Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125819 (CHEMBL3623895) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.110 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125820 (CHEMBL3623894) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.190 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125941 (CHEMBL3623875) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.230 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125818 (CHEMBL3623896) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.380 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125824 (CHEMBL3623893) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.530 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125818 (CHEMBL3623896) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.570 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125825 (CHEMBL3623892) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.670 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125826 (CHEMBL3623891) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.960 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125942 (CHEMBL3623874) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125831 (CHEMBL3623887) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125943 (CHEMBL3623873) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125829 (CHEMBL3623889) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 24 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125899 (CHEMBL3623879) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 30 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125904 (CHEMBL3623878) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125938 (CHEMBL3623877) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 164 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125940 (CHEMBL3623876) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 188 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125827 (CHEMBL3623890) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 483 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125830 (CHEMBL3623888) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 485 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125839 (CHEMBL3623886) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125898 (CHEMBL3623880) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125858 (CHEMBL3623885) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125896 (CHEMBL3623882) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125895 (CHEMBL3623883) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125876 (CHEMBL3623884) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein-serine O-palmitoleoyltransferase porcupine (Homo sapiens (Human)) | BDBM50125897 (CHEMBL3623881) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Soochow University Curated by ChEMBL | Assay Description Inhibition of porcupine (unknown origin) expressed in mouse L Wnt3A cells co-cultured with TM3 cells harboring luciferase reporter gene assessed as r... | Bioorg Med Chem 23: 6855-68 (2015) Article DOI: 10.1016/j.bmc.2015.09.048 BindingDB Entry DOI: 10.7270/Q2J10500 | |||||||||||
More data for this Ligand-Target Pair |