Affinity Data by PubMed id=22560469

PubMed code 22560469

Found 25 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383678 (CHEMBL2030077) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	120	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383684 (CHEMBL1961795) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	400	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as NCoR recruitment by FRET assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383670 (CHEMBL2030069) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	>3.00E+3	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383674 (CHEMBL2030073) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	97	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383681 (CHEMBL2030080) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	780	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383668 (CHEMBL2029898) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	840	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383677 (CHEMBL2030076) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	600	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383669 (CHEMBL2030065) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.20E+3	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383684 (CHEMBL1961795) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	2.30E+3	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383675 (CHEMBL2030074) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	77	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383683 (CHEMBL2030082) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	710	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383661 (CHEMBL2030064) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	650	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383662 (CHEMBL2029876) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	>3.00E+3	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383663 (CHEMBL2029882) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	2.50E+3	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383666 (CHEMBL2029886) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.10E+3	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383667 (CHEMBL2029895) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	>3.00E+3	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383672 (CHEMBL2030071) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	650	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383673 (CHEMBL2030072) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	120	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383680 (CHEMBL2030079) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	620	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383682 (CHEMBL2030081) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	330	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383665 (CHEMBL2029885) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	1.70E+3	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383671 (CHEMBL2030070) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	800	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383676 (CHEMBL2030075) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	140	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383679 (CHEMBL2030078) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	2.00E+3	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair
Nuclear receptor subfamily 1 group D member 1 (Homo sapiens (Human))	BDBM50383664 (CHEMBL2029883) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	n/a	n/a	2.10E+3	n/a	n/a	n/a	n/a
The Scripps Research Institute Curated by ChEMBL					Assay Description Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assay				Bioorg Med Chem Lett 22: 3739-42 (2012) Article DOI: 10.1016/j.bmcl.2012.04.023 BindingDB Entry DOI: 10.7270/Q2CN74ZF
The Scripps Research Institute Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%