Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Serine/threonine-protein kinase pim-1 (Homo sapiens (Human)) | BDBM50154291 (CHEMBL3775181) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | <5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Russia; Mendeleyev University of Chemical Technology Curated by ChEMBL | Assay Description Inhibition of full length human N-terminal GST-HIS6-tagged PIM1 expressed in sf9 cells by flashplate based radiometric 33pan-quinase assay | Eur J Med Chem 112: 114-29 (2016) Article DOI: 10.1016/j.ejmech.2016.01.050 BindingDB Entry DOI: 10.7270/Q2VQ34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual serine/threonine and tyrosine protein kinase (Homo sapiens (Human)) | BDBM50154291 (CHEMBL3775181) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | <5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Russia; Mendeleyev University of Chemical Technology Curated by ChEMBL | Assay Description Inhibition of human RIPK5 by flashplate based radiometric 33pan-quinase assay | Eur J Med Chem 112: 114-29 (2016) Article DOI: 10.1016/j.ejmech.2016.01.050 BindingDB Entry DOI: 10.7270/Q2VQ34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase tousled-like 1 (Homo sapiens (Human)) | BDBM50154291 (CHEMBL3775181) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | <5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Russia; Mendeleyev University of Chemical Technology Curated by ChEMBL | Assay Description Inhibition of human N-terminal FLAG, C-terminal HIS8-tagged TLK1 expressed in sf9 cells by flashplate based radiometric 33pan-quinase assay | Eur J Med Chem 112: 114-29 (2016) Article DOI: 10.1016/j.ejmech.2016.01.050 BindingDB Entry DOI: 10.7270/Q2VQ34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Serine/threonine-protein kinase pim-3 (Homo sapiens (Human)) | BDBM50154291 (CHEMBL3775181) | KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | <5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Russia; Mendeleyev University of Chemical Technology Curated by ChEMBL | Assay Description Inhibition of full length human N-terminal GST-HIS6-tagged PIM3 expressed in sf9 cells by flashplate based radiometric 33pan-quinase assay | Eur J Med Chem 112: 114-29 (2016) Article DOI: 10.1016/j.ejmech.2016.01.050 BindingDB Entry DOI: 10.7270/Q2VQ34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aurora kinase B (Homo sapiens (Human)) | BDBM50154291 (CHEMBL3775181) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | <5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Russia; Mendeleyev University of Chemical Technology Curated by ChEMBL | Assay Description Inhibition of full length human N-terminal GST-HIS6-tagged Aurora B expressed in sf9 cells by flashplate based radiometric 33pan-quinase assay | Eur J Med Chem 112: 114-29 (2016) Article DOI: 10.1016/j.ejmech.2016.01.050 BindingDB Entry DOI: 10.7270/Q2VQ34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Mitogen-activated protein kinase kinase kinase 7 (Homo sapiens (Human)) | BDBM50154291 (CHEMBL3775181) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | <5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Russia; Mendeleyev University of Chemical Technology Curated by ChEMBL | Assay Description Inhibition of human MAP3K7 by flashplate based radiometric 33pan-quinase assay | Eur J Med Chem 112: 114-29 (2016) Article DOI: 10.1016/j.ejmech.2016.01.050 BindingDB Entry DOI: 10.7270/Q2VQ34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aurora kinase C (Homo sapiens (Human)) | BDBM50154291 (CHEMBL3775181) | PDB NCI pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | <5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Russia; Mendeleyev University of Chemical Technology Curated by ChEMBL | Assay Description Inhibition of full length human N-terminal GST-HIS6-tagged Aurora C expressed in sf9 cells by flashplate based radiometric 33pan-quinase assay | Eur J Med Chem 112: 114-29 (2016) Article DOI: 10.1016/j.ejmech.2016.01.050 BindingDB Entry DOI: 10.7270/Q2VQ34K1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
MAP kinase-interacting serine/threonine-protein kinase 1 (Homo sapiens (Human)) | BDBM50154291 (CHEMBL3775181) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | <5.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Russia; Mendeleyev University of Chemical Technology Curated by ChEMBL | Assay Description Inhibition of human MKNK1 by flashplate based radiometric 33pan-quinase assay | Eur J Med Chem 112: 114-29 (2016) Article DOI: 10.1016/j.ejmech.2016.01.050 BindingDB Entry DOI: 10.7270/Q2VQ34K1 | |||||||||||
More data for this Ligand-Target Pair |