Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Progesterone receptor (Homo sapiens (Human)) | BDBM50417609 (CHEMBL1645397) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 251 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50417615 (CHEMBL1645402) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50417606 (CHEMBL1645398) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 794 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50417610 (CHEMBL1645394) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 31.6 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50417615 (CHEMBL1645402) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 12.6 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50417607 (CHEMBL1645401) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.98 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50417605 (CHEMBL1645393) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50417607 (CHEMBL1645401) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 794 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50417606 (CHEMBL1645398) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50417616 (CHEMBL1645403) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 12.6 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mineralocorticoid receptor (Homo sapiens (Human)) | BDBM50417616 (CHEMBL1645403) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Antagonist activity at human MR ligand binding domain transfected in CHO cells co-transfected with MMTV-luciferase gene assessed as inhibition of cor... | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50417608 (CHEMBL1645399) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 631 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50417614 (CHEMBL1645396) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 50.1 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50417617 (CHEMBL1645392) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 7.94 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50417608 (CHEMBL1645399) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 10 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50417612 (CHEMBL1645395) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 12.6 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50417605 (CHEMBL1645393) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.00E+3 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50417612 (CHEMBL1645395) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 126 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50417609 (CHEMBL1645397) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 25.1 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50417611 (CHEMBL1641638) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5.01 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50417616 (CHEMBL1645403) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Antagonist activity at human GR DNA binding domain transfected in CHO cells co-transfected with MMTV-luciferase gene assessed as inhibition of cortis... | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50417610 (CHEMBL1645394) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 200 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50417611 (CHEMBL1641638) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 200 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50417613 (CHEMBL1645400) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 79.4 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50417613 (CHEMBL1645400) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.31 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50417617 (CHEMBL1645392) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.98 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid receptor (Homo sapiens (Human)) | BDBM50417614 (CHEMBL1645396) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant GR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Progesterone receptor (Homo sapiens (Human)) | BDBM50417616 (CHEMBL1645403) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a |
Merck Research Laboratories (MSD) Curated by ChEMBL | Assay Description Binding affinity to human recombinant PR by competition ligand binding fluorescence polarization assay | Bioorg Med Chem Lett 21: 137-40 (2010) Article DOI: 10.1016/j.bmcl.2010.11.054 BindingDB Entry DOI: 10.7270/Q2FN17F9 | |||||||||||
More data for this Ligand-Target Pair |