Affinity Data by PubMed id=2362282

PubMed code 2362282

Found 7 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Sodium-dependent dopamine transporter (BOVINE)	BDBM50366564 (CHEMBL1790051 \| CHEMBL83729 \| WIN-35065-2) Show SMILES Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	22	n/a	n/a	n/a	n/a	n/a	n/a
University of Maryland Curated by ChEMBL					Assay Description Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissue				J Med Chem 33: 2024-7 (1990) BindingDB Entry DOI: 10.7270/Q2BG2PMN
University of Maryland Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium-dependent dopamine transporter (BOVINE)	BDBM50366564 (CHEMBL1790051 \| CHEMBL83729 \| WIN-35065-2) Show SMILES Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	22	n/a	n/a	n/a	n/a	n/a	n/a
University of Maryland Curated by ChEMBL					Assay Description Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissue				J Med Chem 33: 2024-7 (1990) BindingDB Entry DOI: 10.7270/Q2BG2PMN
University of Maryland Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium-dependent dopamine transporter (BOVINE)	BDBM50015692 (8-Methyl-3-(4-nitro-phenyl)-8-aza-bicyclo[3.2.1]oc...) Show SMILES Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	137	n/a	n/a	n/a	n/a	n/a	n/a
University of Maryland Curated by ChEMBL					Assay Description Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissue				J Med Chem 33: 2024-7 (1990) BindingDB Entry DOI: 10.7270/Q2BG2PMN
University of Maryland Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium-dependent dopamine transporter (BOVINE)	BDBM50015692 (8-Methyl-3-(4-nitro-phenyl)-8-aza-bicyclo[3.2.1]oc...) Show SMILES Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	137	n/a	n/a	n/a	n/a	n/a	n/a
University of Maryland Curated by ChEMBL					Assay Description Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissue				J Med Chem 33: 2024-7 (1990) BindingDB Entry DOI: 10.7270/Q2BG2PMN
University of Maryland Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium-dependent dopamine transporter (BOVINE)	BDBM22418 (Cocaine \| Cocaine (-) \| methyl (1R,2R,3S,5S)-3-(be...) Show SMILES Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	Purchase DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	PubMed	n/a	n/a	139	n/a	n/a	n/a	n/a	n/a	n/a
University of Maryland Curated by ChEMBL					Assay Description Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissue				J Med Chem 33: 2024-7 (1990) BindingDB Entry DOI: 10.7270/Q2BG2PMN
University of Maryland Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium-dependent dopamine transporter (BOVINE)	BDBM50015695 (3-(4-Amino-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...) Show SMILES Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	192	n/a	n/a	n/a	n/a	n/a	n/a
University of Maryland Curated by ChEMBL					Assay Description Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissue				J Med Chem 33: 2024-7 (1990) BindingDB Entry DOI: 10.7270/Q2BG2PMN
University of Maryland Curated by ChEMBL					More data for this Ligand-Target Pair
Sodium-dependent dopamine transporter (BOVINE)	BDBM50015694 (3-(2,4-Dinitro-phenyl)-8-methyl-8-aza-bicyclo[3.2....) Show SMILES Show InChI	UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	1.10E+4	n/a	n/a	n/a	n/a	n/a	n/a
University of Maryland Curated by ChEMBL					Assay Description Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissue				J Med Chem 33: 2024-7 (1990) BindingDB Entry DOI: 10.7270/Q2BG2PMN
University of Maryland Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%