Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
B2 bradykinin receptor (Cavia porcellus) | BDBM50403371 (Firazyr | HOE-140 | ICATIBANT) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.0900 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50403371 (Firazyr | HOE-140 | ICATIBANT) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.0900 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067263 (5-{2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.360 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067263 (5-{2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.360 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067242 (3-(6-Acetylamino-pyridin-3-yl)-N-({[3-(3-bromo-2-m...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.380 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067242 (3-(6-Acetylamino-pyridin-3-yl)-N-({[3-(3-bromo-2-m...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.380 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067248 (5-{2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.440 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067247 (4-{(E)-2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyr...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067247 (4-{(E)-2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyr...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067253 ((E)-3-(4-Acetylamino-phenyl)-N-({[3-(3-bromo-2-met...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.550 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067240 ((E)-N-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.590 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067240 ((E)-N-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.590 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067251 (4-{(E)-2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyr...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.660 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067257 (3-[3-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.760 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067264 ((Z)-N-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.780 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067235 (3-[3-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.790 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067235 (3-[3-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.790 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067233 (2-[3-(3-Acetyl-phenyl)-ureido]-N-[3-(3-bromo-2-met...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.790 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067258 ((E)-N-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.890 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067236 ((E)-3-[4-(Acetyl-methyl-amino)-phenyl]-N-({[3-(3-b...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067251 (4-{(E)-2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyr...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067239 (CHEMBL555556 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067260 (CHEMBL130452 | N-({[3-(3-Bromo-2-methyl-imidazo[1,...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067256 (CHEMBL559195 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067239 (CHEMBL555556 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067253 ((E)-3-(4-Acetylamino-phenyl)-N-({[3-(3-bromo-2-met...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067238 (3-[3-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067238 (3-[3-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067245 (CHEMBL542473 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50062860 (CHEMBL132620 | N-({[3-(3-Bromo-2-methyl-imidazo[1,...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50062860 (CHEMBL132620 | N-({[3-(3-Bromo-2-methyl-imidazo[1,...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067258 ((E)-N-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067241 (CHEMBL543188 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067246 (CHEMBL130660 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067241 (CHEMBL543188 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067248 (5-{2-[({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067261 (CHEMBL556816 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067261 (CHEMBL556816 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067250 ((E)-N-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067259 (CHEMBL130196 | N-({[3-(3-Bromo-2-methyl-imidazo[1,...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067244 (CHEMBL545765 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067244 (CHEMBL545765 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067250 ((E)-N-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067249 (CHEMBL544600 | N-({[3-(3-Bromo-2-methyl-imidazo[1,...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067252 (CHEMBL338682 | Hexanoic acid ({[3-(3-bromo-2-methy...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50062878 (CHEMBL131517 | N-({[3-(3-Bromo-2-methyl-imidazo[1,...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50062878 (CHEMBL131517 | N-({[3-(3-Bromo-2-methyl-imidazo[1,...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067255 (CHEMBL130438 | N-({[3-(3-Bromo-2-methyl-imidazo[1,...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067255 (CHEMBL130438 | N-({[3-(3-Bromo-2-methyl-imidazo[1,...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50062864 (CHEMBL336116 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067243 (2-(3-Benzyl-ureido)-N-[3-(3-bromo-2-methyl-imidazo...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067243 (2-(3-Benzyl-ureido)-N-[3-(3-bromo-2-methyl-imidazo...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067265 (CHEMBL542472 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067266 (2-[3-(3-Amino-phenyl)-ureido]-N-[3-(3-bromo-2-meth...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067266 (2-[3-(3-Amino-phenyl)-ureido]-N-[3-(3-bromo-2-meth...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50062863 (2-Acetylamino-N-[3-(3-bromo-2-methyl-imidazo[1,2-a...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [ 3H]BK (0.06 nM) to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50% | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067236 ((E)-3-[4-(Acetyl-methyl-amino)-phenyl]-N-({[3-(3-b...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067257 (3-[3-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067233 (2-[3-(3-Acetyl-phenyl)-ureido]-N-[3-(3-bromo-2-met...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 61 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067254 (3-[3-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 63 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067254 (3-[3-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin-...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 63 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067246 (CHEMBL130660 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 75 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067237 (CHEMBL336209 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 83 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067264 ((Z)-N-({[3-(3-Bromo-2-methyl-imidazo[1,2-a]pyridin...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067256 (CHEMBL559195 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 150 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067237 (CHEMBL336209 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 150 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067245 (CHEMBL542473 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 200 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067252 (CHEMBL338682 | Hexanoic acid ({[3-(3-bromo-2-methy...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067265 (CHEMBL542472 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 260 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067234 (2-(3-Benzoyl-ureido)-N-[3-(3-bromo-2-methyl-imidaz...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 340 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Cavia porcellus) | BDBM50067234 (2-(3-Benzoyl-ureido)-N-[3-(3-bromo-2-methyl-imidaz...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 340 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 0.06 nM to Bradykinin receptor B2 in guinea pig ileum membrane preparations by 50%. | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067260 (CHEMBL130452 | N-({[3-(3-Bromo-2-methyl-imidazo[1,...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 350 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067259 (CHEMBL130196 | N-({[3-(3-Bromo-2-methyl-imidazo[1,...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 510 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50067249 (CHEMBL544600 | N-({[3-(3-Bromo-2-methyl-imidazo[1,...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 670 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50062864 (CHEMBL336116 | N-[3-(3-Bromo-2-methyl-imidazo[1,2-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
B2 bradykinin receptor (Homo sapiens (Human)) | BDBM50062863 (2-Acetylamino-N-[3-(3-bromo-2-methyl-imidazo[1,2-a...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Fujisawa Pharmaceutical Company, Ltd. Curated by ChEMBL | Assay Description Concentration required to inhibit specific binding of [3H]BK at 1.2 nM to A-431 cells (human epidermoidcarcinoma) which express Bradykinin receptor B... | J Med Chem 41: 4053-61 (1998) Article DOI: 10.1021/jm980214f BindingDB Entry DOI: 10.7270/Q2WQ04GV | |||||||||||
More data for this Ligand-Target Pair |