| Reaction Details |
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 | Report a problem with these data |
| Target | Estrogen receptor |
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| Ligand | BDBM40151 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | Estrogen Receptor-alpha Coactivator Binding Inhibitors Dose Response Confirmation |
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| IC50 | 7851.33±n/a nM |
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| Citation |  PubChem, PC Estrogen Receptor-alpha Coactivator Binding Inhibitors Dose Response Confirmation PubChem Bioassay(2007)[AID] |
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| More Info.: | Get all data from this article, Solution Info, Assay Method |
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| Estrogen receptor |
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| Name: | Estrogen receptor |
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| Synonyms: | ER | ER-alpha | ESR | ESR1 | ESR1_HUMAN | Estradiol receptor | Estrogen receptor | Estrogen receptor (ER alpha) | Estrogen receptor (ER-alpha) | Estrogen receptor alpha (ER alpha) | Estrogen receptor alpha (ER) | NR3A1 | Nuclear receptor subfamily 3 group A member 1 |
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| Type: | Protein |
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| Mol. Mass.: | 66230.44 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P03372 |
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| Residue: | 595 |
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| Sequence: | MTMTLHTKASGMALLHQIQGNELEPLNRPQLKIPLERPLGEVYLDSSKPAVYNYPEGAAY
EFNAAAAANAQVYGQTGLPYGPGSEAAAFGSNGLGGFPPLNSVSPSPLMLLHPPPQLSPF
LQPHGQQVPYYLENEPSGYTVREAGPPAFYRPNSDNRRQGGRERLASTNDKGSMAMESAK
ETRYCAVCNDYASGYHYGVWSCEGCKAFFKRSIQGHNDYMCPATNQCTIDKNRRKSCQAC
RLRKCYEVGMMKGGIRKDRRGGRMLKHKRQRDDGEGRGEVGSAGDMRAANLWPSPLMIKR
SKKNSLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINW
AKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEG
MVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLD
KITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLYDLL
LEMLDAHRLHAPTSRGGASVEETDQSHLATAGSTSSHSLQKYYITGEAEGFPATV
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| BDBM40151 |
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| n/a |
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| Name | BDBM40151 |
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| Synonyms: | 8-Methoxy-3-(7-methyl-imidazo[1,2-a]pyridin-2-yl)-chromen-2-one | 8-methoxy-3-(7-methyl-2-imidazo[1,2-a]pyridinyl)-1-benzopyran-2-one | 8-methoxy-3-(7-methylimidazo[1,2-a]pyridin-2-yl)chromen-2-one | 8-methoxy-3-(7-methylimidazo[1,2-a]pyridin-2-yl)coumarin | MLS000526145 | SMR000116619 | cid_767326 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H14N2O3 |
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| Mol. Mass. | 306.3154 |
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| SMILES | COc1cccc2cc(-c3cn4ccc(C)cc4n3)c(=O)oc12 |
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| Structure | 
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