Found 31 hits of Enzyme Inhibition Constant Data Target/Host
(Institution) | Ligand | Target/Host
Links | Ligand
Links | Trg + Lig
Links | Ki
nM | ΔG°
kJ/mole | IC50
nM | Kd
nM | EC50/IC50
nM | koff
s-1 | kon
M-1s-1 | pH | Temp
°C |
|---|
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363514
(CHEMBL1946091)Show InChI InChI=1S/C20H27FN2O/c1-3-13-22(4-2)20(24)16-9-7-11-18-19(16)15-8-5-6-10-17(15)23(18)14-12-21/h5-6,8,10,16H,3-4,7,9,11-14H2,1-2H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet 
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 0.380 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363527
(CHEMBL1945412 | US9481685, [18F]FE-PBR)Show InChI InChI=1S/C22H23FN2OS/c1-3-24(4-2)22(26)21-19-15-9-5-7-11-17(15)25(14-13-23)20(19)16-10-6-8-12-18(16)27-21/h5-12,21H,3-4,13-14H2,1-2H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
| Article
PubMed
| 0.670 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363516
(CHEMBL1946093)Show InChI InChI=1S/C21H29FN2O/c1-3-13-23(14-4-2)21(25)17-9-7-11-19-20(17)16-8-5-6-10-18(16)24(19)15-12-22/h5-6,8,10,17H,3-4,7,9,11-15H2,1-2H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 0.700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363517
(CHEMBL1946094)Show InChI InChI=1S/C27H41FN2O/c1-3-5-7-11-19-29(20-12-8-6-4-2)27(31)23-15-13-17-25-26(23)22-14-9-10-16-24(22)30(25)21-18-28/h9-10,14,16,23H,3-8,11-13,15,17-21H2,1-2H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 0.700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363519
(CHEMBL1946096)Show InChI InChI=1S/C24H27FN2O/c1-2-26(17-18-9-4-3-5-10-18)24(28)20-12-8-14-22-23(20)19-11-6-7-13-21(19)27(22)16-15-25/h3-7,9-11,13,20H,2,8,12,14-17H2,1H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 0.730 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363523
(CHEMBL1944785)Show SMILES CCN(CC)C(=O)[C@H]1CCCc2c1c1c(OC)cccc1n2CCF |r| Show InChI InChI=1S/C20H27FN2O2/c1-4-22(5-2)20(24)14-8-6-9-15-18(14)19-16(23(15)13-12-21)10-7-11-17(19)25-3/h7,10-11,14H,4-6,8-9,12-13H2,1-3H3/t14-/m0/s1 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| Article
PubMed
| 0.870 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363504
(CHEMBL1945634)Show InChI InChI=1S/C19H24F2N2O/c1-3-22(4-2)19(24)15-6-5-7-16-18(15)14-9-8-13(21)12-17(14)23(16)11-10-20/h8-9,12,15H,3-7,10-11H2,1-2H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 1.05 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363515
(CHEMBL1946092)Show InChI InChI=1S/C23H25FN2O/c1-25(16-17-8-3-2-4-9-17)23(27)19-11-7-13-21-22(19)18-10-5-6-12-20(18)26(21)15-14-24/h2-6,8-10,12,19H,7,11,13-16H2,1H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 1.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363521
(CHEMBL1946098)Show SMILES CN(Cc1ccccc1)C(=O)C1CCCc2c1c1cc(F)ccc1n2CCF Show InChI InChI=1S/C23H24F2N2O/c1-26(15-16-6-3-2-4-7-16)23(28)18-8-5-9-21-22(18)19-14-17(25)10-11-20(19)27(21)13-12-24/h2-4,6-7,10-11,14,18H,5,8-9,12-13,15H2,1H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 1.45 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363505
(CHEMBL1945635)Show InChI InChI=1S/C20H26F2N2O2/c1-4-23(5-2)20(25)13-7-6-8-16-19(13)14-11-18(26-3)15(22)12-17(14)24(16)10-9-21/h11-13H,4-10H2,1-3H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 1.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363513
(CHEMBL1946090)Show InChI InChI=1S/C21H29FN2O/c1-14(2)24(15(3)4)21(25)17-9-7-11-19-20(17)16-8-5-6-10-18(16)23(19)13-12-22/h5-6,8,10,14-15,17H,7,9,11-13H2,1-4H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 1.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363528
(CHEMBL1945416)Show InChI InChI=1S/C20H27FN2O2/c1-4-22(5-2)20(24)15-7-6-8-18-19(15)16-13-14(25-3)9-10-17(16)23(18)12-11-21/h9-10,13,15H,4-8,11-12H2,1-3H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 1.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363511
(CHEMBL1945641)Show InChI InChI=1S/C19H25FN2O/c1-3-12-21(2)19(23)15-8-6-10-17-18(15)14-7-4-5-9-16(14)22(17)13-11-20/h4-5,7,9,15H,3,6,8,10-13H2,1-2H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 2.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363523
(CHEMBL1944785)Show SMILES CCN(CC)C(=O)[C@H]1CCCc2c1c1c(OC)cccc1n2CCF |r| Show InChI InChI=1S/C20H27FN2O2/c1-4-22(5-2)20(24)14-8-6-9-15-18(14)19-16(23(15)13-12-21)10-7-11-17(19)25-3/h7,10-11,14H,4-6,8-9,12-13H2,1-3H3/t14-/m0/s1 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| Article
PubMed
| 2.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363531
(CHEMBL1945631)Show InChI InChI=1S/C21H29FN2O2/c1-4-23(5-2)21(25)16-8-7-9-19-20(16)17-14-15(26-6-3)10-11-18(17)24(19)13-12-22/h10-11,14,16H,4-9,12-13H2,1-3H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 3.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363506
