Found 29 hits of Enzyme Inhibition Constant Data Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223118
(CHEMBL31530)Show InChI InChI=1S/C16H23N3S/c1-2-3-9-14-18-13-10-11-20-15(13)16(19-14)17-12-7-5-4-6-8-12/h10-12H,2-9H2,1H3,(H,17,18,19) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet 
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 400 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223120
(CHEMBL31063)Show InChI InChI=1S/C14H19N3S/c1-2-3-6-12-15-11-7-10-18-13(11)14(16-12)17-8-4-5-9-17/h7,10H,2-6,8-9H2,1H3 | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223132
(CHEMBL30619)Show InChI InChI=1S/C18H14N4S/c1-2-5-13(6-3-1)11-20-18-16-15(8-10-23-16)21-17(22-18)14-7-4-9-19-12-14/h1-10,12H,11H2,(H,20,21,22) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223052
(CHEMBL30733)Show InChI InChI=1S/C16H17N3S/c1-2-3-9-14-18-13-10-11-20-15(13)16(19-14)17-12-7-5-4-6-8-12/h4-8,10-11H,2-3,9H2,1H3,(H,17,18,19) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223053
(CHEMBL30406)Show InChI InChI=1S/C16H18N4S/c1-2-3-4-14-19-13-7-10-21-15(13)16(20-14)18-11-12-5-8-17-9-6-12/h5-10H,2-4,11H2,1H3,(H,18,19,20) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 600 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223054
(CHEMBL434590)Show InChI InChI=1S/C18H21N3OS/c1-3-4-9-16-20-14-10-11-23-17(14)18(21-16)19-12-13-7-5-6-8-15(13)22-2/h5-8,10-11H,3-4,9,12H2,1-2H3,(H,19,20,21) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 700 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223189
(CHEMBL288545)Show InChI InChI=1S/C18H21N3S/c1-3-4-10-16-19-15-11-12-22-17(15)18(20-16)21(2)13-14-8-6-5-7-9-14/h5-9,11-12H,3-4,10,13H2,1-2H3 | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 800 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223121
(CHEMBL281244)Show SMILES CCCCc1nc(NCc2cccc(c2)[N+]([O-])=O)c2sccc2n1 Show InChI InChI=1S/C17H18N4O2S/c1-2-3-7-15-19-14-8-9-24-16(14)17(20-15)18-11-12-5-4-6-13(10-12)21(22)23/h4-6,8-10H,2-3,7,11H2,1H3,(H,18,19,20) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 840 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223129
(CHEMBL30379)Show InChI InChI=1S/C17H19N3S/c1-2-3-9-15-19-14-10-11-21-16(14)17(20-15)18-12-13-7-5-4-6-8-13/h4-8,10-11H,2-3,9,12H2,1H3,(H,18,19,20) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 900 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223125
(CHEMBL30407)Show InChI InChI=1S/C17H17F2N3S/c1-2-3-7-15-21-14-8-9-23-16(14)17(22-15)20-10-11-12(18)5-4-6-13(11)19/h4-6,8-9H,2-3,7,10H2,1H3,(H,20,21,22) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223099
(CHEMBL288547)Show InChI InChI=1S/C17H18N4O2S/c1-2-3-8-15-19-13-9-10-24-16(13)17(20-15)18-11-12-6-4-5-7-14(12)21(22)23/h4-7,9-10H,2-3,8,11H2,1H3,(H,18,19,20) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
| PubMed
| n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223055
(CHEMBL31439)Show InChI InChI=1S/C17H25N3S/c1-2-3-9-15-19-14-10-11-21-16(14)17(20-15)18-12-13-7-5-4-6-8-13/h10-11,13H,2-9,12H2,1H3,(H,18,19,20) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
| PubMed
| n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223187
(CHEMBL30966)Show InChI InChI=1S/C19H21N3S/c1-2-8-15(9-3-1)13-20-19-18-16(10-11-23-18)21-17(22-19)12-14-6-4-5-7-14/h1-3,8-11,14H,4-7,12-13H2,(H,20,21,22) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223122
(CHEMBL31035)Show InChI InChI=1S/C17H19N3O/c1-2-3-9-15-19-14-10-11-21-16(14)17(20-15)18-12-13-7-5-4-6-8-13/h4-8,10-11H,2-3,9,12H2,1H3,(H,18,19,20) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223051
(CHEMBL31390)Show InChI InChI=1S/C19H16N4S/c1-2-4-15(5-3-1)13-21-19-18-16(8-11-24-18)22-17(23-19)12-14-6-9-20-10-7-14/h1-11H,12-13H2,(H,21,22,23) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223097
