Found 5 hits of Enzyme Inhibition Constant Data Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Protein tyrosine phosphatase receptor type C-associated protein
(Homo sapiens (Human)) | BDBM50083572
((S)-1,2-Dimethoxy-5,6,6a,7-tetrahydro-4H-dibenzo[d...)Show InChI InChI=1S/C18H19NO2/c1-20-15-10-12-7-8-19-14-9-11-5-3-4-6-13(11)17(16(12)14)18(15)21-2/h3-6,10,14,19H,7-9H2,1-2H3/t14-/m0/s1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL PC cid PC sid UniChem
Similars
| Article
| n/a | n/a | 5.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description In vitro inhibitory activity against recombinant CD45 protein tyrosine phosphatase |
Bioorg Med Chem Lett 5: 1519-1522 (1995)
Article DOI: 10.1016/0960-894X(95)00250-W BindingDB Entry DOI: 10.7270/Q2V69K2S |
More data for this Ligand-Target Pair | |
Protein tyrosine phosphatase receptor type C-associated protein
(Homo sapiens (Human)) | BDBM50202322
((-)-anonaine | (R)-6,7,7a,8-tetrahydro-5H-benzo[g]...)Show InChI InChI=1S/C17H15NO2/c1-2-4-12-10(3-1)7-13-15-11(5-6-18-13)8-14-17(16(12)15)20-9-19-14/h1-4,8,13,18H,5-7,9H2/t13-/m1/s1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Similars
| Article
| n/a | n/a | 1.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description In vitro inhibitory activity against recombinant CD45 protein tyrosine phosphatase |
Bioorg Med Chem Lett 5: 1519-1522 (1995)
Article DOI: 10.1016/0960-894X(95)00250-W BindingDB Entry DOI: 10.7270/Q2V69K2S |
More data for this Ligand-Target Pair | |
Protein tyrosine phosphatase receptor type C-associated protein
(Homo sapiens (Human)) | BDBM50197829
((S)-1,2,9,10-tetramethoxy-6-methyl-5,6,6a,7-tetrah...)Show SMILES COc1cc2C[C@@H]3N(C)CCc4cc(OC)c(OC)c(-c2cc1OC)c34 |r| Show InChI InChI=1S/C21H25NO4/c1-22-7-6-12-9-18(25-4)21(26-5)20-14-11-17(24-3)16(23-2)10-13(14)8-15(22)19(12)20/h9-11,15H,6-8H2,1-5H3/t15-/m0/s1 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid PDB UniChem
Patents
Similars
| Article
| n/a | n/a | 8.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description In vitro inhibitory activity against recombinant CD45 protein tyrosine phosphatase |
Bioorg Med Chem Lett 5: 1519-1522 (1995)
Article DOI: 10.1016/0960-894X(95)00250-W BindingDB Entry DOI: 10.7270/Q2V69K2S |
More data for this Ligand-Target Pair | |
Protein tyrosine phosphatase receptor type C-associated protein
(Homo sapiens (Human)) | BDBM50284797
(7-Methyl-6,7,7a,8-tetrahydro-5H-benzo[g][1,3]dioxo...)Show InChI InChI=1S/C18H17NO2/c1-19-7-6-12-9-15-18(21-10-20-15)17-13-5-3-2-4-11(13)8-14(19)16(12)17/h2-5,9,14H,6-8,10H2,1H3 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| Article
| n/a | n/a | 1.07E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description In vitro inhibitory activity against recombinant CD45 protein tyrosine phosphatase |
Bioorg Med Chem Lett 5: 1519-1522 (1995)
Article DOI: 10.1016/0960-894X(95)00250-W BindingDB Entry DOI: 10.7270/Q2V69K2S |
More data for this Ligand-Target Pair | |
Protein tyrosine phosphatase receptor type C-associated protein
(Homo sapiens (Human)) | BDBM50202301
(CHEMBL37736 | Liriodenine | hiriodenine)Show InChI InChI=1S/C17H9NO3/c19-16-11-4-2-1-3-10(11)14-13-9(5-6-18-15(13)16)7-12-17(14)21-8-20-12/h1-7H,8H2 | KEGG
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
CHEMBL MCE KEGG PC cid PC sid UniChem
Patents
Similars
| Article
| n/a | n/a | 1.82E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA
Curated by ChEMBL
| Assay Description In vitro inhibitory activity against recombinant CD45 protein tyrosine phosphatase |
Bioorg Med Chem Lett 5: 1519-1522 (1995)
Article DOI: 10.1016/0960-894X(95)00250-W BindingDB Entry DOI: 10.7270/Q2V69K2S |
More data for this Ligand-Target Pair | |