Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Prolyl endopeptidase (Homo sapiens (Human)) | BDBM50038879 ((S)-2-(2-Formyl-pyrrolidine-1-carbonyl)-pyrrolidin...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE PC cid PC sid PDB UniChem Similars | PDB Article PubMed | 4.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Warwick Curated by ChEMBL | Assay Description Inhibition of prolyl oligopeptidase | Bioorg Med Chem 18: 4775-82 (2011) Article DOI: 10.1016/j.bmc.2010.05.012 BindingDB Entry DOI: 10.7270/Q2000319 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Prolyl endopeptidase (Homo sapiens (Human)) | BDBM50321860 ((S)-benzyl2-((S)-2-formylpiperidine-1-carbonyl)pyr...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 26 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Warwick Curated by ChEMBL | Assay Description Inhibition of prolyl oligopeptidase | Bioorg Med Chem 18: 4775-82 (2011) Article DOI: 10.1016/j.bmc.2010.05.012 BindingDB Entry DOI: 10.7270/Q2000319 | |||||||||||
More data for this Ligand-Target Pair |