Reaction Details |
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Target | Transmembrane anterior posterior transformation protein 1 homolog |
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Ligand | BDBM575122 |
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Substrate/Competitor | n/a |
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Meas. Tech. | Assessing Antiviral Activity Against Human Cytomegalovirus (HCMV) |
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IC50 | 730±n/a nM |
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Citation | Remiszewski, S; Chiang, LW; Murphy, EA; Sun, Q; Kayser, F; Fink, SJ Broad spectrum antiviral compositions and methods US Patent US11459321 Publication Date 10/4/2022 |
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More Info.: | Get all data from this article, Assay Method |
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Transmembrane anterior posterior transformation protein 1 homolog |
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Name: | Transmembrane anterior posterior transformation protein 1 homolog |
Synonyms: | CMVFR | Cytomegalovirus partial fusion receptor | TAPT1 | TAPT1_HUMAN |
Type: | Protein |
Mol. Mass.: | 64270.48 |
Organism: | Human |
Description: | Q6NXT6 |
Residue: | 567 |
Sequence: | MAGVGDAAAPGEGGGGGVDGPQRDGRGEAEQPGGSGGQGPPPAPQLTETLGFYESDRRRE
RRRGRTELSLLRFLSAELTRGYFLEHNEAKYTERRERVYTCLRIPRELEKLMVFGIFLCL
DAFLYVFTLLPLRVFLALFRLLTLPCYGLRDRRLLQPAQVCDILKGVILVICYFMMHYVD
YSMMYHLIRGQSVIKLYIIYNMLEVADRLFSSFGQDILDALYWTATEPKERKRAHIGVIP
HFFMAVLYVFLHAILIMVQATTLNVAFNSHNKSLLTIMMSNNFVEIKGSVFKKFEKNNLF
QMSNSDIKERFTNYVLLLIVCLRNMEQFSWNPDHLWVLFPDVCMVIASEIAVDIVKHAFI
TKFNDITADVYSEYRASLAFDLVSSRQKNAYTDYSDSVARRMGFIPLPLAVLLIRVVTSS
IKVQGILSYACVILFYFGLISLKVLNSIVLLGKSCQYVKEAKMEEKLSNPPATCTPGKPS
SKSQNKCKPSQGLSTEENLSASITKQPIHQKENIIPLLVTSNSDQFLTTPDGDEKDITQD
NSELKHRSSKKDLLEIDRFTICGNRID
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BDBM575122 |
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n/a |
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Name | BDBM575122 |
Synonyms: | US11459321, Example 59 |
Type | Small organic molecule |
Emp. Form. | C29H34N4O2S |
Mol. Mass. | 502.671 |
SMILES | CN1CCCN(C1=O)c1ccc2CCN(Cc2c1)c1ncc(Cc2ccc(cc2)C2CCOCC2)s1 |
Structure |
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