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PubMed code 11327594

Compile data set for download or QSAR
Found 26 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099023
PNG
(CHEMBL11149 | N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCCc1ccc(NS(C)(=O)=O)cc1
Show InChI InChI=1S/C29H35N3O2S/c1-21-18-22(2)20-24(19-21)29-27(26-9-4-5-10-28(26)31-29)15-17-30-16-7-6-8-23-11-13-25(14-12-23)32-35(3,33)34/h4-5,9-14,18-20,30-32H,6-8,15-17H2,1-3H3
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Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099036
PNG
(CHEMBL11009 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCCc1ccncc1
Show InChI InChI=1S/C27H31N3/c1-20-17-21(2)19-23(18-20)27-25(24-8-3-4-9-26(24)30-27)12-16-28-13-6-5-7-22-10-14-29-15-11-22/h3-4,8-11,14-15,17-19,28,30H,5-7,12-13,16H2,1-2H3
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Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50097007
PNG
(4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCCc1ccc(O)cc1
Show InChI InChI=1S/C28H32N2O/c1-20-17-21(2)19-23(18-20)28-26(25-8-3-4-9-27(25)30-28)14-16-29-15-6-5-7-22-10-12-24(31)13-11-22/h3-4,8-13,17-19,29-31H,5-7,14-16H2,1-2H3
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Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099041
PNG
(CHEMBL11014 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCCc1cnc2ccccc2c1
Show InChI InChI=1S/C31H33N3/c1-22-17-23(2)19-26(18-22)31-28(27-11-4-6-13-30(27)34-31)14-16-32-15-8-7-9-24-20-25-10-3-5-12-29(25)33-21-24/h3-6,10-13,17-21,32,34H,7-9,14-16H2,1-2H3
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Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099033
PNG
(CHEMBL262715 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indo...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCCc1cccnc1
Show InChI InChI=1S/C27H31N3/c1-20-16-21(2)18-23(17-20)27-25(24-10-3-4-11-26(24)30-27)12-15-28-13-6-5-8-22-9-7-14-29-19-22/h3-4,7,9-11,14,16-19,28,30H,5-6,8,12-13,15H2,1-2H3
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Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099051
PNG
(5-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCCc1ccc(N)nc1
Show InChI InChI=1S/C27H32N4/c1-19-15-20(2)17-22(16-19)27-24(23-8-3-4-9-25(23)31-27)12-14-29-13-6-5-7-21-10-11-26(28)30-18-21/h3-4,8-11,15-18,29,31H,5-7,12-14H2,1-2H3,(H2,28,30)
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Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099045
PNG
(CHEMBL273625 | N-[5-(4-{2-[2-(3,5-Dimethyl-phenyl)...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCCc1ccc(NS(C)(=O)=O)nc1
Show InChI InChI=1S/C28H34N4O2S/c1-20-16-21(2)18-23(17-20)28-25(24-9-4-5-10-26(24)31-28)13-15-29-14-7-6-8-22-11-12-27(30-19-22)32-35(3,33)34/h4-5,9-12,16-19,29,31H,6-8,13-15H2,1-3H3,(H,30,32)
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Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099043
PNG
(CHEMBL11253 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCCCc1cccnc1
Show InChI InChI=1S/C28H33N3/c1-21-17-22(2)19-24(18-21)28-26(25-11-5-6-12-27(25)31-28)13-16-29-14-7-3-4-9-23-10-8-15-30-20-23/h5-6,8,10-12,15,17-20,29,31H,3-4,7,9,13-14,16H2,1-2H3
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Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099046
PNG
(5-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCCc1ccc(=O)[nH]c1
Show InChI InChI=1S/C27H31N3O/c1-19-15-20(2)17-22(16-19)27-24(23-8-3-4-9-25(23)30-27)12-14-28-13-6-5-7-21-10-11-26(31)29-18-21/h3-4,8-11,15-18,28,30H,5-7,12-14H2,1-2H3,(H,29,31)
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Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099040
PNG
(CHEMBL11310 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Show SMILES COc1ccc(CCCCNCCc2c([nH]c3ccccc23)-c2cc(C)cc(C)c2)cn1
Show InChI InChI=1S/C28H33N3O/c1-20-16-21(2)18-23(17-20)28-25(24-9-4-5-10-26(24)31-28)13-15-29-14-7-6-8-22-11-12-27(32-3)30-19-22/h4-5,9-12,16-19,29,31H,6-8,13-15H2,1-3H3
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Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099030
PNG
(CHEMBL11263 | N-[5-(4-{2-[2-(3,5-Dimethyl-phenyl)-...)
Show SMILES CC(=O)Nc1ccc(CCCCNCCc2c([nH]c3ccccc23)-c2cc(C)cc(C)c2)cn1
