rat brain membranes using [3H]-DADLE as a radioligand. | J Med Chem 43: 3193-6 (2000) BindingDB Entry DOI: 10.7270/Q21835RR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50091224 (4-[(4-But-2-enyl-2,5-dimethyl-piperazin-1-yl)-(3-m...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1 | J Med Chem 43: 3193-6 (2000) BindingDB Entry DOI: 10.7270/Q21835RR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50091221 (4-[(4-Butyl-2,5-dimethyl-piperazin-1-yl)-(3-methox...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1 | J Med Chem 43: 3193-6 (2000) BindingDB Entry DOI: 10.7270/Q21835RR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50091223 (4-[(4-Cyclopropylmethyl-2,5-dimethyl-piperazin-1-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 3.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1 | J Med Chem 43: 3193-6 (2000) BindingDB Entry DOI: 10.7270/Q21835RR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50091226 (CHEMBL323733 | N,N-Diethyl-4-[(3-methoxy-phenyl)-(...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 4.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1 | J Med Chem 43: 3193-6 (2000) BindingDB Entry DOI: 10.7270/Q21835RR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50091225 (4-[(2,5-Dimethyl-4-pentyl-piperazin-1-yl)-(3-metho...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 4.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1 | J Med Chem 43: 3193-6 (2000) BindingDB Entry DOI: 10.7270/Q21835RR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50091217 (4-[(2,5-Dimethyl-piperazin-1-yl)-(3-methoxy-phenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 4.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1 | J Med Chem 43: 3193-6 (2000) BindingDB Entry DOI: 10.7270/Q21835RR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50091219 (4-[[2,5-Dimethyl-4-(2-methyl-allyl)-piperazin-1-yl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 4.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1 | J Med Chem 43: 3193-6 (2000) BindingDB Entry DOI: 10.7270/Q21835RR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50091222 (CHEMBL111389 | N,N-Diethyl-4-[(4-ethyl-2,5-dimethy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 5.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1 | J Med Chem 43: 3193-6 (2000) BindingDB Entry DOI: 10.7270/Q21835RR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50091218 (4-[(4-Benzyl-2,5-dimethyl-piperazin-1-yl)-(3-metho...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 6.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1 | J Med Chem 43: 3193-6 (2000) BindingDB Entry DOI: 10.7270/Q21835RR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50091216 (CHEMBL321927 | N,N-Diethyl-4-[(4-hexyl-2,5-dimethy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 10.4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1 | J Med Chem 43: 3193-6 (2000) BindingDB Entry DOI: 10.7270/Q21835RR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50091220 (4-[[2,5-Dimethyl-4-(3-phenyl-propyl)-piperazin-1-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 16.7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1 | J Med Chem 43: 3193-6 (2000) BindingDB Entry DOI: 10.7270/Q21835RR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Rattus norvegicus (rat)) | BDBM50091215 (4-[(2,5-Dimethyl-4-phenethyl-piperazin-1-yl)-(3-me...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 30.6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1 | J Med Chem 43: 3193-6 (2000) BindingDB Entry DOI: 10.7270/Q21835RR | |||||||||||
More data for this Ligand-Target Pair |