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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27642 (1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-3-y...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet  | KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 60 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27641 (1-(3-{[(2S)-2-aminopropanamido]methyl}phenyl)-N-[(...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 60 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27659 (1-(3-{[(2S)-2-aminopropanamido]methyl}phenyl)-N-be...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 80 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27650 (1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-3-y...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 220 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27655 (1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-2-y...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 230 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27651 (1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-3-y...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 260 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27643 (1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-2-y...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 300 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27652 (1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-3-y...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 370 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27653 (methyl 2-({[1-(5-{[(2S)-2-aminopropanamido]methyl}...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 770 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27649 (1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-3-y...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 790 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27644 (1-(4-{[(2S)-2-aminopropanamido]methyl}-1,3-thiazol...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 2.20E+3 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27654 (1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-2-y...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.31E+3 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27657 (1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-2-y...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.92E+3 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27646 (1-(6-{[(2S)-2-aminopropanamido]methyl}pyridin-2-yl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.05E+3 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27658 (1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-3-y...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.35E+3 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27645 (1-(4-{[(2S)-2-aminopropanamido]methyl}pyridin-2-yl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.20E+3 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27656 (1-(5-{[(2S)-2-aminopropanamido]methyl}thiophen-2-y...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.48E+3 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27647 (1-{2-[(2S)-2-aminopropanoyl]-2,3-dihydro-1H-isoind...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Histone-arginine methyltransferase CARM1 (Mus musculus (mouse)) | BDBM27648 (1-(2-{[(2S)-2-aminopropanamido]methyl}-1-benzofura...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | 9.0 | 22 |
MethylGene Inc. | Assay Description Histone H3 is used as the substrate for CARM-1 enzyme, and the methylation is monitored using tritiated S-Adenosyl-Methionine (SAM) as a methyl donor... | Bioorg Med Chem Lett 19: 1218-23 (2009) Article DOI: 10.1016/j.bmcl.2008.12.075 BindingDB Entry DOI: 10.7270/Q2K64GC6 | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
