Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Type-2 angiotensin II receptor (RAT) | BDBM50117831 (CHEMBL3613974) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 34 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Economics Curated by ChEMBL | Assay Description Inhibition of rat AT2 receptor | Bioorg Med Chem 23: 6087-99 (2015) Article DOI: 10.1016/j.bmc.2015.07.045 BindingDB Entry DOI: 10.7270/Q2S75J31 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Macrophage metalloelastase (Homo sapiens (Human)) | BDBM50215926 (4-(4,5-dibromo-1H-pyrrol-2-yl)-1H-imidazo[4,5-c]py...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.66E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroclaw University of Economics Curated by ChEMBL | Assay Description Inhibition of MMP12 (unknown origin) | Bioorg Med Chem 23: 6087-99 (2015) Article DOI: 10.1016/j.bmc.2015.07.045 BindingDB Entry DOI: 10.7270/Q2S75J31 | |||||||||||
More data for this Ligand-Target Pair |