Affinity Data by PubMed id=24456902

PubMed code 24456902

Found 14 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Platelet-derived growth factor receptor alpha (Homo sapiens (Human))	BDBM50447827 (CHEMBL3114023) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	52	n/a	n/a	n/a	n/a	n/a	n/a
Tianjin University Curated by ChEMBL					Assay Description Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF method				Bioorg Med Chem Lett 24: 1108-10 (2014) Article DOI: 10.1016/j.bmcl.2014.01.003 BindingDB Entry DOI: 10.7270/Q2GF0W1N
Tianjin University Curated by ChEMBL					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor alpha (Homo sapiens (Human))	BDBM26474 (5-({4-[(2,3-dimethyl-2H-indazol-6-yl)(methyl)amino...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	Purchase DrugBank MCE PC cid PC sid UniChem Patents Similars	DrugBank Article PubMed	n/a	n/a	71	n/a	n/a	n/a	n/a	n/a	n/a
Tianjin University Curated by ChEMBL					Assay Description Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF method				Bioorg Med Chem Lett 24: 1108-10 (2014) Article DOI: 10.1016/j.bmcl.2014.01.003 BindingDB Entry DOI: 10.7270/Q2GF0W1N
Tianjin University Curated by ChEMBL					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor alpha (Homo sapiens (Human))	BDBM50447821 (CHEMBL3114029) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	72	n/a	n/a	n/a	n/a	n/a	n/a
Tianjin University Curated by ChEMBL					Assay Description Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF method				Bioorg Med Chem Lett 24: 1108-10 (2014) Article DOI: 10.1016/j.bmcl.2014.01.003 BindingDB Entry DOI: 10.7270/Q2GF0W1N
Tianjin University Curated by ChEMBL					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor alpha (Homo sapiens (Human))	BDBM50447820 (CHEMBL3114030) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	75	n/a	n/a	n/a	n/a	n/a	n/a
Tianjin University Curated by ChEMBL					Assay Description Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF method				Bioorg Med Chem Lett 24: 1108-10 (2014) Article DOI: 10.1016/j.bmcl.2014.01.003 BindingDB Entry DOI: 10.7270/Q2GF0W1N
Tianjin University Curated by ChEMBL					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor alpha (Homo sapiens (Human))	BDBM50447828 (CHEMBL3114022) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	80	n/a	n/a	n/a	n/a	n/a	n/a
Tianjin University Curated by ChEMBL					Assay Description Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF method				Bioorg Med Chem Lett 24: 1108-10 (2014) Article DOI: 10.1016/j.bmcl.2014.01.003 BindingDB Entry DOI: 10.7270/Q2GF0W1N
Tianjin University Curated by ChEMBL					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor alpha (Homo sapiens (Human))	BDBM50447830 (CHEMBL3114020) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	85	n/a	n/a	n/a	n/a	n/a	n/a
Tianjin University Curated by ChEMBL					Assay Description Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF method				Bioorg Med Chem Lett 24: 1108-10 (2014) Article DOI: 10.1016/j.bmcl.2014.01.003 BindingDB Entry DOI: 10.7270/Q2GF0W1N
Tianjin University Curated by ChEMBL					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor alpha (Homo sapiens (Human))	BDBM50447822 (CHEMBL3114028) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	86	n/a	n/a	n/a	n/a	n/a	n/a
Tianjin University Curated by ChEMBL					Assay Description Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF method				Bioorg Med Chem Lett 24: 1108-10 (2014) Article DOI: 10.1016/j.bmcl.2014.01.003 BindingDB Entry DOI: 10.7270/Q2GF0W1N
Tianjin University Curated by ChEMBL					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor alpha (Homo sapiens (Human))	BDBM50447826 (CHEMBL3114024) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	94	n/a	n/a	n/a	n/a	n/a	n/a
Tianjin University Curated by ChEMBL					Assay Description Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF method				Bioorg Med Chem Lett 24: 1108-10 (2014) Article DOI: 10.1016/j.bmcl.2014.01.003 BindingDB Entry DOI: 10.7270/Q2GF0W1N
Tianjin University Curated by ChEMBL					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor alpha (Homo sapiens (Human))	BDBM50447823 (CHEMBL3114027) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	95	n/a	n/a	n/a	n/a	n/a	n/a
Tianjin University Curated by ChEMBL					Assay Description Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF method				Bioorg Med Chem Lett 24: 1108-10 (2014) Article DOI: 10.1016/j.bmcl.2014.01.003 BindingDB Entry DOI: 10.7270/Q2GF0W1N
Tianjin University Curated by ChEMBL					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor alpha (Homo sapiens (Human))	BDBM50447829 (CHEMBL3114021) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	96	n/a	n/a	n/a	n/a	n/a	n/a
Tianjin University Curated by ChEMBL					Assay Description Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF method				Bioorg Med Chem Lett 24: 1108-10 (2014) Article DOI: 10.1016/j.bmcl.2014.01.003 BindingDB Entry DOI: 10.7270/Q2GF0W1N
Tianjin University Curated by ChEMBL					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor alpha (Homo sapiens (Human))	BDBM50447831 (CHEMBL3114019) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	97	n/a	n/a	n/a	n/a	n/a	n/a
Tianjin University Curated by ChEMBL					Assay Description Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF method				Bioorg Med Chem Lett 24: 1108-10 (2014) Article DOI: 10.1016/j.bmcl.2014.01.003 BindingDB Entry DOI: 10.7270/Q2GF0W1N
Tianjin University Curated by ChEMBL					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor alpha (Homo sapiens (Human))	BDBM50447825 (CHEMBL3114025) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	104	n/a	n/a	n/a	n/a	n/a	n/a
Tianjin University Curated by ChEMBL					Assay Description Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF method				Bioorg Med Chem Lett 24: 1108-10 (2014) Article DOI: 10.1016/j.bmcl.2014.01.003 BindingDB Entry DOI: 10.7270/Q2GF0W1N
Tianjin University Curated by ChEMBL					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor alpha (Homo sapiens (Human))	BDBM50447832 (CHEMBL3114018) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	130	n/a	n/a	n/a	n/a	n/a	n/a
Tianjin University Curated by ChEMBL					Assay Description Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF method				Bioorg Med Chem Lett 24: 1108-10 (2014) Article DOI: 10.1016/j.bmcl.2014.01.003 BindingDB Entry DOI: 10.7270/Q2GF0W1N
Tianjin University Curated by ChEMBL					More data for this Ligand-Target Pair
Platelet-derived growth factor receptor alpha (Homo sapiens (Human))	BDBM50447824 (CHEMBL3114026) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	140	n/a	n/a	n/a	n/a	n/a	n/a
Tianjin University Curated by ChEMBL					Assay Description Inhibition of PDGFR-alpha tyrosine kinase (unknown origin) after 30 mins by HTRF method				Bioorg Med Chem Lett 24: 1108-10 (2014) Article DOI: 10.1016/j.bmcl.2014.01.003 BindingDB Entry DOI: 10.7270/Q2GF0W1N
Tianjin University Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%