Reaction Details |
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Target | Thyroid hormone receptor beta [209-461] |
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Ligand | BDBM18833 |
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Substrate/Competitor | Peptide SRC2-2 |
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Meas. Tech. | Fluorescence Polarization (FP) Competition Assay |
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IC50 | 100000±n/a nM |
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Citation | Arnold, LA; Kosinski, A; Estebanez-Perpina, E; Fletterick, RJ; Guy, RK Inhibitors of the Interaction of a Thyroid Hormone Receptor and Coactivators: Preliminary Structure-Activity Relationships. J Med Chem50:5269-5280 (2007) [PubMed] Article |
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More Info.: | Get all data from this article, Solution Info, Assay Method |
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Thyroid hormone receptor beta [209-461] |
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Name: | Thyroid hormone receptor beta [209-461] |
Synonyms: | ERBA2 | NR1A2 | THB_HUMAN | THR1 | THRB | Thyroid Hormone Receptor (TR-beta) |
Type: | Ligand-Binding Domain |
Mol. Mass.: | 28584.77 |
Organism: | Homo sapiens (Human) |
Description: | The hTRbeta LBD (His6 T209-D461) was cloned and expressed in E. coli. |
Residue: | 253 |
Sequence: | THKPEPTDEEWELIKTVTEAHVATNAQGSHWKQKRKFLPEDIGQAPIVNAPEGGKVDLEA
FSHFTKIITPAITRVVDFAKKLPMFCELPCEDQIILLKGCCMEIMSLRAAVRYDPESETL
TLNGEMAVTRGQLKNGGLGVVSDAIFDLGMSLSSFNLDDTEVALLQAVLLMSSDRPGLAC
VERIEKYQDSFLLAFEHYINYRKHHVTHFWPKLLMKVTDLRMIGACHASRFLHMKVECPT
ELFPPLFLEVFED
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BDBM18833 |
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Peptide SRC2-2 |
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Name: | Peptide SRC2-2 |
Synonyms: | n/a |
Type: | Peptide |
Mol. Mass.: | 2334.76 |
Organism: | n/a |
Description: | The peptide is labeled with 5-iodoacetamidofluorescien. |
Residue: | 20 |
Sequence: | |