| Reaction Details |
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 | Report a problem with these data |
| Target | kappa-type opioid receptor isoform 1 |
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| Ligand | BDBM81936 |
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| Substrate/Competitor | n/a |
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| Ki | >10000±n/a nM |
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| Comments | PDSP_7134 |
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| Citation |  Benyhe, S; Varga, E; Hepp, J; Magyar, A; Borsodi, A; Wollemann, M Characterization of kappa 1 and kappa 2 opioid binding sites in frog (Rana esculenta) brain membrane preparation. Neurochem Res15:899-904 (1990) [PubMed] Article |
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| More Info.: | Get all data from this article |
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| kappa-type opioid receptor isoform 1 |
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| Name: | kappa-type opioid receptor isoform 1 |
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| Synonyms: | OPIATE Kappa | OPRK1 | Opioid receptor kappa 1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 44032.90 |
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| Organism: | Frog |
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| Description: | F7A0F2 |
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| Residue: | 392 |
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| Sequence: | MVMESPVQIFREEEAIIPERAPVGSTCSSSCAPACPSSCFPNTSWLLGWDDHDNVSAYPD
LPLNEGNHTSISPTISVIITAVYSMVFVVGLVGNALVMFVIIRYTKMKTATNIYIFNLAL
ADALVTTTMPFQSTSFLMNSWPFGDVLCKIVVSIDYYNMFTSIFTLTMMSVDRYIAVCHP
VKALDFRTPLKAKCINICIWMLSSSVGISAIVLGGTKISDGSTECALQFPTHYWYWDTVM
KMCVFIFAFIIPVFIITICYTLMILRLKSVRLLSGSREKDRNLRRITRLVLVVVAVFIVC
WTPIHIFVLVEALVDVPQSIAVVSIYYFCIALGYTNSSLNPILYAFLDENFKRCFKDFCF
PSKHRLDRQPNSRVGNTVQDPACNRHGSQKPV
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| BDBM81936 |
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| n/a |
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| Name | BDBM81936 |
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| Synonyms: | CAS_111728-01-9 | NSC_122115 | PD117302 |
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| Type | Small organic molecule |
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| Emp. Form. | C21H28N2OS |
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| Mol. Mass. | 356.525 |
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| SMILES | CN(C1CCCCC1N1CCCC1)C(=O)Cc1cccc2sccc12 |
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| Structure | 
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