Show InChI InChI=1S/C29H34N4O/c1-20-16-21(2)18-24(17-20)29-26(25-9-4-5-10-27(25)33-29)13-15-30-14-7-6-8-23-11-12-28(31-19-23)32-22(3)34/h4-5,9-12,16-19,30,33H,6-8,13-15H2,1-3H3,(H,31,32,34)
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Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099050
PNG
(CHEMBL11420 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCCCc1ccncc1
Show InChI InChI=1S/C28H33N3/c1-21-18-22(2)20-24(19-21)28-26(25-9-5-6-10-27(25)31-28)13-17-29-14-7-3-4-8-23-11-15-30-16-12-23/h5-6,9-12,15-16,18-20,29,31H,3-4,7-8,13-14,17H2,1-2H3
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Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099042
PNG
(CHEMBL275287 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indo...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCc1ccncc1
Show InChI InChI=1S/C25H27N3/c1-18-15-19(2)17-21(16-18)25-23(22-5-3-4-6-24(22)28-25)10-14-27-13-9-20-7-11-26-12-8-20/h3-8,11-12,15-17,27-28H,9-10,13-14H2,1-2H3
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Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Homo sapiens (Human))		BDBM50099023
PNG
(CHEMBL11149 | N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCCc1ccc(NS(C)(=O)=O)cc1
Show InChI InChI=1S/C29H35N3O2S/c1-21-18-22(2)20-24(19-21)29-27(26-9-4-5-10-28(26)31-29)15-17-30-16-7-6-8-23-11-13-25(14-12-23)32-35(3,33)34/h4-5,9-14,18-20,30-32H,6-8,15-17H2,1-3H3
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Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibitory activity of the compound evaluated against human Gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099034
PNG
(CHEMBL11021 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCc1cccnc1
Show InChI InChI=1S/C26H29N3/c1-19-15-20(2)17-22(16-19)26-24(23-9-3-4-10-25(23)29-26)11-14-27-12-5-7-21-8-6-13-28-18-21/h3-4,6,8-10,13,15-18,27,29H,5,7,11-12,14H2,1-2H3
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Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099048
PNG
(CHEMBL11436 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCc1cccnc1
Show InChI InChI=1S/C25H27N3/c1-18-14-19(2)16-21(15-18)25-23(22-7-3-4-8-24(22)28-25)10-13-26-12-9-20-6-5-11-27-17-20/h3-8,11,14-17,26,28H,9-10,12-13H2,1-2H3
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Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099032
PNG
(CHEMBL273725 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indo...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCc1ccncc1
Show InChI InChI=1S/C26H29N3/c1-19-16-20(2)18-22(17-19)26-24(23-7-3-4-8-25(23)29-26)11-15-27-12-5-6-21-9-13-28-14-10-21/h3-4,7-10,13-14,16-18,27,29H,5-6,11-12,15H2,1-2H3
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Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099037
PNG
(CHEMBL275920 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indo...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCCc1cncnc1
Show InChI InChI=1S/C26H30N4/c1-19-13-20(2)15-22(14-19)26-24(23-8-3-4-9-25(23)30-26)10-12-27-11-6-5-7-21-16-28-18-29-17-21/h3-4,8-9,13-18,27,30H,5-7,10-12H2,1-2H3
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Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Homo sapiens (Human))		BDBM50097007
PNG
(4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCCc1ccc(O)cc1
Show InChI InChI=1S/C28H32N2O/c1-20-17-21(2)19-23(18-20)28-26(25-8-3-4-9-27(25)30-28)14-16-29-15-6-5-7-22-10-12-24(31)13-11-22/h3-4,8-13,17-19,29-31H,5-7,14-16H2,1-2H3
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Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibitory activity of the compound evaluated against human Gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099039
PNG
(CHEMBL11087 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCCc1ccccn1
Show InChI InChI=1S/C27H31N3/c1-20-17-21(2)19-22(18-20)27-25(24-11-3-4-12-26(24)30-27)13-16-28-14-7-5-9-23-10-6-8-15-29-23/h3-4,6,8,10-12,15,17-19,28,30H,5,7,9,13-14,16H2,1-2H3
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Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099044
PNG
(CHEMBL11375 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCCc1cnc[nH]1
Show InChI InChI=1S/C25H30N4/c1-18-13-19(2)15-20(14-18)25-23(22-8-3-4-9-24(22)29-25)10-12-26-11-6-5-7-21-16-27-17-28-21/h3-4,8-9,13-17,26,29H,5-7,10-12H2,1-2H3,(H,27,28)
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n/an/a 450n/an/an/an/an/an/a



Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099038
PNG
(CHEMBL11623 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCCCc1ccc2CCCCc2c1
Show InChI InChI=1S/C32H38N2/c1-23-19-24(2)21-28(20-23)32-30(29-12-5-6-13-31(29)34-32)16-18-33-17-8-7-9-25-14-15-26-10-3-4-11-27(26)22-25/h5-6,12-15,19-22,33-34H,3-4,7-11,16-18H2,1-2H3
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n/an/a 1.26E+3n/an/an/an/an/an/a



Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099035
PNG
(CHEMBL269636 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indo...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCCc1ccccn1
Show InChI InChI=1S/C25H27N3/c1-18-15-19(2)17-20(16-18)25-23(22-8-3-4-9-24(22)28-25)11-14-26-13-10-21-7-5-6-12-27-21/h3-9,12,15-17,26,28H,10-11,13-14H2,1-2H3
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n/an/a 2.17E+3n/an/an/an/an/an/a



Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099047
PNG
(CHEMBL11523 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCc1cccnc1
Show InChI InChI=1S/C24H25N3/c1-17-12-18(2)14-20(13-17)24-22(21-7-3-4-8-23(21)27-24)9-11-26-16-19-6-5-10-25-15-19/h3-8,10,12-15,26-27H,9,11,16H2,1-2H3
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n/an/a 4.50E+3n/an/an/an/an/an/a



Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099049
PNG
(CHEMBL11134 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCc1ccncc1
Show InChI InChI=1S/C24H25N3/c1-17-13-18(2)15-20(14-17)24-22(21-5-3-4-6-23(21)27-24)9-12-26-16-19-7-10-25-11-8-19/h3-8,10-11,13-15,26-27H,9,12,16H2,1-2H3
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n/an/a 9.00E+3n/an/an/an/an/an/a



Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
Gonadotropin-releasing hormone receptor


(Rattus norvegicus)		BDBM50099031
PNG
(CHEMBL274441 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indo...)
Show SMILES Cc1cc(C)cc(c1)-c1[nH]c2ccccc2c1CCNCc1ccccn1
Show InChI InChI=1S/C24H25N3/c1-17-13-18(2)15-19(14-17)24-22(21-8-3-4-9-23(21)27-24)10-12-25-16-20-7-5-6-11-26-20/h3-9,11,13-15,25,27H,10,12,16H2,1-2H3
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n/an/a>1.00E+4n/an/an/an/an/an/a



Merck Research Laboratories

Curated by ChEMBL


Assay Description
Inhibition of rat gonadotropin-releasing hormone receptor

Bioorg Med Chem Lett 11: 1077-80 (2001)


BindingDB Entry DOI: 10.7270/Q2J102FK
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%