Affinity Data by BDB articleid=50029164

Articleid 50029164

Found 4 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
D(2) dopamine receptor (Rattus norvegicus (rat))	BDBM50001888 ((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...) Show SMILES CN(C)CCCN1c2ccccc2Sc2ccc(Cl)cc12 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	Article	50	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Tested for Competitive binding inhibition of [3H]-Spiperone to Dopamine receptor D2 in rat striatal membrane.				Bioorg Med Chem Lett 3: 1241-1244 (1993) Article DOI: 10.1016/S0960-894X(00)80323-6 BindingDB Entry DOI: 10.7270/Q26W9B00
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
D(2) dopamine receptor (Rattus norvegicus (rat))	BDBM50281901 (CHEMBL21564 \| MethanesulfonateN-[3-(2-chloro-pheno...) Show SMILES C[N+](C)(N)CCCN1c2ccccc2Sc2ccc(Cl)cc12 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article	820	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Tested for Competitive binding inhibition of [3H]-Spiperone to Dopamine receptor D2 in rat striatal membrane.				Bioorg Med Chem Lett 3: 1241-1244 (1993) Article DOI: 10.1016/S0960-894X(00)80323-6 BindingDB Entry DOI: 10.7270/Q26W9B00
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
D(2) dopamine receptor (Rattus norvegicus (rat))	BDBM50281900 (CHEMBL21398 \| N'-[2-(2-Chloro-phenothiazin-10-yl)-...) Show SMILES C[N+](C)(C)NCCN1c2ccccc2Sc2ccc(Cl)cc12 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article	4.88E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Tested for Competitive binding inhibition of [3H]-Spiperone to Dopamine receptor D2 in rat striatal membrane.				Bioorg Med Chem Lett 3: 1241-1244 (1993) Article DOI: 10.1016/S0960-894X(00)80323-6 BindingDB Entry DOI: 10.7270/Q26W9B00
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
D(2) dopamine receptor (Rattus norvegicus (rat))	BDBM50019879 (CHEMBL279905 \| [3-(2-Chloro-phenothiazin-10-yl)-pr...) Show SMILES C[N+](C)(C)CCCN1c2ccccc2Sc2ccc(Cl)cc12 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article	8.57E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Tested for Competitive binding inhibition of [3H]-Spiperone to Dopamine receptor D2 in rat striatal membrane.				Bioorg Med Chem Lett 3: 1241-1244 (1993) Article DOI: 10.1016/S0960-894X(00)80323-6 BindingDB Entry DOI: 10.7270/Q26W9B00
TBA Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%