| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Mu-type opioid receptor |
|---|
| Ligand | BDBM50018634 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEBML_147107 |
|---|
| IC50 | 16800±n/a nM |
|---|
| Citation |  Schiller, PW; Nguyen, TM; Maziak, LA; Wilkes, BC; Lemieux, C Structure-activity relationships of cyclic opioid peptide analogues containing a phenylalanine residue in the 3-position. J Med Chem30:2094-9 (1987) [PubMed] |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Mu-type opioid receptor |
|---|
| Name: | Mu-type opioid receptor |
|---|
| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 11165.58 |
|---|
| Organism: | GUINEA PIG |
|---|
| Description: | P97266 |
|---|
| Residue: | 98 |
|---|
| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
|
|
|
|---|
| BDBM50018634 |
|---|
| n/a |
|---|
| Name | BDBM50018634 |
|---|
| Synonyms: | 12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-2-benzyl-3,7,13-trioxo-1,4,8triaza-cyclotridecane-5-carboxylic acid amide | CHEMBL64949 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C27H34N6O6 |
|---|
| Mol. Mass. | 538.5955 |
|---|
| SMILES | N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@H]1CCCNC(=O)C[C@H](NC(=O)[C@H](Cc2ccccc2)NC1=O)C(N)=O |
|---|
| Structure | 
|
|---|
Search and Browse
