Affinity Data by PubMed id=20384315

PubMed code 20384315

Found 16 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Nuclear factor NF-kappa-B p105 subunit (Homo sapiens (Human))	BDBM50196926 (CHEMBL438139 \| Rocaglamide \| US10085988, Compound ...) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars	Article PubMed	n/a	n/a	75	n/a	n/a	n/a	n/a	n/a	n/a
The Ohio State University Curated by ChEMBL					Assay Description Inhibition of NFkappa p50 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by chem...				J Nat Prod 73: 949-55 (2010) Article DOI: 10.1021/np1002065 BindingDB Entry DOI: 10.7270/Q28S4QWW
The Ohio State University Curated by ChEMBL					More data for this Ligand-Target Pair
Transcription factor p65 (Homo sapiens (Human))	BDBM50317857 (Artorigidin A \| CHEMBL1094756) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
The Ohio State University Curated by ChEMBL					Assay Description Inhibition of NFkappa p65 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by chem...				J Nat Prod 73: 949-55 (2010) Article DOI: 10.1021/np1002065 BindingDB Entry DOI: 10.7270/Q28S4QWW
The Ohio State University Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear factor NF-kappa-B p105 subunit (Homo sapiens (Human))	BDBM50317859 (CHEMBL1099162 \| artobiloxanthone) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
The Ohio State University Curated by ChEMBL					Assay Description Inhibition of NFkappa p50 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by chem...				J Nat Prod 73: 949-55 (2010) Article DOI: 10.1021/np1002065 BindingDB Entry DOI: 10.7270/Q28S4QWW
The Ohio State University Curated by ChEMBL					More data for this Ligand-Target Pair
Transcription factor p65 (Homo sapiens (Human))	BDBM50317859 (CHEMBL1099162 \| artobiloxanthone) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.70E+3	n/a	n/a	n/a	n/a	n/a	n/a
The Ohio State University Curated by ChEMBL					Assay Description Inhibition of NFkappa p65 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by chem...				J Nat Prod 73: 949-55 (2010) Article DOI: 10.1021/np1002065 BindingDB Entry DOI: 10.7270/Q28S4QWW
The Ohio State University Curated by ChEMBL					More data for this Ligand-Target Pair
Transcription factor p65 (Homo sapiens (Human))	BDBM50196926 (CHEMBL438139 \| Rocaglamide \| US10085988, Compound ...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars	Article PubMed	n/a	n/a	4.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
The Ohio State University Curated by ChEMBL					Assay Description Inhibition of NFkappa p65 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by chem...				J Nat Prod 73: 949-55 (2010) Article DOI: 10.1021/np1002065 BindingDB Entry DOI: 10.7270/Q28S4QWW
The Ohio State University Curated by ChEMBL					More data for this Ligand-Target Pair
Transcription factor p65 (Homo sapiens (Human))	BDBM50317858 (CHEMBL1095556 \| cycloartobiloxanthone) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
The Ohio State University Curated by ChEMBL					Assay Description Inhibition of NFkappa p65 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by chem...				J Nat Prod 73: 949-55 (2010) Article DOI: 10.1021/np1002065 BindingDB Entry DOI: 10.7270/Q28S4QWW
The Ohio State University Curated by ChEMBL					More data for this Ligand-Target Pair
Transcription factor p65 (Homo sapiens (Human))	BDBM50317860 (Artonin O \| CHEMBL1096733) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
The Ohio State University Curated by ChEMBL					Assay Description Inhibition of NFkappa p65 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by chem...				J Nat Prod 73: 949-55 (2010) Article DOI: 10.1021/np1002065 BindingDB Entry DOI: 10.7270/Q28S4QWW
The Ohio State University Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear factor NF-kappa-B p105 subunit (Homo sapiens (Human))	BDBM50317857 (Artorigidin A \| CHEMBL1094756) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
The Ohio State University Curated by ChEMBL					Assay Description Inhibition of NFkappa p50 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by chem...				J Nat Prod 73: 949-55 (2010) Article DOI: 10.1021/np1002065 BindingDB Entry DOI: 10.7270/Q28S4QWW
