Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Reverse transcriptase (Human immunodeficiency virus 1) | BDBM50046719 (CHEMBL3310874) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 490 | n/a | n/a | n/a | n/a | n/a | n/a |
Hebei University Curated by ChEMBL | Assay Description Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISA plate reader analysis | Bioorg Med Chem Lett 24: 3426-9 (2014) Article DOI: 10.1016/j.bmcl.2014.05.079 BindingDB Entry DOI: 10.7270/Q25H7HWV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase (Human immunodeficiency virus 1) | BDBM50046726 (CHEMBL3310879) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.32E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hebei University Curated by ChEMBL | Assay Description Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISA plate reader analysis | Bioorg Med Chem Lett 24: 3426-9 (2014) Article DOI: 10.1016/j.bmcl.2014.05.079 BindingDB Entry DOI: 10.7270/Q25H7HWV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase (Human immunodeficiency virus 1) | BDBM50046721 (CHEMBL3310876) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.41E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hebei University Curated by ChEMBL | Assay Description Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISA plate reader analysis | Bioorg Med Chem Lett 24: 3426-9 (2014) Article DOI: 10.1016/j.bmcl.2014.05.079 BindingDB Entry DOI: 10.7270/Q25H7HWV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase (Human immunodeficiency virus 1) | BDBM50046717 (CHEMBL2018791) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.58E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hebei University Curated by ChEMBL | Assay Description Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISA plate reader analysis | Bioorg Med Chem Lett 24: 3426-9 (2014) Article DOI: 10.1016/j.bmcl.2014.05.079 BindingDB Entry DOI: 10.7270/Q25H7HWV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase (Human immunodeficiency virus 1) | BDBM50046724 (CHEMBL2018793) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.83E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hebei University Curated by ChEMBL | Assay Description Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISA plate reader analysis | Bioorg Med Chem Lett 24: 3426-9 (2014) Article DOI: 10.1016/j.bmcl.2014.05.079 BindingDB Entry DOI: 10.7270/Q25H7HWV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase (Human immunodeficiency virus 1) | BDBM50046725 (CHEMBL3310878) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.02E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Hebei University Curated by ChEMBL | Assay Description Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISA plate reader analysis | Bioorg Med Chem Lett 24: 3426-9 (2014) Article DOI: 10.1016/j.bmcl.2014.05.079 BindingDB Entry DOI: 10.7270/Q25H7HWV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase (Human immunodeficiency virus 1) | BDBM50046718 (CHEMBL3310873) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.29E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Hebei University Curated by ChEMBL | Assay Description Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISA plate reader analysis | Bioorg Med Chem Lett 24: 3426-9 (2014) Article DOI: 10.1016/j.bmcl.2014.05.079 BindingDB Entry DOI: 10.7270/Q25H7HWV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase (Human immunodeficiency virus 1) | BDBM50002692 ((AZT) 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.82E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Hebei University Curated by ChEMBL | Assay Description Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISA plate reader analysis | Bioorg Med Chem Lett 24: 3426-9 (2014) Article DOI: 10.1016/j.bmcl.2014.05.079 BindingDB Entry DOI: 10.7270/Q25H7HWV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase (Human immunodeficiency virus 1) | BDBM50046729 (CHEMBL3310881) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.97E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Hebei University Curated by ChEMBL | Assay Description Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISA plate reader analysis | Bioorg Med Chem Lett 24: 3426-9 (2014) Article DOI: 10.1016/j.bmcl.2014.05.079 BindingDB Entry DOI: 10.7270/Q25H7HWV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase (Human immunodeficiency virus 1) | BDBM50046727 (CHEMBL3310880) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.68E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Hebei University Curated by ChEMBL | Assay Description Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISA plate reader analysis | Bioorg Med Chem Lett 24: 3426-9 (2014) Article DOI: 10.1016/j.bmcl.2014.05.079 BindingDB Entry DOI: 10.7270/Q25H7HWV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase (Human immunodeficiency virus 1) | BDBM50046720 (CHEMBL3310875) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.14E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Hebei University Curated by ChEMBL | Assay Description Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISA plate reader analysis | Bioorg Med Chem Lett 24: 3426-9 (2014) Article DOI: 10.1016/j.bmcl.2014.05.079 BindingDB Entry DOI: 10.7270/Q25H7HWV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Reverse transcriptase (Human immunodeficiency virus 1) | BDBM50046722 (CHEMBL3310877) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.38E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Hebei University Curated by ChEMBL | Assay Description Inhibition of HIV-1 reverse transcriptase after 1 hr by ELISA plate reader analysis | Bioorg Med Chem Lett 24: 3426-9 (2014) Article DOI: 10.1016/j.bmcl.2014.05.079 BindingDB Entry DOI: 10.7270/Q25H7HWV | |||||||||||
More data for this Ligand-Target Pair |