(CHEMBL28562)Show InChI InChI=1S/C18H21N3OS/c1-3-4-8-16-20-15-9-10-23-17(15)18(21-16)19-12-13-6-5-7-14(11-13)22-2/h5-7,9-11H,3-4,8,12H2,1-2H3,(H,19,20,21) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
| PubMed
| n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223126
(CHEMBL31715)Show InChI InChI=1S/C18H21N3OS/c1-3-4-5-16-20-15-10-11-23-17(15)18(21-16)19-12-13-6-8-14(22-2)9-7-13/h6-11H,3-5,12H2,1-2H3,(H,19,20,21) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223188
(CHEMBL30941)Show InChI InChI=1S/C20H17N3S/c1-3-7-15(8-4-1)13-18-22-17-11-12-24-19(17)20(23-18)21-14-16-9-5-2-6-10-16/h1-12H,13-14H2,(H,21,22,23) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223050
(CHEMBL31157)Show InChI InChI=1S/C17H19N3S/c1-3-12(2)16-19-14-9-10-21-15(14)17(20-16)18-11-13-7-5-4-6-8-13/h4-10,12H,3,11H2,1-2H3,(H,18,19,20) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223127
(CHEMBL32673)Show InChI InChI=1S/C21H19N3S/c1-3-7-16(8-4-1)11-12-19-23-18-13-14-25-20(18)21(24-19)22-15-17-9-5-2-6-10-17/h1-10,13-14H,11-12,15H2,(H,22,23,24) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223130
(CHEMBL30671)Show InChI InChI=1S/C15H15N3S/c1-2-13-17-12-8-9-19-14(12)15(18-13)16-10-11-6-4-3-5-7-11/h3-9H,2,10H2,1H3,(H,16,17,18) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223133
(CHEMBL31305)Show InChI InChI=1S/C20H25N3S/c1-3-5-11-18-21-17-12-14-24-19(17)20(22-18)23(13-4-2)15-16-9-7-6-8-10-16/h6-10,12,14H,3-5,11,13,15H2,1-2H3 | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223162
(CHEMBL31743)Show InChI InChI=1S/C19H21N3S/c1-2-3-8-17-20-16-10-12-23-18(16)19(21-17)22-11-9-14-6-4-5-7-15(14)13-22/h4-7,10,12H,2-3,8-9,11,13H2,1H3 | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| PubMed
| n/a | n/a | 2.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223131
(CHEMBL435363)Show InChI InChI=1S/C19H15N3S/c1-3-7-14(8-4-1)13-20-19-17-16(11-12-23-17)21-18(22-19)15-9-5-2-6-10-15/h1-12H,13H2,(H,20,21,22) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223124
(CHEMBL31773)Show InChI InChI=1S/C24H25N3S/c1-2-3-14-22-25-21-15-16-28-23(21)24(26-22)27(17-19-10-6-4-7-11-19)18-20-12-8-5-9-13-20/h4-13,15-16H,2-3,14,17-18H2,1H3 | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223128
(CHEMBL31795)Show InChI InChI=1S/C20H23N3S/c1-3-7-15(8-4-1)13-18-22-17-11-12-24-19(17)20(23-18)21-14-16-9-5-2-6-10-16/h2,5-6,9-12,15H,1,3-4,7-8,13-14H2,(H,21,22,23) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223119
(CHEMBL30879)Show InChI InChI=1S/C23H23N3OS/c1-3-9-18(10-4-1)17-24-23-22-20(14-16-28-22)25-21(26-23)13-7-8-15-27-19-11-5-2-6-12-19/h1-6,9-12,14,16H,7-8,13,15,17H2,(H,24,25,26) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 4.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223123
(CHEMBL31877)Show InChI InChI=1S/C13H11N3S/c1-2-4-10(5-3-1)8-14-13-12-11(6-7-17-12)15-9-16-13/h1-7,9H,8H2,(H,14,15,16) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| Purchase
CHEMBL
PC cid
PC sid
UniChem
Similars
| PubMed
| n/a | n/a | 1.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D
(Homo sapiens (Human)) | BDBM50223098
(CHEMBL30567)Show InChI InChI=1S/C19H22N4S/c1-3-7-15(8-4-1)13-20-19-18-16(9-12-24-18)21-17(22-19)14-23-10-5-2-6-11-23/h1,3-4,7-9,12H,2,5-6,10-11,13-14H2,(H,20,21,22) | PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
| PubMed
| n/a | n/a | 6.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Pharmaceutical Education and Research (NIPER)
Curated by ChEMBL
| Assay Description
Inhibitory activity against (PDE IV) phosphodiesterase IV in guinea pig articular tissue |
Bioorg Med Chem Lett 13: 1403-8 (2003)
BindingDB Entry DOI: 10.7270/Q29025ZS |
More data for this
Ligand-Target Pair | |
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