| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Estrogen receptor beta |
|---|
| Ligand | BDBM40941 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Estrogen Receptor-beta Coactivator Binding Inhibitors ELISA Secondary Assay |
|---|
| IC50 | 23±n/a nM |
|---|
| Citation |  PubChem, PC Estrogen Receptor-beta Coactivator Binding Inhibitors ELISA Secondary Assay PubChem Bioassay(2008)[AID] |
|---|
| More Info.: | Get all data from this article, Solution Info, Assay Method |
|---|
| |
| Estrogen receptor beta |
|---|
| Name: | Estrogen receptor beta |
|---|
| Synonyms: | ER-beta | ESR2 | ESR2_HUMAN | ESTRB | Estradiol receptor beta (ERβ) | Estrogen receptor | Estrogen receptor (ER beta) | Estrogen receptor beta | Estrogen receptor beta (ER beta) | Estrogen receptor beta (ER) | NR3A2 | Nuclear receptor subfamily 3 group A member 2 | estrogen beta |
|---|
| Type: | Protein |
|---|
| Mol. Mass.: | 59238.43 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | Q92731 |
|---|
| Residue: | 530 |
|---|
| Sequence: | MDIKNSPSSLNSPSSYNCSQSILPLEHGSIYIPSSYVDSHHEYPAMTFYSPAVMNYSIPS
NVTNLEGGPGRQTTSPNVLWPTPGHLSPLVVHRQLSHLYAEPQKSPWCEARSLEHTLPVN
RETLKRKVSGNRCASPVTGPGSKRDAHFCAVCSDYASGYHYGVWSCEGCKAFFKRSIQGH
NDYICPATNQCTIDKNRRKSCQACRLRKCYEVGMVKCGSRRERCGYRLVRRQRSADEQLH
CAGKAKRSGGHAPRVRELLLDALSPEQLVLTLLEAEPPHVLISRPSAPFTEASMMMSLTK
LADKELVHMISWAKKIPGFVELSLFDQVRLLESCWMEVLMMGLMWRSIDHPGKLIFAPDL
VLDRDEGKCVEGILEIFDMLLATTSRFRELKLQHKEYLCVKAMILLNSSMYPLVTATQDA
DSSRKLAHLLNAVTDALVWVIAKSGISSQQQSMRLANLLMLLSHVRHASNKGMEHLLNMK
CKNVVPVYDLLLEMLNAHVLRGCKSSITGSECSPAEDSKSKEGSQNPQSQ
|
|
|
|---|
| BDBM40941 |
|---|
| n/a |
|---|
| Name | BDBM40941 |
|---|
| Synonyms: | (4-Morpholin-4-yl-phenyl)-(6-o-tolyl-pyridazin-3-yl)-amine | (4-morpholinophenyl)-[6-(o-tolyl)pyridazin-3-yl]amine | 6-(2-methylphenyl)-N-(4-morpholin-4-ylphenyl)pyridazin-3-amine | 6-(2-methylphenyl)-N-[4-(4-morpholinyl)phenyl]-3-pyridazinamine | MLS000076246 | SMR000007231 | cid_646977 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C21H22N4O |
|---|
| Mol. Mass. | 346.4256 |
|---|
| SMILES | Cc1ccccc1-c1ccc(Nc2ccc(cc2)N2CCOCC2)nn1 |
|---|
| Structure | 
|
|---|
Search and Browse
