Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50463323 (CHEMBL4247814) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.27E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Siberian Branch of the Russian Academy of Sciences Curated by ChEMBL | Assay Description Inhibition of recombinant human DPP4 using H-Gly-Pro-AMC as substrate measured after 10 mins | Bioorg Med Chem 26: 4402-4409 (2018) Article DOI: 10.1016/j.bmc.2018.07.018 BindingDB Entry DOI: 10.7270/Q2RV0RBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50463326 (CHEMBL4242321) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.78E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Siberian Branch of the Russian Academy of Sciences Curated by ChEMBL | Assay Description Inhibition of recombinant human DPP4 using H-Gly-Pro-AMC as substrate measured after 10 mins | Bioorg Med Chem 26: 4402-4409 (2018) Article DOI: 10.1016/j.bmc.2018.07.018 BindingDB Entry DOI: 10.7270/Q2RV0RBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50463324 (CHEMBL4238607) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.58E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Siberian Branch of the Russian Academy of Sciences Curated by ChEMBL | Assay Description Inhibition of recombinant human DPP4 using H-Gly-Pro-AMC as substrate measured after 10 mins | Bioorg Med Chem 26: 4402-4409 (2018) Article DOI: 10.1016/j.bmc.2018.07.018 BindingDB Entry DOI: 10.7270/Q2RV0RBN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50463325 (CHEMBL4238169) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.58E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Siberian Branch of the Russian Academy of Sciences Curated by ChEMBL | Assay Description Inhibition of recombinant human DPP4 using H-Gly-Pro-AMC as substrate measured after 10 mins | Bioorg Med Chem 26: 4402-4409 (2018) Article DOI: 10.1016/j.bmc.2018.07.018 BindingDB Entry DOI: 10.7270/Q2RV0RBN | |||||||||||
More data for this Ligand-Target Pair |