Affinity Data by PubMed id=26004580

PubMed code 26004580

Found 5 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Protein-glutamine gamma-glutamyltransferase 2 (Homo sapiens (Human))	BDBM50342583 ((E)-4-chloro-3-(2-(2-methoxyphenyl)-2-oxoethyliden...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	3.30E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Stanford University Curated by ChEMBL					Assay Description Non-competitive inhibition of recombinant human TG2 V224 mutant deamidation activity using Cbz-Gln-Gly as substrate preincubated for 30 mins followed...				Bioorg Med Chem Lett 25: 4922-6 (2015) Article DOI: 10.1016/j.bmcl.2015.05.006 BindingDB Entry DOI: 10.7270/Q2W95C07
Stanford University Curated by ChEMBL					More data for this Ligand-Target Pair
Protein-glutamine gamma-glutamyltransferase 2 (Homo sapiens (Human))	BDBM50342590 ((E)-4-chloro-3-(2-oxo-2-(pyridin-3-yl)ethylidene)-...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	9.10E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Stanford University Curated by ChEMBL					Assay Description Non-competitive inhibition of recombinant human TG2 V224 mutant deamidation activity using Cbz-Gln-Gly as substrate preincubated for 30 mins followed...				Bioorg Med Chem Lett 25: 4922-6 (2015) Article DOI: 10.1016/j.bmcl.2015.05.006 BindingDB Entry DOI: 10.7270/Q2W95C07
Stanford University Curated by ChEMBL					More data for this Ligand-Target Pair
Protein-glutamine gamma-glutamyltransferase 2 (Homo sapiens (Human))	BDBM81791 (Dopamine + GPP(NH)p \| GPP(NH)P(+) \| GPP(NH)p(-) \| ...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	KEGG PC cid PC sid UniChem Similars	Article PubMed	2.70E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Stanford University Curated by ChEMBL					Assay Description Competitive inhibition of recombinant human TG2 V224 mutant deamidation activity using Cbz-Gln-Gly as substrate preincubated for 30 mins followed by ...				Bioorg Med Chem Lett 25: 4922-6 (2015) Article DOI: 10.1016/j.bmcl.2015.05.006 BindingDB Entry DOI: 10.7270/Q2W95C07
Stanford University Curated by ChEMBL					More data for this Ligand-Target Pair
Protein-glutamine gamma-glutamyltransferase 2 (Homo sapiens (Human))	BDBM50342582 ((E)-4-chloro-3-(2-(4-chlorophenyl)-2-oxoethylidene...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	4.70E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Stanford University Curated by ChEMBL					Assay Description Non-competitive inhibition of recombinant human TG2 V224 mutant deamidation activity using Cbz-Gln-Gly as substrate preincubated for 30 mins followed...				Bioorg Med Chem Lett 25: 4922-6 (2015) Article DOI: 10.1016/j.bmcl.2015.05.006 BindingDB Entry DOI: 10.7270/Q2W95C07
Stanford University Curated by ChEMBL					More data for this Ligand-Target Pair
Protein-glutamine gamma-glutamyltransferase 2 (Homo sapiens (Human))	BDBM50342569 ((E)-3-(2-oxo-2-(pyridin-3-yl)ethylidene)indolin-2-...) Show SMILES O=C(\C=C1\C(=O)Nc2ccccc12)c1cccnc1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	8.60E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Stanford University Curated by ChEMBL					Assay Description Non-competitive inhibition of recombinant human TG2 V224 mutant deamidation activity using Cbz-Gln-Gly as substrate preincubated for 30 mins followed...				Bioorg Med Chem Lett 25: 4922-6 (2015) Article DOI: 10.1016/j.bmcl.2015.05.006 BindingDB Entry DOI: 10.7270/Q2W95C07
Stanford University Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%