Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Follicle-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50173578 (CHEMBL3263694) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | <100 | n/a | n/a | n/a | n/a |
Therachem Research Medilab (India) Pvt. Ltd. Curated by ChEMBL | Assay Description Positive allosteric modulation of FSHR (unknown origin) expressed in CHO cells assessed as FSH-induced cAMP accumulation incubated for 1 hr by HTRF a... | ACS Med Chem Lett 7: 345-7 (2016) Article DOI: 10.1021/acsmedchemlett.6b00082 BindingDB Entry DOI: 10.7270/Q2HQ41T6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Follicle-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50012105 (CHEMBL3263667) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a |
Therachem Research Medilab (India) Pvt. Ltd. Curated by ChEMBL | Assay Description Positive allosteric modulation of human FSHR expressed in rat granulocytes assessed as FSH-induced estradiol production after 72 hrs by radioimmunoss... | ACS Med Chem Lett 7: 345-7 (2016) Article DOI: 10.1021/acsmedchemlett.6b00082 BindingDB Entry DOI: 10.7270/Q2HQ41T6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Follicle-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50173579 (CHEMBL3809148) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a |
Therachem Research Medilab (India) Pvt. Ltd. Curated by ChEMBL | Assay Description Positive allosteric modulation of human FSHR expressed in rat granulocytes assessed as FSH-induced estradiol production after 72 hrs by radioimmunoss... | ACS Med Chem Lett 7: 345-7 (2016) Article DOI: 10.1021/acsmedchemlett.6b00082 BindingDB Entry DOI: 10.7270/Q2HQ41T6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Follicle-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50173579 (CHEMBL3809148) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a |
Therachem Research Medilab (India) Pvt. Ltd. Curated by ChEMBL | Assay Description Positive allosteric modulation of FSHR (unknown origin) expressed in CHO cells assessed as FSH-induced cAMP accumulation incubated for 1 hr by HTRF a... | ACS Med Chem Lett 7: 345-7 (2016) Article DOI: 10.1021/acsmedchemlett.6b00082 BindingDB Entry DOI: 10.7270/Q2HQ41T6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Follicle-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50012120 (CHEMBL3263691) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a |
Therachem Research Medilab (India) Pvt. Ltd. Curated by ChEMBL | Assay Description Positive allosteric modulation of human FSHR expressed in rat granulocytes assessed as FSH-induced estradiol production after 72 hrs by radioimmunoss... | ACS Med Chem Lett 7: 345-7 (2016) Article DOI: 10.1021/acsmedchemlett.6b00082 BindingDB Entry DOI: 10.7270/Q2HQ41T6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Follicle-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50173581 (CHEMBL3809644) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | <100 | n/a | n/a | n/a | n/a |
Therachem Research Medilab (India) Pvt. Ltd. Curated by ChEMBL | Assay Description Positive allosteric modulation of FSHR (unknown origin) expressed in CHO cells assessed as FSH-induced cAMP accumulation incubated for 1 hr by HTRF a... | ACS Med Chem Lett 7: 345-7 (2016) Article DOI: 10.1021/acsmedchemlett.6b00082 BindingDB Entry DOI: 10.7270/Q2HQ41T6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Follicle-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50173580 (CHEMBL3808949) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | <100 | n/a | n/a | n/a | n/a |
Therachem Research Medilab (India) Pvt. Ltd. Curated by ChEMBL | Assay Description Positive allosteric modulation of FSHR (unknown origin) expressed in CHO cells assessed as FSH-induced cAMP accumulation incubated for 1 hr by HTRF a... | ACS Med Chem Lett 7: 345-7 (2016) Article DOI: 10.1021/acsmedchemlett.6b00082 BindingDB Entry DOI: 10.7270/Q2HQ41T6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Follicle-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50173578 (CHEMBL3263694) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a |
Therachem Research Medilab (India) Pvt. Ltd. Curated by ChEMBL | Assay Description Positive allosteric modulation of human FSHR expressed in rat granulocytes assessed as FSH-induced estradiol production after 72 hrs by radioimmunoss... | ACS Med Chem Lett 7: 345-7 (2016) Article DOI: 10.1021/acsmedchemlett.6b00082 BindingDB Entry DOI: 10.7270/Q2HQ41T6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Follicle-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50012120 (CHEMBL3263691) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | <100 | n/a | n/a | n/a | n/a |
Therachem Research Medilab (India) Pvt. Ltd. Curated by ChEMBL | Assay Description Positive allosteric modulation of FSHR (unknown origin) expressed in CHO cells assessed as FSH-induced cAMP accumulation incubated for 1 hr by HTRF a... | ACS Med Chem Lett 7: 345-7 (2016) Article DOI: 10.1021/acsmedchemlett.6b00082 BindingDB Entry DOI: 10.7270/Q2HQ41T6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Follicle-stimulating hormone receptor (Homo sapiens (Human)) | BDBM50012105 (CHEMBL3263667) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | <100 | n/a | n/a | n/a | n/a |
Therachem Research Medilab (India) Pvt. Ltd. Curated by ChEMBL | Assay Description Positive allosteric modulation of FSHR (unknown origin) expressed in CHO cells assessed as FSH-induced cAMP accumulation incubated for 1 hr by HTRF a... | ACS Med Chem Lett 7: 345-7 (2016) Article DOI: 10.1021/acsmedchemlett.6b00082 BindingDB Entry DOI: 10.7270/Q2HQ41T6 | |||||||||||
More data for this Ligand-Target Pair |