Affinity Data by PubMed id=23395110

PubMed code 23395110

Found 4 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Protein arginine N-methyltransferase 1 [11-371] (Homo sapiens (Human))	BDBM50446399 (CHEMBL3109664) Show SMILES OC(=O)CCCCCNC(=O)NCCCCCC(O)=O Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	6.10E+3	n/a	n/a	n/a	n/a	n/a	n/a
Universidade de Vigo Curated by ChEMBL					Assay Description Inhibition of recombinant human PRMT1 expressed in Escherichia coli using histone H4 peptide as substrate by chemiluminescence assay				Bioorg Med Chem 21: 2056-67 (2013) Article DOI: 10.1016/j.bmc.2013.01.017 BindingDB Entry DOI: 10.7270/Q22N53S7
Universidade de Vigo Curated by ChEMBL					More data for this Ligand-Target Pair
Protein arginine N-methyltransferase 1 [11-371] (Homo sapiens (Human))	BDBM50446401 (CHEMBL3109656) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	8.80E+3	n/a	n/a	n/a	n/a	n/a	n/a
Universidade de Vigo Curated by ChEMBL					Assay Description Inhibition of recombinant human PRMT1 expressed in Escherichia coli using histone H4 peptide as substrate by chemiluminescence assay				Bioorg Med Chem 21: 2056-67 (2013) Article DOI: 10.1016/j.bmc.2013.01.017 BindingDB Entry DOI: 10.7270/Q22N53S7
Universidade de Vigo Curated by ChEMBL					More data for this Ligand-Target Pair
Protein arginine N-methyltransferase 1 [11-371] (Homo sapiens (Human))	BDBM50446400 (CHEMBL3109657) Show SMILES COc1ccc2C(=O)N(C)C(=O)c3cccc1c23 Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	Purchase CHEMBL MCE PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.63E+4	n/a	n/a	n/a	n/a	n/a	n/a
Universidade de Vigo Curated by ChEMBL					Assay Description Inhibition of recombinant human PRMT1 expressed in Escherichia coli using histone H4 peptide as substrate by chemiluminescence assay				Bioorg Med Chem 21: 2056-67 (2013) Article DOI: 10.1016/j.bmc.2013.01.017 BindingDB Entry DOI: 10.7270/Q22N53S7
Universidade de Vigo Curated by ChEMBL					More data for this Ligand-Target Pair
Protein arginine N-methyltransferase 1 [11-371] (Homo sapiens (Human))	BDBM50446398 (CHEMBL3109661) Show SMILES Show InChI	PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	2.52E+4	n/a	n/a	n/a	n/a	n/a	n/a
Universidade de Vigo Curated by ChEMBL					Assay Description Inhibition of recombinant human PRMT1 expressed in Escherichia coli using histone H4 peptide as substrate by chemiluminescence assay				Bioorg Med Chem 21: 2056-67 (2013) Article DOI: 10.1016/j.bmc.2013.01.017 BindingDB Entry DOI: 10.7270/Q22N53S7
Universidade de Vigo Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%