(CHEMBL1945636)Show InChI InChI=1S/C20H26F2N2O2/c1-4-23(5-2)20(25)13-7-6-8-16-19(13)14-11-15(22)18(26-3)12-17(14)24(16)10-9-21/h11-13H,4-10H2,1-3H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 3.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363503
(CHEMBL1945633)Show InChI InChI=1S/C19H24F2N2O/c1-3-22(4-2)19(24)14-6-5-7-17-18(14)15-12-13(21)8-9-16(15)23(17)11-10-20/h8-9,12,14H,3-7,10-11H2,1-2H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 3.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363524
(CHEMBL1944786)Show SMILES CCN(CC)C(=O)[C@@H]1CCCc2c1c1c(OC)cccc1n2CCF |r| Show InChI InChI=1S/C20H27FN2O2/c1-4-22(5-2)20(24)14-8-6-9-15-18(14)19-16(23(15)13-12-21)10-7-11-17(19)25-3/h7,10-11,14H,4-6,8-9,12-13H2,1-3H3/t14-/m1/s1 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Patents
Similars
| Article
PubMed
| 3.87 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363512
(CHEMBL1946089)Show InChI InChI=1S/C19H25FN2O/c1-13(2)21(3)19(23)15-8-6-10-17-18(15)14-7-4-5-9-16(14)22(17)12-11-20/h4-5,7,9,13,15H,6,8,10-12H2,1-3H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363530
(CHEMBL1945418)Show InChI InChI=1S/C21H29FN2O3/c1-5-23(6-2)21(25)15-8-7-9-16-19(15)20-17(24(16)11-10-22)12-14(26-3)13-18(20)27-4/h12-13,15H,5-11H2,1-4H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 4.34 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363510
(CHEMBL1945640)Show InChI InChI=1S/C21H27FN2O/c22-12-15-24-18-10-4-3-8-16(18)20-17(9-7-11-19(20)24)21(25)23-13-5-1-2-6-14-23/h3-4,8,10,17H,1-2,5-7,9,11-15H2 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 4.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363526
(CHEMBL1945413)Show InChI InChI=1S/C19H25FN2O/c1-3-21(4-2)19(23)15-9-7-11-17-18(15)14-8-5-6-10-16(14)22(17)13-12-20/h5-6,8,10,15H,3-4,7,9,11-13H2,1-2H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 5.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363529
(CHEMBL1945417)Show InChI InChI=1S/C20H27FN2O2/c1-4-22(5-2)20(24)16-7-6-8-17-19(16)15-10-9-14(25-3)13-18(15)23(17)12-11-21/h9-10,13,16H,4-8,11-12H2,1-3H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 5.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363532
(CHEMBL1945632)Show InChI InChI=1S/C19H24F2N2O/c1-3-22(4-2)19(24)13-7-5-9-15-17(13)18-14(21)8-6-10-16(18)23(15)12-11-20/h6,8,10,13H,3-5,7,9,11-12H2,1-2H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 7.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363522
(CHEMBL1946099)Show InChI InChI=1S/C19H24F2N2O/c1-12(2)22(3)19(24)14-5-4-6-17-18(14)15-11-13(21)7-8-16(15)23(17)10-9-20/h7-8,11-12,14H,4-6,9-10H2,1-3H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 8.23 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363509
(CHEMBL1945639)Show InChI InChI=1S/C20H25FN2O/c21-11-14-23-17-9-3-2-7-15(17)19-16(8-6-10-18(19)23)20(24)22-12-4-1-5-13-22/h2-3,7,9,16H,1,4-6,8,10-14H2 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 18.3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363520
(CHEMBL1946097)Show InChI InChI=1S/C22H23FN2O/c23-13-14-25-19-11-5-4-9-17(19)21-18(10-6-12-20(21)25)22(26)24-15-16-7-2-1-3-8-16/h1-5,7-9,11,18H,6,10,12-15H2,(H,24,26) | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 28.6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363525
(CHEMBL1945414)Show InChI InChI=1S/C19H25FN2O2/c1-3-21(4-2)19(24)14-6-5-7-17-18(14)15-12-13(23)8-9-16(15)22(17)11-10-20/h8-9,12,14,23H,3-7,10-11H2,1-2H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 135 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363518
(CHEMBL1946095)Show InChI InChI=1S/C17H21FN2O/c1-19(2)17(21)13-7-5-9-15-16(13)12-6-3-4-8-14(12)20(15)11-10-18/h3-4,6,8,13H,5,7,9-11H2,1-2H3 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 502 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363508
(CHEMBL1945638)Show InChI InChI=1S/C19H23FN2O/c20-10-13-22-16-8-2-1-6-14(16)18-15(7-5-9-17(18)22)19(23)21-11-3-4-12-21/h1-2,6,8,15H,3-5,7,9-13H2 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 503 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
Translocator protein
(Rattus norvegicus (rat)) | BDBM50363507
(CHEMBL1945637)Show InChI InChI=1S/C19H23FN2O2/c20-8-9-22-16-6-2-1-4-14(16)18-15(5-3-7-17(18)22)19(23)21-10-12-24-13-11-21/h1-2,4,6,15H,3,5,7-13H2 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
AffyNet
| CHEMBL
PC cid
PC sid
UniChem
Similars
| Article
PubMed
| 607 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GE Healthcare
Curated by ChEMBL
| Assay Description
Displacement of [3H]PK11195 from TSPO receptor in Wistar rat heart homogenate after 15 mins |
Bioorg Med Chem Lett 22: 1308-13 (2012)
Article DOI: 10.1016/j.bmcl.2011.12.084
BindingDB Entry DOI: 10.7270/Q2RR1ZPZ |
More data for this
Ligand-Target Pair | |
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