| Reaction Details |
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 | Report a problem with these data |
| Target | PPAR delta protein |
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| Ligand | BDBM323604 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Luciferase Assay |
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| EC50 | 1757±n/a nM |
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| Citation |  Downes, M; Evans, R; Kluge, A; Lagu, B; Miura, M; Panigrahi, SK; Patane, M; Samajdar, S; Senaiar, R; Takahashi, T PPAR agonists, compounds, pharmaceutical compositions, and methods of use thereof US Patent US10188627 Publication Date 1/29/2019 |
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| More Info.: | Get all data from this article, Assay Method |
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| PPAR delta protein |
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| Name: | PPAR delta protein |
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| Synonyms: | PPAR delta |
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| Type: | n/a |
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| Mol. Mass.: | 49664.60 |
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| Organism: | Rattus norvegicus (Rat) |
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| Description: | Q62879 |
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| Residue: | 440 |
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| Sequence: | MEQPQEETPEAREEEKEEVATGDGAPELNGGPEHTLPSSSCTDLSQNSSPSSLLDQLQMG
CDGASGGSLNMECRVCGDKASGFHYGVHACEGCKGFFRRTIRMKLKYEKCDRICKIQKKN
RNKCQYCRFQKCLALGMSHNAIRFGRMPEAEKRKLVAGLTASEGCQQNPQLADLKAFSKH
IYNAYLKNFNMTKKKARSILTGKSSHNAPFIIHDIETLWQAEKGLVWKQLVNGPPPYNEI
SVHVFYRCQSTTVETVRELTEFAKNIPNFSSLFLNDQVTLLKYGVHEAIFAMLASIVNKD
GLLVANGSGFVTHEFLRSIRKPFSDIIEPKFEFAVKFNALELVDSDLALFIAAIILCGDR
PGLMNVPQVEAIQDTILQALEFHLQVNHPDSQYLFPKLLQKMADLRQLVTEHAQMMQWLK
KTESETLLHPLLQEIYKDMY
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| BDBM323604 |
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| n/a |
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| Name | BDBM323604 |
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| Synonyms: | 3-(3-((2-((4-(furan-2-yl)-N-methylbenzamido)methyl)phenoxy) methyl)phenyl)propanoic acid | US10188627, Compound 8p |
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| Type | Small organic molecule |
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| Emp. Form. | C29H27NO5 |
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| Mol. Mass. | 469.5284 |
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| SMILES | CN(Cc1ccccc1OCc1cccc(CCC(O)=O)c1)C(=O)c1ccc(cc1)-c1ccco1 |
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| Structure | 
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