Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50035738 ((R)-3-(4-Chloro-phenyl)-8-methyl-8-aza-bicyclo[3.2...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50006239 (3-(4-Amino-3-iodo-phenyl)-8-methyl-8-aza-bicyclo[3...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50006234 (3-(4-Chloro-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]o...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50006230 (2-(4-aminophenyl)ethyl (2S,3S)-3-(4-chlorophenyl)-...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50006227 (3-(4-Chloro-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]o...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50006238 (3-(4-Chloro-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]o...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50006225 (3-(4-Azido-3-iodo-phenyl)-8-methyl-8-aza-bicyclo[3...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 4.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50006226 (2-(4-isothiocyanatophenyl)ethyl (2S,3S)-3-(4-chlor...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50006231 (3-(4-Chloro-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]o...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50005578 (4-azido-3-iodophenethyl 3-(4-chlorophenyl)-8-methy...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50005572 ((3S,8R)-3-(4-Amino-phenyl)-8-methyl-8-aza-bicyclo[...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 25 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50006236 (3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 61 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50005575 (3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 72 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM22418 (Cocaine | Cocaine (-) | methyl (1R,2R,3S,5S)-3-(be...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 102 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50006776 (3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 139 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50005574 (3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 196 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50005567 (3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 227 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50005546 (3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 248 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50005582 (3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 601 | n/a | n/a | n/a | n/a | n/a | n/a |
Research Triangle Institute Curated by ChEMBL | Assay Description Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes. | J Med Chem 35: 1813-7 (1992) BindingDB Entry DOI: 10.7270/Q29024D6 | |||||||||||
More data for this Ligand-Target Pair |