Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443088 (CHEMBL3087216) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443089 (CHEMBL3086715) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443089 (CHEMBL3086715) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 28.4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443090 (CHEMBL3086712) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 37 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443091 (CHEMBL3087511) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 47 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443092 (CHEMBL3085792) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 48 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443093 (CHEMBL3087217) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 51 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443087 (CHEMBL3087214) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 61 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443086 (CHEMBL3087508) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 65 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443085 (AFQ056 | Mavoglurant) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 72 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443084 (CHEMBL3087220) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 72 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443083 (CHEMBL3087219) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 76 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443082 (CHEMBL3087513) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 85 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443081 (CHEMBL3087212) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 86 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443080 (CHEMBL3087514) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 103 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443080 (CHEMBL3087514) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 103 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443079 (CHEMBL3087225) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 132 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443078 (CHEMBL3087509) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 137 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443077 (CHEMBL3087505) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 168 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443076 (CHEMBL3087507) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443075 (CHEMBL3086717) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 180 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443074 (CHEMBL3087218) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 187 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443073 (CHEMBL3086716) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 189 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443072 (CHEMBL3087226) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 210 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443071 (CHEMBL3086718) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 227 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443070 (CHEMBL3087213) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 298 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443069 (CHEMBL3086719) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 306 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443068 (CHEMBL3087224) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 308 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443067 (CHEMBL3087211) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 340 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443066 (CHEMBL3087223) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 543 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443065 (CHEMBL3087506) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 575 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443064 (CHEMBL3086720) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 813 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443063 (CHEMBL3087221) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 818 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443062 (CHEMBL3086713) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 930 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443057 (CHEMBL3086714) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.01E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443061 (CHEMBL3087510) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.02E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443060 (CHEMBL3087215) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.19E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443059 (CHEMBL3087512) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.35E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443058 (CHEMBL3086711) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 5 (Homo sapiens (Human)) | BDBM50443056 (CHEMBL3087222) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Merz Pharmaceuticals GmbH Curated by ChEMBL | Assay Description Negative allosteric modulation of human mGlu5 receptor expressed in CHO cells assessed as inhibition of L-quisqualate-induced intracellular calcium m... | Bioorg Med Chem Lett 23: 6370-6 (2013) Article DOI: 10.1016/j.bmcl.2013.09.059 BindingDB Entry DOI: 10.7270/Q2W37XRD | |||||||||||
More data for this Ligand-Target Pair |