The Ohio State University Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear factor NF-kappa-B p105 subunit (Homo sapiens (Human))	BDBM50317861 (Artoristilbene \| CHEMBL1096732) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
The Ohio State University Curated by ChEMBL					Assay Description Inhibition of NFkappa p50 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by chem...				J Nat Prod 73: 949-55 (2010) Article DOI: 10.1021/np1002065 BindingDB Entry DOI: 10.7270/Q28S4QWW
The Ohio State University Curated by ChEMBL					More data for this Ligand-Target Pair
Transcription factor p65 (Homo sapiens (Human))	BDBM50317862 (CHEMBL1096731 \| Cyclorigidol) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
The Ohio State University Curated by ChEMBL					Assay Description Inhibition of NFkappa p65 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by chem...				J Nat Prod 73: 949-55 (2010) Article DOI: 10.1021/np1002065 BindingDB Entry DOI: 10.7270/Q28S4QWW
The Ohio State University Curated by ChEMBL					More data for this Ligand-Target Pair
Transcription factor p65 (Homo sapiens (Human))	BDBM50085545 (3-[(E)-2-(3,4-Dimethoxy-phenyl)-vinyl]-5-methoxy-p...) Show SMILES COc1cc(O)cc(\C=C\c2ccc(OC)c(OC)c2)c1 Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
The Ohio State University Curated by ChEMBL					Assay Description Inhibition of NFkappa p65 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by chem...				J Nat Prod 73: 949-55 (2010) Article DOI: 10.1021/np1002065 BindingDB Entry DOI: 10.7270/Q28S4QWW
The Ohio State University Curated by ChEMBL					More data for this Ligand-Target Pair
Transcription factor p65 (Homo sapiens (Human))	BDBM50317861 (Artoristilbene \| CHEMBL1096732) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
The Ohio State University Curated by ChEMBL					Assay Description Inhibition of NFkappa p65 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by chem...				J Nat Prod 73: 949-55 (2010) Article DOI: 10.1021/np1002065 BindingDB Entry DOI: 10.7270/Q28S4QWW
The Ohio State University Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear factor NF-kappa-B p105 subunit (Homo sapiens (Human))	BDBM50317858 (CHEMBL1095556 \| cycloartobiloxanthone) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
The Ohio State University Curated by ChEMBL					Assay Description Inhibition of NFkappa p50 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by chem...				J Nat Prod 73: 949-55 (2010) Article DOI: 10.1021/np1002065 BindingDB Entry DOI: 10.7270/Q28S4QWW
The Ohio State University Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear factor NF-kappa-B p105 subunit (Homo sapiens (Human))	BDBM50085545 (3-[(E)-2-(3,4-Dimethoxy-phenyl)-vinyl]-5-methoxy-p...) Show SMILES COc1cc(O)cc(\C=C\c2ccc(OC)c(OC)c2)c1 Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
The Ohio State University Curated by ChEMBL					Assay Description Inhibition of NFkappa p50 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by chem...				J Nat Prod 73: 949-55 (2010) Article DOI: 10.1021/np1002065 BindingDB Entry DOI: 10.7270/Q28S4QWW
The Ohio State University Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear factor NF-kappa-B p105 subunit (Homo sapiens (Human))	BDBM50317860 (Artonin O \| CHEMBL1096733) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
The Ohio State University Curated by ChEMBL					Assay Description Inhibition of NFkappa p50 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by chem...				J Nat Prod 73: 949-55 (2010) Article DOI: 10.1021/np1002065 BindingDB Entry DOI: 10.7270/Q28S4QWW
The Ohio State University Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear factor NF-kappa-B p105 subunit (Homo sapiens (Human))	BDBM50317862 (CHEMBL1096731 \| Cyclorigidol) Show SMILES Show InChI	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
The Ohio State University Curated by ChEMBL					Assay Description Inhibition of NFkappa p50 isolated from nuclear extract of human HeLa cells assessed as blockade of binding to biotinylated consesus sequence by chem...				J Nat Prod 73: 949-55 (2010) Article DOI: 10.1021/np1002065 BindingDB Entry DOI: 10.7270/Q28S4QWW
The Ohio State University Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%